The G Protein Biased Small Molecule Apelin Agonist CMF-019 is Disease Modifying in Endothelial Cell Apoptosis In Vitro and Induces Vasodilatation Without Desensitisation In Vivo
蛋白偏向的小分子 Apelin 激动剂 CMF-019 可在体外改善内皮细胞凋亡,并在体内诱导血管扩张而不产生脱敏作用
期刊:Frontiers in Pharmacology
影响因子:4.4
doi:10.3389/fphar.2020.588669
Cai Read, Duuamene Nyimanu, Peiran Yang, Rhoda E Kuc, Thomas L Williams, Christopher M Fitzpatrick, Richard Foster, Robert C Glen, Janet J Maguire, Anthony P Davenport