日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Potent Antimalarials with Development Potential Identified by Structure-Guided Computational Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series

通过基于吡咯的二氢乳清酸脱氢酶抑制剂系列的结构导向计算优化,鉴定出具有开发潜力的强效抗疟药物

Palmer, Michael J; Deng, Xiaoyi; Watts, Shawn; Krilov, Goran; Gerasyuto, Aleksey; Kokkonda, Sreekanth; El Mazouni, Farah; White, John; White, Karen L; Striepen, Josefine; Bath, Jade; Schindler, Kyra A; Yeo, Tomas; Shackleford, David M; Mok, Sachel; Deni, Ioanna; Lawong, Aloysus; Huang, Ann; Chen, Gong; Wang, Wen; Jayaseelan, Jaya; Katneni, Kasiram; Patil, Rahul; Saunders, Jessica; Shahi, Shatrughan P; Chittimalla, Rajesh; Angulo-Barturen, Iñigo; Jiménez-Díaz, María Belén; Wittlin, Sergio; Tumwebaze, Patrick K; Rosenthal, Philip J; Cooper, Roland A; Aguiar, Anna Caroline Campos; Guido, Rafael V C; Pereira, Dhelio B; Mittal, Nimisha; Winzeler, Elizabeth A; Tomchick, Diana R; Laleu, Benoît; Burrows, Jeremy N; Rathod, Pradipsinh K; Fidock, David A; Charman, Susan A; Phillips, Margaret A

Lead Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series for the Treatment of Malaria.

吡咯基二氢乳清酸脱氢酶抑制剂系列先导化合物的优化及其在疟疾治疗中的应用

Kokkonda Sreekanth, Deng Xiaoyi, White Karen L, El Mazouni Farah, White John, Shackleford David M, Katneni Kasiram, Chiu Francis C K, Barker Helena, McLaren Jenna, Crighton Elly, Chen Gong, Angulo-Barturen Inigo, Jimenez-Diaz Maria Belen, Ferrer Santiago, Huertas-Valentin Leticia, Martinez-Martinez Maria Santos, Lafuente-Monasterio Maria Jose, Chittimalla Rajesh, Shahi Shatrughan P, Wittlin Sergio, Waterson David, Burrows Jeremy N, Matthews Dave, Tomchick Diana, Rathod Pradipsinh K, Palmer Michael J, Charman Susan A, Phillips Margaret A