日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

QSAR-Guided and Fragment-Based Drug Design of Monoterpenoid Inhibitors Targeting Ebola Virus Glycoprotein

基于QSAR指导和片段的单萜类抑制剂靶向埃博拉病毒糖蛋白的药物设计

Ait Lahcen, Nouhaila; Liman, Wissal; Zekri, Saad; Ait Lahcen, Adnane; Alanazi, Ashwag S; Alanazi, Mohammed M; Delaite, Christelle; Maatallah, Mohamed; Cherqaoui, Driss

Bioactive oxadiazolo-benzodiazepines: synthesis, α amylase inhibition, antioxidant activity, molecular docking and DFT calculation

生物活性恶二唑并苯二氮卓类化合物:合成、α-淀粉酶抑制、抗氧化活性、分子对接和DFT计算

Ait Lahcen, Marouane; El Karfi, Wissal; Ait Lahcen, Nouhaila; Fadili, Driss; Hmaimou, Samir; Adardour, Mohamed; Hdoufane, Ismail; Zaballos-García, Elena; Faouzi, My El Abbes; Maatallah, Mohamed; Cherqaoui, Driss; Baouid, Abdesselam

Identification of potent TMPRSS4 inhibitors through structural modeling and molecular dynamics simulations.

通过结构建模和分子动力学模拟鉴定有效的TMPRSS4抑制剂

Hdoufane Ismail, Oubahmane Mehdi, Habibi Youssef, Delaite Christelle, Alanazi Mohammed M, Cherqaoui Driss

A longitudinal study of the effects of risk perception and response efficacy on adaptation of elderly individuals and individuals with chronic health conditions to heat waves

一项纵向研究,旨在探讨风险感知和应对效能对老年人和慢性病患者适应热浪的影响

Mehiriz, Kaddour; Cherqaoui, Sara

Degradation behavior of austenite, ferrite, and martensite present in biodegradable Fe-based alloys in three protein-rich pseudo-physiological solutions

在三种富含蛋白质的拟生理溶液中,可生物降解的铁基合金中奥氏体、铁素体和马氏体的降解行为

Cherqaoui, Abdelhakim; Cao, Quang Nguyen; Gatto, Maria Laura; Paternoster, Carlo; Mengucci, Paolo; Mantovani, Diego

TGFβ signaling pathway is altered by HLA-B27 expression, resulting in pathogenic consequences relevant for spondyloarthritis

TGFβ 信号通路因 HLA-B27 表达而改变,导致与脊柱关节炎相关的致病后果

Marc Lauraine, Maxence de Taffin de Tilques, Dganit Melamed-Kadosh, Bilade Cherqaoui, Vincent Rincheval, Erwan Prevost, Aurore Rincheval-Arnold, Eneida Cela, Arie Admon, Isabelle Guénal, Luiza M Araujo, Maxime Breban

Computational design of potent dimeric phenylthiazole NS5A inhibitors for hepatitis C virus

利用计算机设计高效二聚苯基噻唑NS5A抑制剂治疗丙型肝炎病毒感染

Liman, Wissal; Oubahmane, Mehdi; Lahcen, Nouhaila Ait; Hdoufane, Ismail; Cherqaoui, Driss; Daoud, Rachid; El Allali, Achraf

STAT1 deficiency underlies a proinflammatory imprint of naive CD4(+) T cells in spondyloarthritis

STAT1 缺陷是强直性脊柱炎中初始 CD4(+) T 细胞促炎特征的基础

Cherqaoui, Bilade; Crémazy, Frédéric; Lauraine, Marc; Shammas, Ghazal; Said-Nahal, Roula; Mambu Mambueni, Hendrick; Costantino, Félicie; Fourmont, Marine; Hulot, Audrey; Garchon, Henri-Jean; Glatigny, Simon; Araujo, Luiza M; Breban, Maxime

Interleukin 27 is a novel cytokine with anti-inflammatory effects against spondyloarthritis through the suppression of Th17 responses

白细胞介素 27 是一种新型细胞因子,通过抑制 Th17 反应发挥抗炎作用,对抗脊柱关节炎

Quentin Jouhault, Bilade Cherqaoui, Aude Jobart-Malfait, Simon Glatigny, Marc Lauraine, Audrey Hulot, Guillaume Morelle, Benjamin Hagege, Kétia Ermoza, Ahmed El Marjou, Brigitte Izac, Benjamin Saintpierre, Franck Letourneur, Séverine Rémy, Ignacio Anegon, Marie-Christophe Boissier, Gilles Chiocchia,

Design of Potent Inhibitors Targeting the Main Protease of SARS-CoV-2 Using QSAR Modeling, Molecular Docking, and Molecular Dynamics Simulations

利用QSAR建模、分子对接和分子动力学模拟设计靶向SARS-CoV-2主要蛋白酶的高效抑制剂

Oubahmane, Mehdi; Hdoufane, Ismail; Delaite, Christelle; Sayede, Adlane; Cherqaoui, Driss; El Allali, Achraf