日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Development of Optimized Exatecan-Based Immunoconjugates with Potent Antitumor Efficacy in HER2-Positive Breast Cancer

开发对HER2阳性乳腺癌具有强效抗肿瘤疗效的优化型依沙替康免疫偶联物

Auvert, Etienne; Douez, Emmanuel; Jolivet, Louis; Witkowski, Tiffany; Jallas, Anne-Catherine; Boursin, Fanny; Molnar, Ioana; Colas, Cyril; Wittmann, Sandrine Valsesia; Auriol, Manon; Chezal, Jean-Michel; Aubrey, Nicolas; Allard-Vannier, Emilie; Maisonial-Besset, Aurélie; Joubert, Nicolas; Denevault-Sabourin, Caroline

Tumor sink effect on melanin-ligand [(131)I]ICF01012 in melanoma and its implications for targeted radionuclide therapy.

黑色素瘤中黑色素配体[(131)I]ICF01012的肿瘤吸收效应及其对靶向放射性核素治疗的影响。

Jouberton Elodie, Besse Sophie, Billoux Tommy, Auzeloux Philippe, Schmitt Sébastien, Chezal Jean-Michel, Sas Nicolas, Noirault Laurine, Auriol Manon, Levesque Sophie, Delmas Marine, Chaussin Benjamin, Chautard Emmanuel, Miot-Noirault Elisabeth, Rouanet Jacques, Cachin Florent

Improved automated one-pot two-step radiosynthesis of (S)-[18F]FETrp, a radiotracer for PET imaging of indoleamine 2,3-dioxygenase 1 (IDO1)

改进的自动化一锅两步放射合成 (S)-[18F]FETrp,用于吲哚胺 2,3-双加氧酶 1 (IDO1) PET 成像的放射性示踪剂

Aurélie Maisonial-Besset, David Kryza, Klaus Kopka, Sophie Levesque, Emmanuel Moreau, Barbara Wenzel, Jean-Michel Chezal

A Convenient Route to New (Radio)Fluorinated and (Radio)Iodinated Cyclic Tyrosine Analogs

合成新型(放射性)氟化和(放射性)碘化环状酪氨酸类似物的便捷途径

Chao, Maria Noelia; Chezal, Jean-Michel; Debiton, Eric; Canitrot, Damien; Witkowski, Tiffany; Levesque, Sophie; Degoul, Françoise; Tarrit, Sébastien; Wenzel, Barbara; Miot-Noirault, Elisabeth; Serre, Audrey; Maisonial-Besset, Aurélie

Novel Radioiodinated and Radiofluorinated Analogues of FT-2102 for SPECT or PET Imaging of mIDH1 Mutant Tumours

FT-2102 的新型放射性碘化和放射性氟化类似物,用于 mIDH1 突变肿瘤的 SPECT 或 PET 成像

Valérie Weber, Lucie Arnaud, Sladjana Dukic-Stefanovic, Barbara Wenzel, Valérie Roux, Jean-Michel Chezal, Thu-Hang Lai, Rodrigo Teodoro, Klaus Kopka, Elisabeth Miot-Noirault, Winnie Deuther-Conrad, Aurélie Maisonial-Besset

Synthesis and In Vitro Comparison of DOTA, NODAGA and 15-5 Macrocycles as Chelators for the 64Cu-Labelling of Immunoconjugates

DOTA、NODAGA 和 15-5 大环化合物作为免疫偶联物 64Cu 标记螯合剂的合成及体外比较

Aurélie Maisonial-Besset, Tiffany Witkowski, Mercedes Quintana, Sophie Besse, Vincent Gaumet, Axel Cordonnier, Cyrille Alliot, Aurélien Vidal, Caroline Denevault-Sabourin, Sébastien Tarrit, Sophie Levesque, Elisabeth Miot-Noirault, Jean-Michel Chezal

Phase I study of [(131)I] ICF01012, a targeted radionuclide therapy, in metastatic melanoma: MELRIV-1 protocol

[(131)I] ICF01012(一种靶向放射性核素疗法)治疗转移性黑色素瘤的 I 期研究:MELRIV-1 方案

Thivat, Emilie; Rouanet, Jacques; Auzeloux, Philippe; Sas, Nicolas; Jouberton, Elodie; Levesque, Sophie; Billoux, Tommy; Mansard, Sandrine; Molnar, Ioana; Chanchou, Marion; Fois, Giovanna; Maigne, Lydia; Chezal, Jean-Michel; Miot-Noirault, Elisabeth; D'Incan, Michel; Durando, Xavier; Cachin, Florent

[(18)F]ML-10 PET imaging fails to assess early response to neoadjuvant chemotherapy in a preclinical model of triple negative breast cancer

[(18)F]ML-10 PET 成像无法评估三阴性乳腺癌临床前模型中新辅助化疗的早期疗效

Jouberton, Elodie; Schmitt, Sébastien; Chautard, Emmanuel; Maisonial-Besset, Aurélie; Roy, Marie; Radosevic-Robin, Nina; Chezal, Jean-Michel; Miot-Noirault, Elisabeth; Bouvet, Yann; Cachin, Florent

Pretargeted radioimmunotherapy and SPECT imaging of peritoneal carcinomatosis using bioorthogonal click chemistry: probe selection and first proof-of-concept

利用生物正交点击化学进行腹膜癌预靶向放射免疫治疗和SPECT成像:探针选择和初步概念验证

Rondon, Aurélie; Schmitt, Sébastien; Briat, Arnaud; Ty, Nancy; Maigne, Lydia; Quintana, Mercedes; Membreno, Rosemery; Zeglis, Brian M; Navarro-Teulon, Isabelle; Pouget, Jean-Pierre; Chezal, Jean-Michel; Miot-Noirault, Elisabeth; Moreau, Emmanuel; Degoul, Françoise

Targeted Radionuclide Therapy Decreases Melanoma Lung Invasion by Modifying Epithelial-Mesenchymal Transition-Like Mechanisms

靶向放射性核素疗法通过改变上皮-间质转化样机制来减少黑色素瘤肺部侵袭

Akil, Hussein; Rouanet, Jacques; Viallard, Claire; Besse, Sophie; Auzeloux, Philippe; Chezal, Jean-Michel; Miot-Noirault, Elisabeth; Quintana, Mercedes; Degoul, Françoise