文献库，生知库 | 链接生命科学的每一步

日期影响因子

Explorations of Agonist Selectivity for the α9* nAChR with Novel Substituted Carbamoyl/Amido/Heteroaryl Dialkylpiperazinium Salts and Their Therapeutic Implications in Pain and Inflammation

探索新型取代的氨基甲酰基/酰胺基/杂芳基二烷基哌嗪盐对 α9* nAChR 的激动剂选择性及其在疼痛和炎症中的治疗意义

期刊:Journal of Medicinal Chemistry

影响因子:6.8

doi:10.1021/acs.jmedchem.3c02429

Hina Andleeb, Roger L Papke, Clare Stokes, Katrin Richter, Sara M Herz, Ka Chiang, Siva R Raju Kanumuri, Abhisheak Sharma, M Imad Damaj, Veronika Grau, Nicole A Horenstein, Ganesh A Thakur

Immunology/Inflammation

发表日期：2024

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New Alpha9 nAChR Ligands Based on a 5-(Quinuclidin-3-ylmethyl)-1,2,4-oxadiazole Scaffold

基于 5-(奎宁环-3-基甲基)-1,2,4-恶二唑骨架的新型 Alpha9 nAChR 配体

期刊:ACS Chemical Neuroscience

影响因子:4.1

doi:10.1021/acschemneuro.3c00720

Clelia Dallanoce, Katrin Richter, Clare Stokes, Claudio Papotto, Hina Andleeb, Ganesh A Thakur, Andrew Kerr, Veronika Grau, Roger L Papke

发表日期：2024

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Pharmacological profiles and anti-inflammatory activity of pCN-diEPP and mCN-diEPP, new alpha9alpha10 nicotinic receptor ligands

新型 alpha9alpha10 烟碱受体配体 pCN-diEPP 和 mCN-diEPP 的药理学特征和抗炎活性

期刊:Neuropharmacology

影响因子:4.6

doi:10.1016/j.neuropharm.2023.109717

Katrin Richter, Sara M Herz, Clare Stokes, M Imad Damaj, Veronika Grau, Roger L Papke

发表日期：2023

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Insights Into the Differential Desensitization of α 4 β 2 Nicotinic Acetylcholine Receptor Isoforms Obtained With Positive Allosteric Modulation of Mutant Receptors

通过突变受体的正向变构调节获得对 α 4 β 2 烟碱型乙酰胆碱受体异构体的差异脱敏的洞察

期刊:Molecular Pharmacology

影响因子:3.2

doi:10.1124/molpharm.122.000591

Roger L Papke, Clare Stokes

发表日期：2023

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Comparison of the Anti-inflammatory Properties of Two Nicotinic Acetylcholine Receptor Ligands, Phosphocholine and p CF3-diEPP

两种烟碱乙酰胆碱受体配体磷酸胆碱和 p CF3-diEPP 的抗炎特性比较

期刊:Frontiers in Cellular Neuroscience

影响因子:4.2

doi:10.3389/fncel.2022.779081

Katrin Richter, Roger L Papke, Clare Stokes, Danika C Roy, Eduardo S Espinosa, Philipp M K Wolf, Andreas Hecker, Juliane Liese, Vijay K Singh, Winfried Padberg, Klaus-Dieter Schlüter, Marius Rohde, J Michael McIntosh, Barbara J Morley, Nicole A Horenstein, Veronika Grau, Alain R Simard2

发表日期：2022

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Selective Agonists and Antagonists of α9 Versus α7 Nicotinic Acetylcholine Receptors

α9 与 α7 烟碱乙酰胆碱受体的选择性激动剂和拮抗剂

期刊:ACS Chemical Neuroscience

影响因子:4.1

doi:10.1021/acschemneuro.1c00747

Roger L Papke, Hina Andleeb, Clare Stokes, Marta Quadri, Nicole A Horenstein

发表日期：2022

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Differential Activation and Desensitization States Promoted by Noncanonical α 7 Nicotinic Acetylcholine Receptor Agonists

非经典 α7 烟碱乙酰胆碱受体激动剂促进的差异激活和脱敏状态

期刊:Journal of Pharmacology and Experimental Therapeutics

影响因子:3.1

doi:10.1124/jpet.122.001354

Clare Stokes, Gisela Andrea Camacho-Hernandez, Ganesh A Thakur, Xiaoxuan Wu, Palmer Taylor, Roger L Papke

发表日期：2022

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A scoping review protocol to map the evidence on the use of action research methodology by healthcare professionals and in healthcare team settings

一项范围界定审查方案，旨在梳理医疗保健专业人员和医疗保健团队中行动研究方法应用方面的证据。

期刊:HRB Open Research

doi:10.12688/hrbopenres.13275.1

Roberts, Kinley; Casey, Mary; Coghlan, David; Cornall, Catherine; Hudson, Clare; Stokes, Diarmuid; Carroll, Aine

发表日期：2021

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The Allosteric Activation of α7 nAChR by α-Conotoxin MrIC Is Modified by Mutations at the Vestibular Site

前庭部位的突变改变了 α-芋螺毒素 MrIC 对 α7 nAChR 的变构激活

doi:10.3390/toxins13080555

Alican Gulsevin, Roger L Papke, Clare Stokes, Hue N T Tran, Aihua H Jin, Irina Vetter, Jens Meiler

发表日期：2021

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Design, synthesis, and electrophysiological evaluation of NS6740 derivatives: Exploration of the structure-activity relationship for alpha7 nicotinic acetylcholine receptor silent activation

NS6740 衍生物的设计、合成和电生理学评价：探索 alpha7 烟碱乙酰胆碱受体静默激活的构效关系

期刊:European Journal of Medicinal Chemistry

doi:10.1016/j.ejmech.2020.112669

Maria Chiara Pismataro, Nicole A Horenstein, Clare Stokes, Marta Quadri, Marco De Amici, Roger L Papke, Clelia Dallanoce

发表日期：2020

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