日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Cell-Active Small Molecule Inhibitors of the DNA-Damage Repair Enzyme Poly(ADP-ribose) Glycohydrolase (PARG): Discovery and Optimization of Orally Bioavailable Quinazolinedione Sulfonamides

DNA 损伤修复酶聚(ADP-核糖)糖水解酶 (PARG) 的细胞活性小分子抑制剂:口服生物可利用的喹唑啉二酮磺酰胺的发现和优化

Bohdan Waszkowycz, Kate M Smith, Alison E McGonagle, Allan M Jordan, Ben Acton, Emma E Fairweather, Louise A Griffiths, Niall M Hamilton, Nicola S Hamilton, James R Hitchin, Colin P Hutton, Dominic I James, Clifford D Jones, Stuart Jones, Daniel P Mould, Helen F Small, Alexandra I J Stowell, Julie A

First-in-Class Chemical Probes against Poly(ADP-ribose) Glycohydrolase (PARG) Inhibit DNA Repair with Differential Pharmacology to Olaparib

针对聚(ADP-核糖)糖水解酶 (PARG) 的首创化学探针可抑制 DNA 修复,具有与 Olaparib 不同的药理学作用

Dominic I James, Kate M Smith, Allan M Jordan, Emma E Fairweather, Louise A Griffiths, Nicola S Hamilton, James R Hitchin, Colin P Hutton, Stuart Jones, Paul Kelly, Alison E McGonagle, Helen Small, Alexandra I J Stowell, Julie Tucker, Ian D Waddell, Bohdan Waszkowycz, Donald J Ogilvie