日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

White Paper: Mimetics of Class 2 Tumor Suppressor Proteins as Novel Drug Candidates for Personalized Cancer Therapy

白皮书:II类肿瘤抑制蛋白模拟物作为个性化癌症治疗的新型候选药物

Dahl, Edgar; Villwock, Sophia; Habenberger, Peter; Choidas, Axel; Rose, Michael; Klebl, Bert M

Synthesis, Biological Evaluation, and Binding Mode of a New Class of Oncogenic K-Ras4b Inhibitors

新型致癌性K-Ras4b抑制剂的合成、生物学评价及结合模式

Jeuken, Stephan; Shkura, Oleksandr; Röger, Marc; Brickau, Victoria; Choidas, Axel; Degenhart, Carsten; Gülden, Daniel; Klebl, Bert; Koch, Uwe; Stoll, Raphael; Scherkenbeck, Jürgen

Anti-leukemic effect of CDK9 inhibition in T-cell prolymphocytic leukemia

CDK9 抑制对 T 细胞幼淋巴细胞白血病的抗白血病作用

Patricia Johansson, Laura Dierichs, Ludger Klein-Hitpass, Anke K Bergmann, Michael Möllmann, Sascha Menninger, Peter Habenberger, Bert Klebl, Jens T Siveke, Ulrich Dührsen, Axel Choidas, Jan Dürig

Gasdermin D plays a vital role in the generation of neutrophil extracellular traps

Gasdermin D 在中性粒细胞胞外陷阱的生成中起着至关重要的作用

Gabriel Sollberger, Axel Choidas, Garth Lawrence Burn, Peter Habenberger, Raffaella Di Lucrezia, Susanne Kordes, Sascha Menninger, Jan Eickhoff, Peter Nussbaumer, Bert Klebl, Renate Krüger, Alf Herzig, Arturo Zychlinsky

SAMHD1 is recurrently mutated in T-cell prolymphocytic leukemia

SAMHD1在T细胞前淋巴细胞白血病中反复发生突变

Johansson, Patricia; Klein-Hitpass, Ludger; Choidas, Axel; Habenberger, Peter; Mahboubi, Bijan; Kim, Baek; Bergmann, Anke; Scholtysik, René; Brauser, Martina; Lollies, Anna; Siebert, Reiner; Zenz, Thorsten; Dührsen, Ulrich; Küppers, Ralf; Dürig, Jan

Identification of an (-)-englerin A analogue, which antagonizes (-)-englerin A at TRPC1/4/5 channels

鉴定出一种(-)-englerin A类似物,该类似物可拮抗TRPC1/4/5通道上的(-)-englerin A。

Rubaiy, Hussein N; Seitz, Tobias; Hahn, Sven; Choidas, Axel; Habenberger, Peter; Klebl, Bert; Dinkel, Klaus; Nussbaumer, Peter; Waldmann, Herbert; Christmann, Mathias; Beech, David J

Dynarrestin, a Novel Inhibitor of Cytoplasmic Dynein

Dynarrestin,一种新型细胞质动力蛋白抑制剂

Susanne Höing, Ting-Yu Yeh, Matthias Baumann, Nancy E Martinez, Peter Habenberger, Lea Kremer, Hannes C A Drexler, Philipp Küchler, Peter Reinhardt, Axel Choidas, Mia-Lisa Zischinsky, Gunther Zischinsky, Swaran Nandini, Aaron P Ledray, Stephanie A Ketcham, Lydia Reinhardt, Masin Abo-Rady, Michael Gl

Potent anti-leukemic activity of a specific cyclin-dependent kinase 9 inhibitor in mouse models of chronic lymphocytic leukemia

特定细胞周期蛋白依赖性激酶 9 抑制剂在慢性淋巴细胞白血病小鼠模型中表现出强效抗白血病活性

Joachim R Göthert, Roze Imsak, Michael Möllmann, Stefanie Kesper, Maria Göbel, Ulrich Dührsen, Arne Scholz, Ulrich Lücking, Matthias Baumann, Anke Unger, Carsten Schultz-Fademrecht, Bert Klebl, Jan Eickhoff, Axel Choidas, Jan Dürig

Systematic Kinase Inhibitor Profiling Identifies CDK9 as a Synthetic Lethal Target in NUT Midline Carcinoma

系统性激酶抑制剂谱分析发现 CDK9 是 NUT 中线癌的合成致死靶点

Brägelmann, Johannes; Dammert, Marcel A; Dietlein, Felix; Heuckmann, Johannes M; Choidas, Axel; Böhm, Stefanie; Richters, André; Basu, Debjit; Tischler, Verena; Lorenz, Carina; Habenberger, Peter; Fang, Zhizhou; Ortiz-Cuaran, Sandra; Leenders, Frauke; Eickhoff, Jan; Koch, Uwe; Getlik, Matthäus; Termathe, Martin; Sallouh, Muhammad; Greff, Zoltán; Varga, Zoltán; Balke-Want, Hyatt; French, Christopher A; Peifer, Martin; Reinhardt, H Christian; Örfi, László; Kéri, György; Ansén, Sascha; Heukamp, Lukas C; Büttner, Reinhard; Rauh, Daniel; Klebl, Bert M; Thomas, Roman K; Sos, Martin L

Immunohistochemical Investigation of HER/AKT/mTOR Pathway and Cellular Adhesion Molecules in Urothelial Carcinomas

尿路上皮癌中HER/AKT/mTOR通路和细胞粘附分子的免疫组织化学研究

Koletsas, Nikolaos; Koletsa, Triantafyllia; Choidas, Spyros; Anagnostopoulos, Konstantinos; Touloupidis, Stavros; Zaramboukas, Thomas; Raptou, Georgia; Papadopoulos, Nikolaos; Lambropoulou, Maria