日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fluorine-18-Labeled Nucleotide Analogs Targeting Ecto-5'-Nucleotidase (CD73) for Positron Emission Tomography Imaging of Solid Tumors

用于实体瘤正电子发射断层扫描成像的靶向胞外5'-核苷酸酶(CD73)的氟-18标记核苷酸类似物

Dobelmann, Clemens; Schmies, Constanze C; Rolshoven, Georg Wilhelm; Scortichini, Mirko; Wagner, Stefan; Isaak, Andreas; Idris, Riham M; Dabel, Jennifer; Grey, Lucie; Losenkova, Karolina; Moschütz, Susanne; Hroub, Haneen Al; Keim, Antje; Höppner, Sandra; Sandholm, Jouko; Boström, Pia; Hollmén, Maija; Sträter, Norbert; Hermann, Sven; Yegutkin, Gennady G; Jacobson, Kenneth A; Schelhaas, Sonja; Müller, Christa E; Junker, Anna

Oncostatin M upregulates CD73 via the MAPK pathway in keratinocytes to promote an adenosine-dependent anti-inflammatory response in psoriasis

抑癌素M通过MAPK通路上调角质形成细胞中的CD73,从而促进银屑病中腺苷依赖性抗炎反应。

Giraulo, Caterina; De Palma, Giacomo; Plaitano, Paola; Esposito, Roberta; Morretta, Elva; Monti, Maria Chiara; Müller, Christa E; Cicala, Carla; Morello, Silvana

Pleiotropic genes linking congenital hypogonadotropic hypogonadism and cleft lip/palate: evidence from a genomic CHH cohort study

多效性基因与先天性促性腺激素低下症和唇腭裂相关:来自基因组CHH队列研究的证据

Correa, Fernanda de Azevedo; Habibi, Imen; Zhai, Jing; Adamo, Michela; Wang, Yi; Boizot, Alexia; Zouaghi, Yassine; Rauch, Anita; Pekic, Sandra; Quinton, Richard; Bonomi, Marco; Cangiano, Biagio; Dhillo, Waljit S; Fluck, Christa E; Nemeth, Attila; Bouloux, Pierre-Marc; Ferrara, Jean-Marc; Pignatelli, Duarte; Halász, Zita; Perdices-Lopez, Cecilia; Messina, Andrea; Niederländer, Nicolas J; Santoni, Federico; Acierno, James S; Pitteloud, Nelly

Phytochemical Screening of 45-Million-Year-Old Colored Angiosperm Leaves Reveals Distinctive Chlorophyll-Derived and Polyphenolic Pigments

对4500万年前有色被子植物叶片的植物化学筛选揭示了独特的叶绿素衍生色素和多酚色素

Wolkenstein, Klaus; Müller, Christa E; Engeser, Marianne; Frauendorf, Holm; McCoy, Victoria E; Gee, Carole T

A brain-penetrant P2X7R antagonist mitigates Alzheimer's disease pathology

一种能穿透血脑屏障的P2X7R拮抗剂可减轻阿尔茨海默病病理。

Turcu, Andreea L; Oken, Adam C; Griñán-Ferré, Christian; Durner, Anna; Sierra-Marquez, Juan; Hinz-Kowalik, Sonja; Nagel, Jessica; Lee, So-Deok; Tzortzini, Efpraxia; Georgiou, Kyriakos; Bhol, Mamina; Baz, Zuriñe; Llop, Jordi; Schneider, Marion; Barbaraci, Carla; Kim, Ga-Ram; Barniol-Xicota, Marta; Val, Cristina; Brea, José; Loza, M Isabel; Pérez, Belén; Naesens, Lieve; Kolocouris, Antonios; Kim, Yong-Chul; Müller, Christa E; Nicke, Annette; Pallàs, Mercè; Mansoor, Steven E; Vázquez, Santiago

Subnanomolar MAS-related G protein-coupled receptor-X2/B2 antagonists with efficacy in human mast cells and disease models

亚纳摩尔级MAS相关G蛋白偶联受体X2/B2拮抗剂,对人肥大细胞和疾病模型均有效

Ghazl Al Hamwi # ,Mohamad Wessam Alnouri # ,Sven Verdonck # ,Piotr Leonczak ,Shaswati Chaki ,Stefan Frischbutter ,Pavel Kolkhir ,Michaela Matthey ,Constantin Kopp ,Marek Bednarski ,Yvonne K Riedel ,Daniel Marx ,Sophie Clemens ,Vigneshwaran Namasivayam ,Susanne Gattner ,Dominik Thimm ,Katharina Sylvester ,Katharina Wolf ,Andreas E Kremer ,Steven De Jonghe ,Daniela Wenzel ,Magdalena Kotańska ,Hydar Ali ,Piet Herdewijn ,Christa E Müller

A polycyclic scaffold identified by structure-based drug design effectively inhibits the human P2X7 receptor

基于结构的药物设计鉴定出的一种多环骨架能有效抑制人P2X7受体。

Oken, Adam C; Turcu, Andreea L; Tzortzini, Eva; Georgiou, Kyriakos; Nagel, Jessica; Westermann, Franka G; Barniol-Xicota, Marta; Seidler, Jonas; Kim, Ga-Ram; Lee, So-Deok; Nicke, Annette; Kim, Yong-Chul; Müller, Christa E; Kolocouris, Antonios; Vázquez, Santiago; Mansoor, Steven E

Discovery of an allosteric binding site for anthraquinones at the human P2X4 receptor

在人P2X4受体上发现蒽醌的变构结合位点

Nagel, Jessica; Namasivayam, Vigneshwaran; Weinhausen, Stephanie; Sierra-Marquez, Juan; Baqi, Younis; Al Musawi, Hashem Ali M; Abdelrahman, Aliaa; Vaaßen, Victoria J; Schlegel, Jonathan G; Taplick, Lisa; Torp, Jane; Kubicek, Jan; Maertens, Barbara; Geyer, Matthias; Claff, Tobias; Nicke, Annette; Hagelueken, Gregor; Müller, Christa E

Psychedelics and Entactogens: Call for Papers

迷幻剂和致幻剂:征稿启事

Aljadeff, Johnatan; Lansdell, Benjamin J; Fairhall, Adrienne L; Kleinfeld, David; Lindsley, Craig W; Hooker, Jacob M; Chibale, Kelly; Müller, Christa E; Booker, Squire J

Call for Papers – Purinergic Signaling: Medicinal Chemistry, Biology, Pharmacology, and Translation into Diagnostic and Therapeutic Drugs

征稿启事——嘌呤能信号传导:药物化学、生物学、药理学及其在诊断和治疗药物中的转化应用

Yang, Song; Sun, Yiran; Yan, Chenchen; Müller, Christa E; Nicke, Annette; Lohr, Christian; Freichel, Marc; Guse, Andreas H