日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

CC48 a new CB2R agonist/FAAH inhibitor dual drug blocks gastric cancer progression and overcomes paclitaxel resistance.

CC48 是一种新型 CB2R 激动剂/FAAH 抑制剂双效药物,可阻断胃癌进展并克服紫杉醇耐药性

Schirizzi Annalisa, Renna Natasha, De Leonardis Giampiero, Montanaro Rosangela, Mastropasqua Francesco, Graziano Giovanni, Riganti Chiara, Pisano Isabella, Laghezza Antonio, Abate Carmen, Stefanachi Angela, Colabufo Nicola Antonio, Caccioppoli Cristina, Bianco Giusy, Valentini Anna Maria, Armentano Raffaele, Giannelli Gianluigi, Contino Marialessandra, D'Alessandro Rosalba

Measurement of cyclosporin induced changes in P-glycoprotein function at the human blood-brain barrier using [(18)F]MC225 and PET

利用[(18)F]MC225和PET测量环孢素诱导的人血脑屏障P-糖蛋白功能变化

Mossel, Pascalle; Salvi de Souza, Giordana; Willemsen, Antoon T M; Stormezand, Gilles N; Colabufo, Nicola A; Toyohara, Jun; Boersma, Hendrikus H; Dierckx, Rudi A J O; Lammertsma, Adriaan A; Bartels, Anna L; Luurtsema, Gert

Designing a Small Molecule for PET Radiotracing: [(18)F]MC225 in Human Trials for Early Diagnosis in CNS Pathologies

设计用于PET放射性示踪的小分子:[(18)F]MC225在人体试验中用于中枢神经系统疾病的早期诊断

Mastropasqua, Francesco; Luurtsema, Gert; Filosa, Cristina; Colabufo, Nicola Antonio

Isolation of endothelial progenitor cells from human adipose tissue

从人脂肪组织中分离内皮祖细胞

Caccioppoli, Cristina; D'Oria, Rossella; Genchi, Valentina Annamaria; Palma, Giuseppe; Andrulli Buccheri, Valentina; Calderoni, Isabella; Tedesco, Carmen; Colabufo, Carmela; Marrano, Nicola; Biondi, Giuseppina; Chaoul, Nada; Braun, Antonio; Pezzolla, Angela; Cignarelli, Angelo; Natalicchio, Annalisa; Laviola, Luigi; Giorgino, Francesco; Perrini, Sebastio

Dual Inhibitors of P-gp and Carbonic Anhydrase XII (hCA XII) against Tumor Multidrug Resistance with Piperazine Scaffold

哌嗪骨架的P-gp和碳酸酐酶XII(hCA XII)双重抑制剂对抗肿瘤多药耐药性

Braconi, Laura; Riganti, Chiara; Parenti, Astrid; Cecchi, Marta; Nocentini, Alessio; Bartolucci, Gianluca; Menicatti, Marta; Contino, Marialessandra; Colabufo, Nicola Antonio; Manetti, Dina; Romanelli, Maria Novella; Supuran, Claudiu T; Teodori, Elisabetta

A scalable route to quaternary ammonium-functionalized AgCl colloidal antimicrobials inhibiting food pathogenic bacteria and biofilms

一种可扩展的制备季铵功能化氯化银胶体抗菌剂的方法,该抗菌剂可抑制食品致病菌和生物膜

Bajrami, Diellza; Hossain, Syed Imdadul; Barbarossa, Alexia; Sportelli, Maria Chiara; Picca, Rosaria Anna; Gentile, Luigi; Mastrolonardo, Francesco; Rosato, Antonio; Carocci, Alessia; Colabufo, Nicola Antonio; Mizaikoff, Boris; Cioffi, Nicola

Nature-Inspired 1-Phenylpyrrolo[2,1- a]isoquinoline Scaffold for Novel Antiproliferative Agents Circumventing P-Glycoprotein-Dependent Multidrug Resistance

受自然启发的 1-苯基吡咯并[2,1- a]异喹啉支架可用于新型抗增殖药物,以规避 P-糖蛋白依赖性多药耐药性

Alisa A Nevskaya, Rosa Purgatorio, Tatiana N Borisova, Alexey V Varlamov, Lada V Anikina, Arina Yu Obydennik, Elena Yu Nevskaya, Mauro Niso, Nicola A Colabufo, Antonio Carrieri, Marco Catto, Modesto de Candia, Leonid G Voskressensky, Cosimo D Altomare

Gut-Derived Uremic Toxins in CKD: An Improved Approach for the Evaluation of Serum Indoxyl Sulfate in Clinical Practice

慢性肾脏病中肠源性尿毒症毒素:临床实践中血清吲哚硫酸盐评估的改进方法

Caggiano, Gianvito; Amodio, Loredana; Stasi, Alessandra; Colabufo, Nicola Antonio; Colangiulo, Santina; Pesce, Francesco; Gesualdo, Loreto

A conformational rearrangement of the SARS-CoV-2 host protein sigma-1 is required for antiviral activity: insights from a combined in-silico/in-vitro approach

SARS-CoV-2 宿主蛋白 sigma-1 的构象重排是抗病毒活性所必需的:通过计算机模拟/体外实验相结合的方法获得的见解

Francesca Serena Abatematteo, Pietro Delre, Ivan Mercurio, Veronica V Rezelj, Dritan Siliqi, Stephanie Beaucourt, Gianluca Lattanzi, Nicola Antonio Colabufo, Marcello Leopoldo, Michele Saviano, Marco Vignuzzi, Giuseppe Felice Mangiatordi, Carmen Abate1

LC-MS/MS Analysis on Infusion Bags and Filled Syringes of Decitabine: New Data on Physicochemical Stability of an Unstable Molecule

利用液相色谱-串联质谱法分析地西他滨输液袋和已灌装注射器:不稳定分子理化稳定性的新数据

Laforgia, Mariarita; Amodio, Loredana; Colangiulo, Santina; Ungaro, Valentina; Gatti, Letizia; Lucarelli, Gianpiero; Leopoldo, Marcello; Nardulli, Patrizia; Colabufo, Nicola A