日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Next-generation rifamycins for the treatment of mycobacterial infections

用于治疗分枝杆菌感染的新一代利福霉素

Dartois, Véronique; Lan, Tian; Ganapathy, Uday S; Wong, Chui Fann; Sarathy, Jickky P; Jimenez, Diana C; Alshiraihi, Ilham M; Lam, Ha; Rodriguez, Suyapa; Xie, Min; Soto-Ojeda, Maritza; Jackson, Mary; Wheat, William; Dillman, Nathan C; Kostenkova, Kateryna; Schmitt, Jake; Mann, Lea; Richter, Adrian; Imming, Peter; Sarathy, Jansy; Kaya, Firat; Paruchuri, Sindhuja; Tatek, Betelhem; Folvar, Camilla; Proietto, Julianna; Zimmerman, Matthew; Gonzalez-Juarrero, Mercedes; Aldrich, Courtney C; Dick, Thomas

Cryo-EM reveals transition states of the Acinetobacter baumannii F(1)-ATPase rotary subunits γ and ε, unveiling novel compound targets

冷冻电镜揭示了鲍曼不动杆菌F(1)-ATPase旋转亚基γ和ε的过渡态,并发现了新的化合物靶点。

Le, Khoa Cong Minh; Wong, Chui Fann; Müller, Volker; Grüber, Gerhard

Cryo-Electron Microscopy Structure of the Mycobacterium tuberculosis Cytochrome bcc:aa(3) Supercomplex and a Novel Inhibitor Targeting Subunit Cytochrome cI

结核分枝杆菌细胞色素bcc:aa(3)超复合物的冷冻电镜结构及靶向亚基细胞色素cI的新型抑制剂

Mathiyazakan, Vikneswaran; Wong, Chui-Fann; Harikishore, Amaravadhi; Pethe, Kevin; Grüber, Gerhard

Structural Elements Involved in ATP Hydrolysis Inhibition and ATP Synthesis of Tuberculosis and Nontuberculous Mycobacterial F-ATP Synthase Decipher New Targets for Inhibitors

结核分枝杆菌和非结核分枝杆菌F-ATP合酶中参与ATP水解抑制和ATP合成的结构元件揭示抑制剂的新靶点

Wong, Chui Fann; Saw, Wuan-Geok; Basak, Sandip; Sano, Mio; Ueno, Hiroshi; Kerk, Hwee Wen; Litty, Dennis; Ragunathan, Priya; Dick, Thomas; Müller, Volker; Noji, Hiroyuki; Grüber, Gerhard

Atomic solution structure of Mycobacterium abscessus F-ATP synthase subunit ε and identification of Ep1MabF1 as a targeted inhibitor

脓肿分枝杆菌F-ATP合酶亚基ε的原子溶液结构及Ep1MabF1作为靶向抑制剂的鉴定

Shin, Joon; Harikishore, Amaravadhi; Wong, Chui Fann; Ragunathan, Priya; Dick, Thomas; Grüber, Gerhard

Targeting Mycobacterial F-ATP Synthase C-Terminal α Subunit Interaction Motif on Rotary Subunit γ

靶向分枝杆菌F-ATP合酶C端α亚基与旋转亚基γ相互作用的基序

Harikishore, Amaravadhi; Wong, Chui-Fann; Ragunathan, Priya; Litty, Dennis; Müller, Volker; Grüber, Gerhard

The Unique C-Terminal Extension of Mycobacterial F-ATP Synthase Subunit α Is the Major Contributor to Its Latent ATP Hydrolysis Activity

分枝杆菌F-ATP合酶亚基α独特的C端延伸是其潜在ATP水解活性的主要贡献者。

Wong, Chui-Fann; Grüber, Gerhard