日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

DAG-MAG-ΒHB: A Novel Ketone Diester Modulates NLRP3 Inflammasome Activation in Microglial Cells in Response to Beta-Amyloid and Low Glucose AD-like Conditions

DAG-MAG-ΒHB:一种新型酮二酯调节小胶质细胞中 NLRP3 炎症小体活化以响应 β-淀粉样蛋白和低葡萄糖 AD 样条件

Valentina Gentili, Giovanna Schiuma, Latha Nagamani Dilliraj, Silvia Beltrami, Sabrina Rizzo, Djidjell Lara, Pier Paolo Giovannini, Matteo Marti, Daria Bortolotti, Claudio Trapella, Marco Narducci, Roberta Rizzo

1,3,8-Triazaspiro[4.5]decane Derivatives Inhibit Permeability Transition Pores through a FO-ATP Synthase c Subunit Glu119-Independent Mechanism That Prevents Oligomycin A-Related Side Effects

1,3,8-三氮杂螺[4.5]癸烷衍生物通过 FO-ATP 合酶 c 亚基 Glu119 非依赖性机制抑制通透性转换孔,从而预防寡霉素 A 相关副作用

Gaia Pedriali, Daniela Ramaccini, Esmaa Bouhamida, Alessio Branchini, Giulia Turrin, Elisabetta Tonet, Antonella Scala, Simone Patergnani, Mirko Pinotti, Claudio Trapella, Carlotta Giorgi, Elena Tremoli, Gianluca Campo, Giampaolo Morciano, Paolo Pinton

Synthesis and NLRP3-Inflammasome Inhibitory Activity of the Naturally Occurring Velutone F and of Its Non-Natural Regioisomeric Chalconoids

天然存在的 Velutone F 及其非天然区域异构体查尔酮的合成及其对 NLRP3 炎症小体的抑制活性

Tiziano De Ventura, Mariasole Perrone, Sonia Missiroli, Paolo Pinton, Paolo Marchetti, Giovanni Strazzabosco, Giulia Turrin, Davide Illuminati, Virginia Cristofori, Anna Fantinati, Martina Fabbri, Carlotta Giorgi, Claudio Trapella, Vinicio Zanirato

Xylitol as a Hydrophilization Moiety for a Biocatalytically Synthesized Ibuprofen Prodrug

木糖醇作为生物催化合成布洛芬前药的亲水化部分

Federico Zappaterra, Chiara Tupini, Daniela Summa, Virginia Cristofori, Stefania Costa, Claudio Trapella, Ilaria Lampronti, Elena Tamburini

Structure-Activity Relationship Studies on Oxazolo[3,4- a]pyrazine Derivatives Leading to the Discovery of a Novel Neuropeptide S Receptor Antagonist with Potent In Vivo Activity

对噁唑并[3,4- a]吡嗪衍生物进行构效关系研究,发现具有强效体内活性的新型神经肽 S 受体拮抗剂

Valentina Albanese, Chiara Ruzza, Erika Marzola, Tatiana Bernardi, Martina Fabbri, Anna Fantinati, Claudio Trapella, Rainer K Reinscheid, Federica Ferrari, Chiara Sturaro, Girolamo Calò, Giorgio Amendola, Sandro Cosconati, Salvatore Pacifico, Remo Guerrini, Delia Preti

GlicoPro, Novel Standardized and Sterile Snail Mucus Extract for Multi-Modulative Ocular Formulations: New Perspective in Dry Eye Disease Management

GlicoPro,新型标准化无菌蜗牛粘液提取物,适用于多调节眼部配方:干眼病管理的新视角

Rita Mencucci, Giovanni Strazzabosco, Virginia Cristofori, Andrea Alogna, Daria Bortolotti, Roberta Gafà, Michela Cennamo, Eleonora Favuzza, Claudio Trapella, Valentina Gentili, Roberta Rizzo

Glyceric Prodrug of Ursodeoxycholic Acid (UDCA): Novozym 435-Catalyzed Synthesis of UDCA-Monoglyceride

熊去氧胆酸 (UDCA) 的甘油前药:Novozym 435 催化合成 UDCA-单甘油酯

Federico Zappaterra, Stefania Costa, Daniela Summa, Bruno Semeraro, Virginia Cristofori, Claudio Trapella, Elena Tamburini

Worsening of the Toxic Effects of (±) Cis-4,4'-DMAR Following Its Co-Administration with (±) Trans-4,4'-DMAR: Neuro-Behavioural, Physiological, Immunohistochemical and Metabolic Studies in Mice

(±) Cis-4,4'-DMAR 与 (±) Trans-4,4'-DMAR 共同给药后毒性作用加剧:小鼠神经行为、生理、免疫组织化学和代谢研究

Micaela Tirri, Paolo Frisoni, Sabrine Bilel, Raffaella Arfè, Claudio Trapella, Anna Fantinati, Giorgia Corli, Beatrice Marchetti, Fabio De-Giorgio, Cristian Camuto, Monica Mazzarino, Rosa Maria Gaudio, Giovanni Serpelloni, Fabrizio Schifano, Francesco Botrè, Matteo Marti1

Pharmacological modulation of mitochondrial calcium uniporter controls lung inflammation in cystic fibrosis

药理调节线粒体钙单向转运体控制囊性纤维化肺部炎症

Alessandro Rimessi, Chiara Pozzato, Lorenzo Carparelli, Alice Rossi, Serena Ranucci, Ida De Fino, Cristina Cigana, Anna Talarico, Mariusz R Wieckowski, Carla M P Ribeiro, Claudio Trapella, Giacomo Rossi, Giulio Cabrini, Alessandra Bragonzi, Paolo Pinton

Design of Nanosystems for the Delivery of Quorum Sensing Inhibitors: A Preliminary Study

用于递送群体感应抑制剂的纳米系统的设计:初步研究

Supandeep Singh Hallan, Paolo Marchetti, Daria Bortolotti, Maddalena Sguizzato, Elisabetta Esposito, Paolo Mariani, Claudio Trapella, Roberta Rizzo, Rita Cortesi