日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Critical assessment of LC3/GABARAP ligands used for degrader development and ligandability of LC3/GABARAP binding pockets

对用于降解剂开发的 LC3/GABARAP 配体和 LC3/GABARAP 结合位点的配体能力进行严格评估

Martin P Schwalm, Johannes Dopfer, Adarsh Kumar, Francesco A Greco, Nicolas Bauer, Frank Löhr, Jan Heering, Sara Cano-Franco, Severin Lechner, Thomas Hanke, Ivana Jaser, Viktoria Morasch, Christopher Lenz, Daren Fearon, Peter G Marples, Charles W E Tomlinson, Lorene Brunello, Krishna Saxena, Nathan

K48- and K63-linked ubiquitin chain interactome reveals branch- and length-specific ubiquitin interactors

K48 和 K63 连接的泛素链相互作用组揭示了分支和长度特异性的泛素相互作用物

Anita Waltho, Oliver Popp, Christopher Lenz, Lukas Pluska, Mahil Lambert, Volker Dötsch, Philipp Mertins, Thomas Sommer

Back-pocket optimization of 2-aminopyrimidine-based macrocycles leads to potent dual EPHA2/GAK kinase inhibitors with antiviral activity

对 2-氨基嘧啶大环化合物进行后袋优化,可得到具有抗病毒活性的强效双重 EPHA2/GAK 激酶抑制剂

Joshua Gerninghaus, Rezart Zhubi, Andreas Krämer, Marwah Karim, Do Hoang Nhu Tran, Andreas C Joerger, Christian Schreiber, Lena M Berger, Benedict-Tilman Berger, Theresa A L Ehret, Lewis Elson, Christopher Lenz, Krishna Saxena, Susanne Müller, Shirit Einav, Stefan Knapp, Thomas Hanke