日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Modulating IDO1 and TDO Inhibition Through Structural Modification of Diaryl Hydroxylamines

通过二芳基羟胺的结构修饰调节IDO1和TDO抑制作用

Foscolos, Angeliki S; Pappas, Alexandros; Petroulias, Christos N; Kapella, Anna; Prifti, Georgia M; Zoidis, Grigoris; Papadopoulos, Minas; Mpakali, Anastasia; Chiotellis, Aristeidis

Synthesis and Evaluation of (99m)Tc(CO)(3) Complexes with Ciprofloxacin Dithiocarbamate for Infection Imaging

合成和评价(99m)Tc(CO)3与环丙沙星二硫代氨基甲酸酯的配合物用于感染成像

Papasavva, Afroditi; Pirmettis, Nektarios N; Shegani, Antonio; Papadopoulou, Eleni; Kiritsis, Christos; Georgoutsou-Spyridonos, Maria; Mastellos, Dimitrios C; Chiotellis, Aristeidis; Kyprianidou, Patricia; Pelecanou, Maria; Papadopoulos, Minas; Pirmettis, Ioannis

Synthesis and Biological Evaluation of Novel Cationic Rhenium and Technetium-99m Complexes Bearing Quinazoline Derivative for Epidermal Growth Factor Receptor Targeting

新型含喹唑啉衍生物的阳离子铼和锝-99m配合物的合成及生物学评价及其在表皮生长因子受体靶向治疗中的应用

Triantopoulou, Sotiria; Roupa, Ioanna; Shegani, Antonio; Pirmettis, Nektarios N; Terzoudi, Georgia I; Chiotellis, Aristeidis; Tolia, Maria; Damilakis, John; Pirmettis, Ioannis; Paravatou-Petsota, Maria

N-Hydroxypiridinedione: A Privileged Heterocycle for Targeting the HBV RNase H

N-羟基吡啶二酮:一种靶向HBV RNase H的优势杂环化合物

Moianos, Dimitrios; Makri, Maria; Prifti, Georgia-Myrto; Chiotellis, Aristeidis; Pappas, Alexandros; Woodson, Molly E; Tajwar, Razia; Tavis, John E; Zoidis, Grigoris

Evaluation of Rhenium and Technetium-99m Complexes Bearing Quinazoline Derivatives as Potential EGFR Agents

评价含喹唑啉衍生物的铼和锝-99m配合物作为潜在的EGFR抑制剂

Makrypidi, Konstantina; Kiritsis, Christos; Roupa, Ioanna; Triantopoulou, Sotiria; Shegani, Antonio; Paravatou-Petsotas, Maria; Chiotellis, Aristeidis; Pelecanou, Maria; Papadopoulos, Minas; Pirmettis, Ioannis

Synthesis and Characterization of Novel [2 + 1] Tricarbonyl Rhenium Complexes with the Hydrophilic Phosphine Ligands PTA and CAP

合成与表征新型[2+1]三羰基铼配合物及其亲水性膦配体PTA和CAP

Roupa, Ioanna; Flampouraris, Charalampos; Shegani, Antonio; Ischyropoulou, Myrto; Makrypidi, Konstantina; Raptopoulou, Catherine; Pirmettis, Ioannis; Papadopoulos, Minas S; Psycharis, Vassilis; Chiotellis, Aristeidis

Synthesis and In Vitro Evaluation of Gold Nanoparticles Functionalized with Thiol Ligands for Robust Radiolabeling with (99m)Tc

合成并体外评价硫醇配体功能化的金纳米粒子,用于与 (99m)Tc 进行稳健的放射性标记

Apostolopoulou, Adamantia; Chiotellis, Aristeidis; Salvanou, Evangelia-Alexandra; Makrypidi, Konstantina; Tsoukalas, Charalampos; Kapiris, Fotis; Paravatou-Petsotas, Maria; Papadopoulos, Minas; Pirmettis, Ioannis C; Koźmiński, Przemysław; Bouziotis, Penelope

Whole-body and adipose tissue-specific mechanisms underlying the metabolic effects of fibroblast growth factor 21 in the Siberian hamster

西伯利亚仓鼠体内成纤维细胞生长因子21代谢效应的全身和脂肪组织特异性机制

Lewis, Jo E; Monnier, Chloe; Marshall, Hayley; Fowler, Maxine; Green, Rebecca; Cooper, Scott; Chiotellis, Aristeidis; Luckett, Jeni; Perkins, Alan C; Coskun, Tamer; Adams, Andrew C; Samms, Ricardo J; Ebling, Francis J P; Tsintzas, Kostas

Evaluation of the radiolabeled boronic acid-based FAP inhibitor MIP-1232 for atherosclerotic plaque imaging

放射性标记硼酸基 FAP 抑制剂 MIP-1232 对动脉粥样硬化斑块成像的评价

Romana Meletta, Adrienne Müller Herde, Aristeidis Chiotellis, Malsor Isa, Zoran Rancic, Nicole Borel, Simon M Ametamey, Stefanie D Krämer, Roger Schibli

Site-Specific Conjugation of Monomethyl Auristatin E to Anti-CD30 Antibodies Improves Their Pharmacokinetics and Therapeutic Index in Rodent Models

单甲基奥瑞他汀 E 与抗 CD30 抗体的位点特异性结合可改善其在啮齿动物模型中的药代动力学和治疗指数

F Lhospice, D Brégeon, C Belmant, P Dennler, A Chiotellis, E Fischer, L Gauthier, A Boëdec, H Rispaud, S Savard-Chambard, A Represa, N Schneider, C Paturel, M Sapet, C Delcambre, S Ingoure, N Viaud, C Bonnafous, R Schibli, F Romagné