Discovery of spirohydantoins as selective, orally bioavailable inhibitors of p300/CBP histone acetyltransferases
发现螺环乙内酰脲类化合物是选择性、口服生物利用度高的p300/CBP组蛋白乙酰转移酶抑制剂
期刊:Bioorganic & Medicinal Chemistry Letters
影响因子:2.2
doi:10.1016/j.bmcl.2021.127854
Ji, Zhiqin; Clark, Richard F; Bhat, Vikram; Matthew Hansen, T; Lasko, Loren M; Bromberg, Kenneth D; Manaves, Vlasios; Algire, Mikkel; Martin, Ruth; Qiu, Wei; Torrent, Maricel; Jakob, Clarissa G; Liu, Hong; Cole, Philip A; Marmorstein, Ronen; Kesicki, Edward A; Lai, Albert; Michaelides, Michael R