日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of an ITK and TRK kinase inhibitor for the potential topical treatment of atopic dermatitis

发现一种ITK和TRK激酶抑制剂,可用于治疗特应性皮炎。

Duffen, Jennifer L; Crouse, Kimberly K; Ji, Lin; Brault, Amy L; Ford, Kristen; Brooks, Jonathan; Jelinsky, Scott A; Li, Yizheng; Shin, Julia H; Zhao, Yajuan; Andreyeva, Tatyana; Hammerman, Katherine; Arnold, Christina; Sheldon, Richard T; Garren, Jeonifer; LaBarge, Wes; Resek, Anthony; Volmer, Jon; Bagley, Scott W; Casimiro-Garcia, Agustin; Chinigo, Gary M; Davoren, Jennifer E; Denny, Rajiah Aldrin; Drozda, Susan; Foley, Timothy L; Hicklin, Robert W; Liu, Shenping; Lovering, Frank E; Nedoma, Nicole L; Parikh, Mihir D; Strohbach, Joseph W; Trujillo, John I; Steyn, Stefanus J; Nocka, Karl; Hegen, Martin; Vincent, Fabien; Lee, Katherine L; Gerstenberger, Brian S; Primiano, Michael J

Radical Sampling Enabled Saturated N-Heterocycle Cyclization

自由基采样实现了饱和N-杂环环化

Cai, Qinyan; Bissonnette, Noah B; Kim, Saegun; Knauber, Thomas; Chinigo, Gary M; Blakemore, David C; MacMillan, David W C

Sharp wave-ripple clusters enhance hippocampal-neocortical engagement for memory consolidation

尖波-涟漪簇增强海马-新皮层参与记忆巩固

Vöröslakos, Mihály; Lafferty, Christopher; Zheng, ZheYang; Paleologos, Nicholas; Chinigo, Elisa; McClain, Kathryn; Aykan, Deren; Yoon, Euisik; Buzsáki, György

Profound Impact of Local Climatic Conditions on IgE Sensitization Profiles: Evidence from Argentine Cities

局部气候条件对IgE致敏谱的深远影响:来自阿根廷城市的证据

Sarzsinszky, Eszter; Smaldini, Paola; Chinigo, Marcela; Ardanaz, María; Benítez, Pablo; Ramos, Ana; Braviz Lopez, María Eugenia; Ramón, Gonzalo; Ramón, Germán; Schlederer, Thomas; Tulaev, Mikhail; Valenta, Rudolf; Huang, Huey-Jy; Vrtala, Susanne; Docena, Guillermo; The Allergochip Working Group

Peptidylarginine Deiminase (PAD) Inhibitor Optimization through Displacement of a Trapped Water Molecule

通过置换被捕获的水分子来优化肽基精氨酸脱亚胺酶(PAD)抑制剂

Schnute, Mark E; Chinigo, Gary M; Futatsugi, Kentaro; Yamaguchi, Masaya; Bagley, Scott W; Banker, Mary Ellen; Chang, Jeanne S; Chen, Ming Z; Choi, Won Young; Corbett, Matthew S; Drozda, Susan E; Ebner, David C; Garcia-Irizarry, Carmen; Hicklin, Robert; Hoy, Susan; Jiao, Wenhua; Kortum, Steven; Lee, Katherine L; Limburg, David C; Lovering, Frank; Moreno, Antonio; Mousseau, James J; Pan, Senliang; Parikh, Mihir D; Pelker, Jeffrey W; Ramsey, Simeon; Reilly, Usa; Rescourio, Gwenaella; Schmitt, Daniel C; Simpson, Brittany; Skrzypek, Grzegorz J; Smaltz, Daniel J; Taylor, Alexandria P; Torella, Rubben; Trujillo, John I; Vajdos, Felix F; Wepy, James A; Wright, Stephen W; Blakemore, David C; Vincent, Fabien; Clerin, Valerie M

Structural basis for CCR6 modulation by allosteric antagonists

变构拮抗剂调节 CCR6 的结构基础

David Jonathan Wasilko, Brian S Gerstenberger, Kathleen A Farley, Wei Li, Jennifer Alley, Mark E Schnute, Ray J Unwalla, Jorge Victorino, Kimberly K Crouse, Ru Ding, Parag V Sahasrabudhe, Fabien Vincent, Richard K Frisbie, Alpay Dermenci, Andrew Flick, Chulho Choi, Gary Chinigo, James J Mousseau, Jo

One-Pot Synthesis of Sulfonamides from Unactivated Acids and Amines via Aromatic Decarboxylative Halosulfonylation

通过芳香脱羧卤代磺酰化反应,由未活化的酸和胺一锅法合成磺酰胺

Pedersen, P Scott; Blakemore, David C; Chinigo, Gary M; Knauber, Thomas; MacMillan, David W C

Decarbonylative Pd-Catalyzed Suzuki Cross-Coupling for the Synthesis of Structurally Diverse Heterobiaryls

脱羰基钯催化Suzuki交叉偶联反应合成结构多样的杂双芳烃

Cervantes-Reyes, Alejandro; Smith, Aaron C; Chinigo, Gary M; Blakemore, David C; Szostak, Michal

Transient Receptor Potential Channel Expression Signatures in Tumor-Derived Endothelial Cells: Functional Roles in Prostate Cancer Angiogenesis

肿瘤来源的内皮细胞中的瞬时受体电位通道表达特征:在前列腺癌血管生成中的功能作用

Michela Bernardini, Alessia Brossa, Giorgia Chinigo, Guillaume P Grolez, Giulia Trimaglio, Laurent Allart, Audrey Hulot, Guillemette Marot, Tullio Genova, Aditi Joshi, Virginie Mattot, Gaelle Fromont, Luca Munaron, Benedetta Bussolati, Natalia Prevarskaya, Alessandra Fiorio Pla, Dimitra Gkika0