日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of SD-436: A Potent, Highly Selective and Efficacious STAT3 PROTAC Degrader Capable of Achieving Complete and Long-Lasting Tumor Regression

SD-436 的发现:一种强效、高选择性和高效的 STAT3 PROTAC 降解剂,能够实现完全且持久的肿瘤消退

Xu, Renqi; Zhou, Haibin; Bai, Longchuan; McEachern, Donna; Wu, Dimin; Acharyya, Ranjan Kumar; Wang, Mi; Tošović, Jelena; Yang, Chao-Yie; Chinnaswamy, Krishnapriya; Meagher, Jennifer L; Stuckey, Jeanne A; Liu, Cai; Wang, Meilin; Wen, Bo; Sun, Duxin; Wang, Shaomeng

Comprehensive Analyses of the Effects of the Small-Molecule Inhibitor of the UHM Domain in the Splicing Factor U2AF1 in Leukemia Cells

对白血病细胞中剪接因子U2AF1的UHM结构域小分子抑制剂作用的综合分析

Yuan, Xinrui; Sabzvar, Mona Kazemi; Patil, Amol D; Chinnaswamy, Krishnapriya; Howie, Kathryn L; Andhavaram, Ramaraju; Wang, Borwyn; Siegler, Maxime A; Dumaz, Arda; Stuckey, Jeanne A; Corey, Seth J; Maciejewski, Jaroslaw P; Visconte, Valeria; Yang, Chao-Yie

Structure-Activity relationship of 1-(Furan-2ylmethyl)Pyrrolidine-Based Stimulation-2 (ST2) inhibitors for treating graft versus host disease

1-(呋喃-2-基甲基)吡咯烷类刺激-2 (ST2) 抑制剂治疗移植物抗宿主病的构效关系

Yuan, Xinrui; Jiang, Hua; Fu, Denggang; Robida, Aaron; Rajanayake, Krishani; Yuan, Hebao; Wen, Bo; Sun, Duxin; Watch, Brennan T; Chinnaswamy, Krishnapriya; Stuckey, Jeanne A; Paczesny, Sophie; Rech, Jason C; Yang, Chao-Yie

Discovery of M-808 as a Highly Potent, Covalent, Small-Molecule Inhibitor of the Menin-MLL Interaction with Strong In Vivo Antitumor Activity.

发现 M-808 是一种高效的共价小分子抑制剂,可抑制 Menin-MLL 相互作用,并具有很强的体内抗肿瘤活性

Xu Shilin, Aguilar Angelo, Huang Liyue, Xu Tianfeng, Zheng Ke, McEachern Donna, Przybranowski Sally, Foster Caroline, Zawacki Kaitlin, Liu Zhaomin, Chinnaswamy Krishnapriya, Stuckey Jeanne, Wang Shaomeng

Changing the Apoptosis Pathway through Evolutionary Protein Design

通过进化蛋白质设计改变细胞凋亡通路

Shultis, David; Mitra, Pralay; Huang, Xiaoqiang; Johnson, Jarrett; Khattak, Naureen Aslam; Gray, Felicia; Piper, Clint; Czajka, Jeff; Hansen, Logan; Wan, Bingbing; Chinnaswamy, Krishnapriya; Liu, Liu; Wang, Mi; Pan, Jingxi; Stuckey, Jeanne; Cierpicki, Tomasz; Borchers, Christoph H; Wang, Shaomeng; Lei, Ming; Zhang, Yang

CSAR Benchmark Exercise 2013: Evaluation of Results from a Combined Computational Protein Design, Docking, and Scoring/Ranking Challenge

2013 年 CSAR 基准测试:综合计算蛋白质设计、对接和评分/排名挑战的结果评估

Smith, Richard D; Damm-Ganamet, Kelly L; Dunbar, James B Jr; Ahmed, Aqeel; Chinnaswamy, Krishnapriya; Delproposto, James E; Kubish, Ginger M; Tinberg, Christine E; Khare, Sagar D; Dou, Jiayi; Doyle, Lindsey; Stuckey, Jeanne A; Baker, David; Carlson, Heather A