日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

The E3-ome gene-centric compendium reveals the human E3 ligase landscape.

以 E3 连接酶组为中心的基因汇编揭示了人类 E3 连接酶的全貌。

Chua Ngee Kiat, González-Robles Tania J, Reddington Cameron J, Dudley-Fraser Jane, Birkinshaw Richard W, Han Jiru, Solano Ashleigh, Wong Soon Wei, Kochańczyk Tomasz, Peter Joshua J, Nakasone Mark A, Aust Florian, Munro Jacob, Tong Yeh Huei, Iskander Julie, Abeysekera Waruni, Garnham Alex, Huckstep Hannah, Ritchie Matthew E, Wertz Ingrid, Hymowitz Sarah, Kumar Sharad, Conaway Ron C, Privé Gilbert G, Bullock Alex N, Babon Jeffrey J, Klevit Rachel E, Lorenz Sonja, Ciulli Alessio, Fischer Eric S, Thomä Nicolas H, Nowak Radosław P, Schulman Brenda A, Rapé Michael, Rittinger Katrin, Pagan Julia K, Bahlo Melanie, Mackay Joel P, Mace Peter D, Lima Christopher D, Hay Ronald T, Komander David, Lechtenberg Bernhard C, Joazeiro Claudio A P, Pagano Michele, Hofmann Kay, Feltham Rebecca

Allosteric PROTACs: Expanding the Horizon of Targeted Protein Degradation

变构PROTACs:拓展靶向蛋白降解的视野

Frost, Aileen; O'Connor, Suzanne; Ciulli, Alessio

Viral Encephalopathy and Retinopathy in Dusky Groupers (Epinephelus marginatus, Lowe 1834) from Two Marine Protected Areas of the Northern Mediterranean Sea

来自北地中海两个海洋保护区的暗色石斑鱼(Epinephelus marginatus, Lowe 1834)的病毒性脑病和视网膜病变

Volpe, Enrico; Mandrioli, Luciana; Napolitano, Riccardo; Hartmann, Manuel Garcia; Merotto, Lorenzo; Girons, Albert; Errani, Francesca; Brunetti, Barbara; Capoccioni, Fabrizio; Ciulli, Sara

Frustration in the protein-protein interface plays a central role in the cooperativity of PROTAC ternary complexes

蛋白质-蛋白质界面处的相互作用受阻在PROTAC三元复合物的协同作用中起着核心作用。

Ma, Ning; Bhattacharya, Supriyo; Muk, Sanychen; Jandova, Zuzana; Schmalhorst, Philipp S; Ghosh, Soumadwip; Le, Keith; Diers, Emelyne; Trainor, Nicole; Farnaby, William; Roy, Michael J; Kofink, Christiane; Greb, Peter; Weinstabl, Harald; Ciulli, Alessio; Bader, Gerd; Sankar, Kyra; Bergner, Andreas; Vaidehi, Nagarajan

Rational Design of PROTAC Linkers Featuring Ferrocene as a Molecular Hinge to Enable Dynamic Conformational Changes

以二茂铁为分子铰链的PROTAC连接子的合理设计,以实现动态构象变化

Salerno, Alessandra; Wieske, Lianne H E; Diehl, Claudia J; Ciulli, Alessio

Identification of a Highly Cooperative PROTAC Degrader Targeting GTP-Loaded KRAS(On) Alleles

鉴定一种高度协同的PROTAC降解酶,该酶靶向GTP结合的KRAS(On)等位基因

Vetma, Vesna; Puoti, Ilaria; Karolak, Natalia K; Chakraborti, Sohini; Diers, Emelyne; Girardi, Enrico; Khan, Shakil; Kidd, Giorgia; Kropatsch, Katrin G; Mclennan, Ross; O'Connor, Suzanne; Samwer, Matthias; Trainor, Nicole; Whitworth, Claire; Wijaya, Andre J; Wong, Jeff Y F; Zollman, David; Farnaby, William; Popow, Johannes; Ciulli, Alessio; Ettmayer, Peter; McAulay, Kirsten

Macrocycle-based PROTACs selectively degrade cyclophilin A and inhibit HIV-1 and HCV

基于大环化合物的PROTACs选择性降解亲环蛋白A,并抑制HIV-1和HCV病毒。

Lydia S Newton # ,Clara Gathmann # ,Sophie Ridewood ,Robert J Smith ,Andre J Wijaya ,Thomas W Hornsby ,Kate L Morling ,Dara Annett ,Riccardo Zenezini Chiozzi ,Ann-Kathrin Reuschl ,Morten L Govasli ,Ying Ying Tan ,Lucy G Thorne ,Clare Jolly ,Konstantinos Thalassinos ,Alessio Ciulli ,Greg J Towers ,David L Selwood

Mode of action of a DCAF16-recruiting targeted glue that can selectively degrade BRD9

能够选择性降解BRD9的DCAF16募集靶向胶的作用机制

Scott J Hughes ,Wojciech J Stec ,Colin T R Davies ,David McGarry ,Alicia Williams ,Marta Carrara ,Ivan Del Barco Barrantes ,Rebecca Harris ,Anna Tasegian ,Dominic D G Owens ,Alexander Fawcett ,John Hellicar ,Aleksandra Azevedo ,Gregor P Meier ,Andrew C Runcie ,Liliana Greger ,Martin O'Rourke ,Ian Churcher ,Martin Pass ,Giles A Brown ,Alessio Ciulli ,Louise K Modis ,Andrea Testa

A method for the detection and enrichment of endogenous cereblon substrates

一种检测和富集内源性cereblon底物的方法

Hannah C Lloyd ,Yuli Li ,N Connor Payne ,Zhenguang Zhao ,Wenqing Xu ,Alena Kroupova ,David Zollman ,Tengfang Long ,Farah Kabir ,Mei Chen ,Rebecca Freeman ,Ethan Yang Feng ,Sarah Y Xi ,Ya-Chieh Hsu ,Alessio Ciulli ,Ralph Mazitschek ,Christina M Woo

Reweighting simulated events using machine-learning techniques in the CMS experiment

在CMS实验中使用机器学习技术对模拟事件进行重新加权

Hayrapetyan, A; Tumasyan, A; Adam, W; Andrejkovic, J W; Benato, L; Bergauer, T; Chatterjee, S; Damanakis, K; Dragicevic, M; Hussain, P S; Jeitler, M; Krammer, N; Li, A; Liko, D; Mikulec, I; Schieck, J; Schöfbeck, R; Schwarz, D; Sonawane, M; Waltenberger, W; Wulz, C-E; Janssen, T; Van Laer, T; Van Mechelen, P; Breugelmans, N; D'Hondt, J; Dansana, S; De Moor, A; Delcourt, M; Heyen, F; Lowette, S; Makarenko, I; Müller, D; Tavernier, S; Tytgat, M; Van Onsem, G P; Van Putte, S; Vannerom, D; Bilin, B; Clerbaux, B; Das, A K; De Bruyn, I; De Lentdecker, G; Evard, H; Favart, L; Gianneios, P; Jaramillo, J; Khalilzadeh, A; Khan, F A; Lee, K; Malara, A; Paredes, S; Shahzad, M A; Thomas, L; Vanden Bemden, M; Vander Velde, C; Vanlaer, P; De Coen, M; Dobur, D; Gokbulut, G; Hong, Y; Knolle, J; Lambrecht, L; Marckx, D; Mota Amarilo, K; Skovpen, K; Van Den Bossche, N; van der Linden, J; Wezenbeek, L; Benecke, A; Bethani, A; Bruno, G; Caputo, C; De Favereau De Jeneret, J; Delaere, C; Donertas, I S; Giammanco, A; 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Spah, J L; Stein, A; Torres Da Silva De Araujo, F; Wiedenbeck, S; Zaleski, S; Dziwok, C; Flügge, G; Kress, T; Nowack, A; Pooth, O; Stahl, A; Ziemons, T; Zotz, A; Aarup Petersen, H; Aldaya Martin, M; Alimena, J; Amoroso, S; An, Y; Bach, J; Baxter, S; Bayatmakou, M; Becerril Gonzalez, H; Behnke, O; Belvedere, A; Blekman, F; Borras, K; Campbell, A; Cardini, A; Cheng, C; Colombina, F; Eckerlin, G; Eckstein, D; Estevez Banos, L I; Gallo, E; Geiser, A; Guglielmi, V; Guthoff, M; Hinzmann, A; Jeppe, L; Kaech, B; Kasemann, M; Kleinwort, C; Kogler, R; Komm, M; Krücker, D; Lange, W; Leyva Pernia, D; Lipka, K; Lohmann, W; Lorkowski, F; Mankel, R; Melzer-Pellmann, I-A; Mendizabal Morentin, M; Meyer, A B; Milella, G; Moral Figueroa, K; Mussgiller, A; Nair, L P; Niedziela, J; Nürnberg, A; Otarid, Y; Park, J; Ranken, E; Raspereza, A; Rastorguev, D; Rübenach, J; Rygaard, L; Saggio, A; Scham, M; Schnake, S; Schütze, P; Schwanenberger, C; Selivanova, D; Sharko, K; Shchedrolosiev, M; Stafford, D; Vazzoler, F; 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