Searching for Synthetic Opioid Rescue Agents: Identification of a Potent Opioid Agonist with Reduced Respiratory Depression
寻找合成阿片类药物解救剂:鉴定一种具有强效阿片类激动剂和降低呼吸抑制作用
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.4c00333
Vu, Loan Y; Luo, Dan; Johnson, Kai; Denehy, Emily D; Songrady, Judy C; Martin, Jocelyn; Trivedi, Riya; Alsum, Alexia R; Shaykin, Jakob D; Chaudhary, Chhabi Lal; Woloshin, Eric J; Kornberger, Lindsay; Bhuiyan, Nazmul; Parkin, Sean; Jiang, Qianru; Che, Tao; Alilain, Warren; Turner, Jill R; Bardo, Michael T; Prisinzano, Thomas E