日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design of Potent Menin-KMT2A Interaction Inhibitors with Improved In Vitro ADME Properties and Reduced hERG Affinity

设计具有改进的体外ADME特性和降低的hERG亲和力的高效Menin-KMT2A相互作用抑制剂

Chapsal, Bruno D; Kimbrough, Jennifer R; Bester, Stephanie M; Bergstrom, Alex; Backos, Donald S; Campos, Bismarck; McDonald, Matthew G; Abrahamsen, Rebecca; Allen, Andrew C; Doerner Barbour, Patrick M; Bettendorf, Tanna; Boys, Mark L; Brown, Karin; Chicarelli, Mark J; Cook, Adam W; Crooks, Amy L; Cruz, Cole L; Dahlke, Joshua R; Eide, Alida; Fell, Jay B; Fulton, Jennifer L; Gargus, Matthew; Gaudino, John J; Guarnieri, Anna L; Hansen, Erik P; Holt, Melissa C; Kahn, Dean R; Laird, Ellen R; Larsen, Paul D; Linwood, Rebecca; Martinson, Matthew C; McCown, Joseph; Mejia, Macedonio J; Moreno, David A; Mou, Tung-Chung; Newhouse, Brad; O'Leary, Jacob M; Rodriguez, Martha E; Singh, Anurag; Sinik, Lenka; Strand, Keith A; Touney, Eric E; Wollenberg, Lance A; Wong, Jim; Zhou, Yeyun; Fischer, John P; Allen, Shelley

Commentary to "Polylactic Acid: Is It Everything the Same? [sic]"

对“聚乳酸:它是否与所有其他物质都相同?[原文如此]”的评论

Chicarelli Martin, Jose Eduardo

Morphometric and volumetric analysis of the frontal sinus in a brazilian population using cone beam computed tomography: a forensic approach for sex, age and facial morphology determination

利用锥形束计算机断层扫描技术对巴西人群额窦进行形态计量学和体积分析:一种用于性别、年龄和面部形态鉴定的法医学方法

Bego de Miranda, Letícia; Felipe, Beatriz Caio; Couto, Matheus Kawana; Takeshita, Wilton Mitsunari; Vessoni Iwaki, Lilian Cristina; Chicarelli da Silva, Mariliani

Discovery of 5-Azaquinoxaline Derivatives as Potent and Orally Bioavailable Allosteric SHP2 Inhibitors

发现5-氮杂喹喔啉衍生物作为高效且口服生物利用度高的变构SHP2抑制剂

Elsayed, Mohamed S A; Blake, James F; Boys, Mark L; Brown, Eric; Chapsal, Bruno D; Chicarelli, Mark J; Cook, Adam W; Fell, Jay B; Fischer, John P; Hanson, Lauren; Lemieux, Christine; Martinson, Matthew C; McCown, Joseph; McNulty, Oren T; Mejia, Macedonio J; Neitzel, Nickolas A; Otten, Jennifer N; Rodriguez, Martha E; Wilcox, Daniel; Wong, Christina E; Zhou, Yeyun; Hinklin, Ronald J

Effect of Tricalcium Silicate on Direct Pulp Capping: Experimental Study in Rats

硅酸三钙对直接盖髓术的影响:大鼠实验研究

Chicarelli, Lúcio P G; Webber, Mariana B F; Amorim, João P A; Rangel, Ana L C A; Camilotti, Veridiana; Sinhoreti, Mario A C; Mendonça, Marcio J

Discovery of Tetrahydropyridopyrimidines as Irreversible Covalent Inhibitors of KRAS-G12C with In Vivo Activity

发现四氢吡啶并嘧啶类化合物作为KRAS-G12C的不可逆共价抑制剂,并具有体内活性

Fell, Jay B; Fischer, John P; Baer, Brian R; Ballard, Joshua; Blake, James F; Bouhana, Karyn; Brandhuber, Barbara J; Briere, David M; Burgess, Laurence E; Burkard, Michael R; Chiang, Harrah; Chicarelli, Mark J; Davidson, Kevin; Gaudino, John J; Hallin, Jill; Hanson, Lauren; Hee, Kenneth; Hicken, Erik J; Hinklin, Ronald J; Marx, Matthew A; Mejia, Macedonio J; Olson, Peter; Savechenkov, Pavel; Sudhakar, Niranjan; Tang, Tony P; Vigers, Guy P; Zecca, Henry; Christensen, James G

C5-Alkyl-2-methylurea-Substituted Pyridines as a New Class of Glucokinase Activators

C5-烷基-2-甲基脲取代的吡啶类化合物作为一类新型葡萄糖激酶激活剂

Du, Xiaohui; Hinklin, Ronald J; Xiong, Yumei; Dransfield, Paul; Park, Jaehyeon; Kohn, Todd J; Pattaropong, Vatee; Lai, SuJen; Fu, Zice; Jiao, Xianyun; Chow, David; Jin, Lixia; Davda, Jasmine; Veniant, Murielle M; Anderson, Deborah A; Baer, Brian R; Bencsik, Josef R; Boyd, Steven A; Chicarelli, Mark Joseph; Mohr, Peter J; Wang, Bin; Condroski, Kevin R; DeWolf, Walter E; Conn, Marion; Tran, Thanhvien; Yang, Jerry; Aicher, Thomas D; Medina, Julio C; Coward, Peter; Houze, Jonathan B

Characterization of a novel glucokinase activator in rat and mouse models

在大鼠和小鼠模型中对一种新型葡萄糖激酶激活剂进行表征

Lu, Min; Li, Pingping; Bandyopadhyay, Gautam; Lagakos, William; Dewolf, Walter E Jr; Alford, Taylor; Chicarelli, Mark Joseph; Williams, Lance; Anderson, Deborah A; Baer, Brian R; McVean, Maralee; Conn, Marion; Véniant, Murielle M; Coward, Peter

Evaluation of diagnostic accuracy of conventional and digital periapical radiography, panoramic radiography, and cone-beam computed tomography in the assessment of alveolar bone loss

评估传统和数字化根尖周X线片、全景X线片和锥形束计算机断层扫描在诊断牙槽骨丢失方面的准确性

Takeshita, Wilton Mitsunari; Vessoni Iwaki, Lilian Cristina; Da Silva, Mariliani Chicarelli; Tonin, Renata Hernandes

Comparison of periapical radiography with cone beam computed tomography in the diagnosis of vertical root fractures in teeth with metallic post

比较根尖周X线片与锥形束计算机断层扫描在诊断金属桩牙垂直根折中的应用

Takeshita, Wilton Mitsunari; Iwaki, Lilian Cristina Vessoni; da Silva, Mariliani Chicarelli; Sabio, Sergio; Albino, Paulo Ricardo Febrairo