日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Prophylactic treatment with the c-Abl inhibitor, neurotinib, diminishes neuronal damage and the convulsive state in pilocarpine-induced mice

使用 c-Abl 抑制剂 Neurotinib 进行预防性治疗可减轻毛果芸香碱诱导小鼠的神经元损伤和惊厥状态。

América Chandía-Cristi,Daniela A Gutiérrez,Andrés E Dulcey,Marcelo Lara,Lina Vargas,Yi-Han Lin,Pablo Jimenez-Muñoz,Gabriela Larenas,Xin Xu,Amy Wang,Ashley Owens,Christopher Dextras,YuChi Chen,Claudio Pinto,Tamara Marín,Hugo Almarza-Salazar,Keryma Acevedo,Gonzalo I Cancino,Xin Hu,Patricio Rojas,Marc Ferrer,Noel Southall,Mark J Henderson,Silvana Zanlungo,Juan J Marugan,Alejandra Álvarez R

Discovery and Optimization of Pyrrolopyrimidine Derivatives as Selective Disruptors of the Perinucleolar Compartment, a Marker of Tumor Progression toward Metastasis

发现并优化吡咯并嘧啶衍生物作为核仁周围区室的选择性破坏剂(肿瘤向转移发展的标志)

Kevin J Frankowski, Samarjit Patnaik, Chen Wang, Noel Southall, Dipannita Dutta, Soumitta De, Dandan Li, Christopher Dextras, Yi-Han Lin, Marthe Bryant-Connah, Danielle Davis, Feijun Wang, Leah M Wachsmuth, Pranav Shah, Jordan Williams, Md Kabir, Edward Zhu, Bolormaa Baljinnyam, Amy Wang, Xin Xu, Jo

Discovery of small molecule inhibitors that effectively disrupt IQGAP1-Cdc42 interaction in breast cancer cells

发现可有效破坏乳腺癌细胞中 IQGAP1-Cdc42 相互作用的小分子抑制剂

Samar Sayedyahossein, Jessica Smith, Elena Barnaeva, Zhigang Li, Jun Choe, Michael Ronzetti, Christopher Dextras, Xin Hu, Juan Marugan, Noel Southall, Bolormaa Baljinnyam, Louise Thines, Andy D Tran, Marc Ferrer, David B Sacks

Identification of Small Molecule Enhancers of Immunotherapy for Melanoma

黑色素瘤免疫治疗小分子增强剂的鉴定

Christopher Dextras, Myagmarjav Dashnyam, Lesley A Mathews Griner, Janani Sundaresan, Bryan Chim, Zhiya Yu, Suman Vodnala, Chyi-Chia Richard Lee, Xin Hu, Noel Southall, Juan J Marugan, Ajit Jadhav, Nicholas P Restifo, Nicolas Acquavella, Marc Ferrer, Anju Singh

Pharmacokinetic evaluation of the PNC disassembler metarrestin in wild-type and Pdx1-Cre;LSL-KrasG12D/+;Tp53R172H/+ (KPC) mice, a genetically engineered model of pancreatic cancer

PNC 分解剂 metarrestin 在野生型和 Pdx1-Cre;LSL-KrasG12D/+;Tp53R172H/+ (KPC) 小鼠(一种胰腺癌基因工程模型)中的药代动力学评估

Tomas Vilimas, Amy Q Wang, Samarjit Patnaik, Emma A Hughes, Marc D Singleton, Zachary Knotts, Dandan Li, Kevin Frankowski, Jerome J Schlomer, Theresa M Guerin, Stephanie Springer, Catherine Drennan, Christopher Dextras, Chen Wang, Debra Gilbert, Noel Southall, Marc Ferrer, Sui Huang, Serguei Kozlov,