The alpha-7 nicotinic acetylcholine receptor agonist GTS-21 engages the glucagon-like peptide-1 incretin hormone axis to lower levels of blood glucose in db/db mice.
α-7 尼古丁乙酰胆碱受体激动剂 GTS-21 激活胰高血糖素样肽-1肠促胰岛素激素轴,从而降低 db/db 小鼠的血糖水平
期刊:Diabetes Obesity & Metabolism
影响因子:5.7
doi:10.1111/dom.14693
Meng Qinghe, Chepurny Oleg G, Leech Colin A, Pruekprasert Napat, Molnar Megan E, Collier James Jason, Cooney Robert N, Holz George G