日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Clonazepam activates the transient receptor potential melastatin 8 (TRPM8) ion channel

氯硝西泮激活瞬时受体电位melastatin 8 (TRPM8)离子通道

Elkin, Logan; Chulkov, Evgeny G; Enders, Jonathan; Menzel, Anthony D; Park, Sang-Kyu; Stucky, Cheryl L; Marchant, Jonathan S

Target-based discovery of a broad-spectrum flukicide.

基于靶点的广谱杀吸虫剂的发现

Sprague Daniel J, Park Sang-Kyu, Gramberg Svenja, Bauer Lisa, Rohr Claudia M, Chulkov Evgeny G, Smith Emery, Scampavia Louis, Spicer Timothy P, Haeberlein Simone, Marchant Jonathan S

The anthelmintic meclonazepam activates a schistosome transient receptor potential channel

驱虫药美氯硝西泮可激活血吸虫瞬时受体电位通道。

Park, Sang-Kyu; Sprague, Daniel J; Rohr, Claudia M; Chulkov, Evgeny G; Petrow, Ian; Kumar, Sushil; Marchant, Jonathan S

Use the force, fluke: Ligand-independent gating of Schistosoma mansoni ion channel TRPM(PZQ)

利用原力,侥幸:曼氏血吸虫离子通道 TRPM(PZQ) 的配体非依赖性门控

Chulkov, Evgeny G; Isaeva, Elena; Stucky, Cheryl L; Marchant, Jonathan S

Electrophysiological characterization of a schistosome transient receptor potential channel activated by praziquantel

吡喹酮激活血吸虫瞬时受体电位通道的电生理特性

Chulkov, Evgeny G; Palygin, Oleg; Yahya, Nawal A; Park, Sang-Kyu; Marchant, Jonathan S

Praziquantel activates a native cation current in Schistosoma mansoni

吡喹酮激活曼氏血吸虫体内的固有阳离子电流

Chulkov, Evgeny G; Rohr, Claudia M; Marchant, Jonathan S

Target-based discovery of a broad spectrum flukicide.

基于靶点的广谱杀吸虫剂的发现

Sprague Daniel J, Park Sang-Kyu, Gramberg Svenja, Bauer Lisa, Rohr Claudia M, Chulkov Evgeny G, Smith Emery, Scampavia Louis, Spicer Timothy P, Haeberlein Simone, Marchant Jonathan S

Loss of Chloride Channel 6 (CLC-6) Affects Vascular Smooth Muscle Contractility and Arterial Stiffness via Alterations to Golgi Calcium Stores

氯离子通道6 (CLC-6) 的缺失通过改变高尔基体钙储存影响血管平滑肌收缩性和动脉僵硬度

Klemens, Christine A; Chulkov, Evgeny G; Wu, Jing; Hye Khan, Md Abdul; Levchenko, Vladislav; Flister, Michael J; Imig, John D; Kriegel, Alison J; Palygin, Oleg; Staruschenko, Alexander

Identification of novel modulators of a schistosome transient receptor potential channel targeted by praziquantel

鉴定吡喹酮靶向的血吸虫瞬时受体电位通道的新型调节剂

Chulkov, Evgeny G; Smith, Emery; Rohr, Claudia M; Yahya, Nawal A; Park, Sang-Kyu; Scampavia, Louis; Spicer, Timothy P; Marchant, Jonathan S

The anthelmintic drug praziquantel activates a schistosome transient receptor potential channel

驱虫药吡喹酮可激活血吸虫瞬时受体电位通道。

Park, Sang-Kyu; Gunaratne, Gihan S; Chulkov, Evgeny G; Moehring, Francie; McCusker, Paul; Dosa, Peter I; Chan, John D; Stucky, Cheryl L; Marchant, Jonathan S