日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Mechanistic insights and in vivo HIV suppression by the BRD4-targeting small molecule ZL0580

靶向BRD4的小分子ZL0580的机制研究及体内HIV抑制作用

Kumar, Naveen; Ma, Zonghui; Long, Fuquan; Bonam, Srinivasa Reddy; Lai, Hsien-Tsung; Wu, Shwu-Yuan; Chen, Haiying; Hazell, Nicholas C; Bei, Jiani; Liu, Xuefeng; Chen, Yeqing; Wei, Zhi; Chiang, Cheng-Ming; Zhou, Jia; Hu, Haitao

Mechanistic insights and in vivo HIV suppression by the BRD4-targeting small molecule ZL0580

靶向BRD4的小分子ZL0580的机制研究及体内HIV抑制作用

Kumar, Naveen; Ma, Zonghui; Long, Fuquan; Bonam, Srinivasa Reddy; Lai, Hsien-Tsung; Wu, Shwu-Yuan; Chen, Haiying; Hazell, Nicholas C; Bei, Jiani; Liu, Xuefeng; Wei, Zhi; Chiang, Cheng-Ming; Zhou, Jia; Hu, Haitao

BRD4 binds the nucleosome via both histone and DNA interactions.

BRD4 通过组蛋白和 DNA 相互作用与核小体结合

Zhu Jiang, Leith Erik M, O'Donnell Erin N, Manzano Bryan P, Wu Shwu-Yuan, Chiang Cheng-Ming, Armache Jean-Paul, Tan Song

Novel BRD4-p53 Inhibitor SDU-071 Suppresses Proliferation and Migration of MDA-MB-231 Triple-Negative Breast Cancer Cells.

新型 BRD4-p53 抑制剂 SDU-071 可抑制 MDA-MB-231 三阴性乳腺癌细胞的增殖和迁移

Wang Shumei, Lei Kang, Lai Hsien-Tsung, Liu Tingting, Du Lupei, Wu Shwu-Yuan, Ye Xiaohan, Chiang Cheng-Ming, Li Minyong

Erratum: N6-methyladenosine-induced ERRγ triggers chemoresistance of cancer cells through upregulation of ABCB1 and metabolic reprogramming: Erratum

勘误:N6-甲基腺苷诱导的ERRγ通过上调ABCB1和代谢重编程触发癌细胞的化疗耐药性:勘误

Chen, Zhuojia; Wu, Long; Zhou, Jiawang; Lin, Xinyao; Peng, Yanxi; Ge, Lichen; Chiang, Cheng-Ming; Huang, Hui; Wang, Hongsheng; He, Weiling

MYC promotes global transcription in part by controlling P-TEFb complex formation via DNA-binding independent inhibition of CDK9 SUMOylation

MYC通过不依赖于DNA结合的CDK9 SUMO化抑制作用,部分地控制P-TEFb复合物的形成,从而促进全局转录。

Guan, Qingqing; Chen, Zhaosu; Yu, Fang; Liu, Lingling; Huang, Yuanyong; Wei, Gang; Chiang, Cheng-Ming; Wong, Jiemin; Li, Jiwen

Direct interaction with the BRD4 carboxyl-terminal motif (CTM) and TopBP1 is required for human papillomavirus 16 E2 association with mitotic chromatin and plasmid segregation function

人乳头瘤病毒16 E2蛋白与有丝分裂染色质的结合以及质粒分离功能需要与BRD4羧基末端基序(CTM)和TopBP1直接相互作用。

Prabhakar, Apurva T; James, Claire D; Fontan, Christian T; Otoa, Raymonde; Wang, Xu; Bristol, Molly L; Hill, Ronald D; Dubey, Aanchal; Wu, Shwu-Yuan; Chiang, Cheng-Ming; Morgan, Iain M

Blood-based biomarkers of human papillomavirus-associated cancers: A systematic review and meta-analysis

人乳头瘤病毒相关癌症的血液生物标志物:系统评价和荟萃分析

Balachandra, Sanjana; Kusin, Samuel B; Lee, Rebecca; Blackwell, James-Michael; Tiro, Jasmin A; Cowell, Lindsay G; Chiang, Cheng-Ming; Wu, Shwu-Yuan; Varma, Sanskriti; Rivera, Erika L; Mayo, Helen G; Ding, Lianghao; Sumer, Baran D; Lea, Jayanthi S; Bagrodia, Aditya; Farkas, Linda M; Wang, Richard; Fakhry, Carole; Dahlstrom, Kristina R; Sturgis, Erich M; Day, Andrew T

Inhibition of BRD4 suppresses the malignancy of breast cancer cells via regulation of Snail

抑制BRD4可通过调控Snail抑制乳腺癌细胞的恶性转化。

Lu, Linlin; Chen, Zhuojia; Lin, Xinyao; Tian, Lin; Su, Qiao; An, Panpan; Li, Wuguo; Wu, Yingmin; Du, Jun; Shan, Hong; Chiang, Cheng-Ming; Wang, Hongsheng

N6-methyladenosine-induced ERRγ triggers chemoresistance of cancer cells through upregulation of ABCB1 and metabolic reprogramming

N6-甲基腺苷诱导的ERRγ通过上调ABCB1和代谢重编程引发癌细胞的化疗耐药性

Chen, Zhuojia; Wu, Long; Zhou, Jiawang; Lin, Xinyao; Peng, Yanxi; Ge, Lichen; Chiang, Cheng-Ming; Huang, Hui; Wang, Hongsheng; He, Weiling