日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Expanding the toolbox to develop IAP-based degraders of TEAD transcription factors.

扩展工具箱,开发基于 IAP 的 TEAD 转录因子降解剂。

Gupta Nishma, Trainor Nicole, Radwan Mona, Nguyen Stephanie, Duncan Luke, Tang Andrew X, Beveridge Julia, Silke Natasha, Yousef Jumana, Bilgilier Ceren, Wachter Johannes, Greb Peter, Jandova Zuzana, Eliaš Ján, Kopf Sara, Gerstberger Thomas, Stolt-Bergner Peggy, Braun Nina, Weinstabl Harald, McConnell Darryl B, Mauri Federico, Lucet Isabelle S, Silke John, Chessum Nicola E A, Roy Michael J

Determination of Ligand-Binding Affinity (K(d)) Using Transverse Relaxation Rate (R(2)) in the Ligand-Observed (1)H NMR Experiment and Applications to Fragment-Based Drug Discovery

利用配体观测的(1)H NMR实验中的横向弛豫速率(R(2))测定配体结合亲和力(K(d))及其在基于片段的药物发现中的应用

Liu, Manjuan; Mirza, Amin; McAndrew, P Craig; Thapaliya, Arjun; Pierrat, Olivier A; Stubbs, Mark; Hahner, Tamas; Chessum, Nicola E A; Innocenti, Paolo; Caldwell, John; Cheeseman, Matthew D; Bellenie, Benjamin R; van Montfort, Rob L M; Newton, Gary K; Burke, Rosemary; Collins, Ian; Hoelder, Swen

HSF1 Pathway Inhibitor Clinical Candidate (CCT361814/NXP800) Developed from a Phenotypic Screen as a Potential Treatment for Refractory Ovarian Cancer and Other Malignancies

HSF1通路抑制剂临床候选药物(CCT361814/NXP800)基于表型筛选开发,有望用于治疗难治性卵巢癌和其他恶性肿瘤。

Pasqua, A Elisa; Sharp, Swee Y; Chessum, Nicola E A; Hayes, Angela; Pellegrino, Loredana; Tucker, Michael J; Miah, Asadh; Wilding, Birgit; Evans, Lindsay E; Rye, Carl S; Mok, N Yi; Liu, Manjuan; Henley, Alan T; Gowan, Sharon; De Billy, Emmanuel; Te Poele, Robert; Powers, Marissa; Eccles, Suzanne A; Clarke, Paul A; Raynaud, Florence I; Workman, Paul; Jones, Keith; Cheeseman, Matthew D

A Comprehensive Chemical and Nutritional Analysis of New Zealand Yacon Concentrate

新西兰雪莲果浓缩物的综合化学和营养分析

Chessum, Keegan; Chen, Tony; Kam, Rothman; Yan, Mary

Biomarkers of coagulation, endothelial function, and fibrinolysis in critically ill patients with COVID-19: A single-center prospective longitudinal study

新冠肺炎危重患者凝血、内皮功能及纤溶生物标志物:一项单中心前瞻性纵向研究

Ganeem K Juneja, Matthew Castelo, Calvin H Yeh, Samantha E Cerroni, Bettina E Hansen, James E Chessum, Joel Abraham, Erblin Cani, Dhruva J Dwivedi, Douglas D Fraser, Marat Slessarev, Claudio Martin, Scott McGilvray, Peter L Gross, Patricia C Liaw, Jeffrey I Weitz, Paul Y Kim; COVID-BEACONS investiga

Universal Southern blot protocol with cold or radioactive probes for the validation of alleles obtained by homologous recombination

使用冷或放射性探针的通用南方印迹法来验证同源重组获得的等位基因

Gemma F Codner, Valerie Erbs, Jorik Loeffler, Lauren Chessum, Adam Caulder, Nicolas Jullien, Sara Wells, Marie-Christine Birling, Lydia Teboul

Investigating the phosphinic acid tripeptide mimetic DG013A as a tool compound inhibitor of the M1-aminopeptidase ERAP1

研究膦酸三肽模拟物DG013A作为M1-氨肽酶ERAP1的工具化合物抑制剂

Wilding, Birgit; Pasqua, A Elisa; E A Chessum, Nicola; Pierrat, Olivier A; Hahner, Tamas; Tomlin, Kathy; Shehu, Erald; Burke, Rosemary; Richards, G Meirion; Whitton, Bradleigh; Arwert, Esther N; Thapaliya, Arjun; Salimraj, Ramya; van Montfort, Rob; Skawinska, Agi; Hayes, Angela; Raynaud, Florence; Chopra, Rajesh; Jones, Keith; Newton, Gary; Cheeseman, Matthew D

Clarin-2 is essential for hearing by maintaining stereocilia integrity and function

Clarin-2 通过维持纤毛的完整性和功能对听力至关重要

Lucy A Dunbar, Pranav Patni, Carlos Aguilar, Philomena Mburu, Laura Corns, Helena Rr Wells, Sedigheh Delmaghani, Andrew Parker, Stuart Johnson, Debbie Williams, Christopher T Esapa, Michelle M Simon, Lauren Chessum, Sherylanne Newton, Joanne Dorning, Prashanthini Jeyarajan, Susan Morse, Andrea Lelli

The epilepsy-associated protein TBC1D24 is required for normal development, survival and vesicle trafficking in mammalian neurons

癫痫相关蛋白 TBC1D24 是哺乳动物神经元正常发育、存活和囊泡运输所必需的

Mattéa J Finelli, Davide Aprile, Enrico Castroflorio, Alexander Jeans, Matteo Moschetta, Lauren Chessum, Matteo T Degiacomi, Julia Grasegger, Alexis Lupien-Meilleur, Andrew Bassett, Elsa Rossignol, Philippe M Campeau, Michael R Bowl, Fabio Benfenati, Anna Fassio, Peter L Oliver

Helios is a key transcriptional regulator of outer hair cell maturation

Helios 是外毛细胞成熟的关键转录调控因子

Lauren Chessum, Maggie S Matern, Michael C Kelly, Stuart L Johnson, Yoko Ogawa, Beatrice Milon, Mark McMurray, Elizabeth C Driver, Andrew Parker, Yang Song, Gemma Codner, Christopher T Esapa, Jack Prescott, Graham Trent, Sara Wells, Abigail K Dragich, Gregory I Frolenkov, Matthew W Kelley, Walter Ma