Targeting oncogenic K-RAS mutants with small-molecule degrader XMU-MP-9 through NEDD4-1.
利用小分子降解剂 XMU-MP-9 通过 NEDD4-1 靶向致癌 K-RAS 突变体。
期刊:Acta Pharmaceutica Sinica B
影响因子:14.6
doi:10.1016/j.apsb.2025.07.031
Zeng Taoling, Jiang Tingting, Zhang Baoding, Zhang Ting, Dai Wanjun, Yin Xun, Li Yunzhan, Yu Zhuoran, Wu Caiming, Wu Yaying, Chi Ximin, Deng Xianming, Wang Hong-Rui