Synthesis, inverse docking-assisted identification and in vitro biological characterization of Flavonol-based analogs of fisetin as c-Kit, CDK2 and mTOR inhibitors against melanoma and non-melanoma skin cancers
合成、逆向对接辅助鉴定和体外生物学表征基于黄酮醇的fisetin类似物作为c-Kit、CDK2和mTOR抑制剂对抗黑色素瘤和非黑色素瘤皮肤癌
期刊:Bioorganic Chemistry
影响因子:4.5
doi:10.1016/j.bioorg.2020.104595
Tithi Roy, Samuel T Boateng, Sergette Banang-Mbeumi, Pankaj K Singh, Pratik Basnet, Roxane-Cherille N Chamcheu, Federico Ladu, Isabel Chauvin, Vladimir S Spiegelman, Ronald A Hill, Konstantin G Kousoulas, Bolni Marius Nagalo, Anthony L Walker, Jean Fotie, Siva Murru, Mario Sechi, Jean Christopher Ch