日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of an allosteric binding site for anthraquinones at the human P2X4 receptor

在人P2X4受体上发现蒽醌的变构结合位点

Nagel, Jessica; Namasivayam, Vigneshwaran; Weinhausen, Stephanie; Sierra-Marquez, Juan; Baqi, Younis; Al Musawi, Hashem Ali M; Abdelrahman, Aliaa; Vaaßen, Victoria J; Schlegel, Jonathan G; Taplick, Lisa; Torp, Jane; Kubicek, Jan; Maertens, Barbara; Geyer, Matthias; Claff, Tobias; Nicke, Annette; Hagelueken, Gregor; Müller, Christa E

Structural basis for lipid-mediated activation of G protein-coupled receptor GPR55

脂质介导的 G 蛋白偶联受体 GPR55 激活的结构基础

Tobias Claff, Rebecca Ebenhoch, Jörg T Kley, Aniket Magarkar, Herbert Nar, Dietmar Weichert

Development of an active-site titrant for SARS-CoV-2 main protease as an indispensable tool for evaluating enzyme kinetics

开发 SARS-CoV-2 主蛋白酶活性位点滴定剂作为评估酶动力学不可或缺的工具

Rabea Voget, Julian Breidenbach, Tobias Claff, Alexandra Hingst, Katharina Sylvester, Christian Steinebach, Lan Phuong Vu, Renato H Weiße, Ulrike Bartz, Norbert Sträter, Christa E Müller, Michael Gütschow

Macrocyclic Azapeptide Nitriles: Structure-Based Discovery of Potent SARS-CoV-2 Main Protease Inhibitors as Antiviral Drugs

大环氮杂肽腈:基于结构发现有效的 SARS-CoV-2 主要蛋白酶抑制剂作为抗病毒药物

Julian Breidenbach, Rabea Voget, Yaoyao Si, Alexandra Hingst, Tobias Claff, Katharina Sylvester, Valentina Wolf, Vesa Krasniqi, Abibe Useini, Norbert Sträter, Yukino Ogura, Atsushi Kawaguchi, Christa E Müller, Michael Gütschow

Structural Insights into Partial Activation of the Prototypic G Protein-Coupled Adenosine A(2A) Receptor

原型G蛋白偶联腺苷A(2A)受体部分激活的结构解析

Claff, Tobias; Mahardhika, Andhika B; Vaaßen, Victoria J; Schlegel, Jonathan G; Vielmuth, Christin; Weiße, Renato H; Sträter, Norbert; Müller, Christa E

Crystal structure of adenosine A(2A) receptor in complex with clinical candidate Etrumadenant reveals unprecedented antagonist interaction.

腺苷 A(2A) 受体与临床候选药物 Etrumadenant 复合物的晶体结构揭示了前所未有的拮抗剂相互作用

Claff Tobias, Schlegel Jonathan G, Voss Jan H, Vaaßen Victoria J, Weiße Renato H, Cheng Robert K Y, Markovic-Mueller Sandra, Bucher Denis, Sträter Norbert, Müller Christa E

Single Stabilizing Point Mutation Enables High-Resolution Co-Crystal Structures of the Adenosine A(2A) Receptor with Preladenant Conjugates.

单个稳定点突变可实现腺苷 A(2A) 受体与前腺苷缀合物的高分辨率共晶结构

Claff Tobias, Klapschinski Tim A, Tiruttani Subhramanyam Udaya K, Vaaßen Victoria J, Schlegel Jonathan G, Vielmuth Christin, Voß Jan H, Labahn Jörg, Müller Christa E

Irreversible Antagonists for the Adenosine A2B Receptor

腺苷 A2B 受体的不可逆拮抗剂

Ahmed Temirak, Jonathan G Schlegel, Jan H Voss, Victoria J Vaaßen, Christin Vielmuth, Tobias Claff, Christa E Müller

Elucidating the active δ-opioid receptor crystal structure with peptide and small-molecule agonists

利用肽和小分子激动剂阐明活性δ-阿片受体晶体结构

Tobias Claff, Jing Yu, Véronique Blais, Nilkanth Patel, Charlotte Martin, Lijie Wu, Gye Won Han, Brian J Holleran, Olivier Van der Poorten, Kate L White, Michael A Hanson, Philippe Sarret, Louis Gendron, Vadim Cherezov, Vsevolod Katritch, Steven Ballet, Zhi-Jie Liu, Christa E Müller, Raymond C Steve

The quality of diabetic care in a London health district

伦敦某卫生区的糖尿病护理质量

Yudkin, J S; Boucher, B J; Schopflin, K E; Harris, B T; Claff, H R; Whyte, N J; Taylor, B; Mellins, D H; Wootliff, A B; Safir, J G; Jones, E J