日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

α-ketoglutarate/succinate ratio imbalance impairs thymine DNA glycosylase function and base excision repair process increasing susceptibility to pancreatic cancer

α-酮戊二酸/琥珀酸比例失衡会损害胸腺嘧啶DNA糖基化酶功能和碱基切除修复过程,从而增加患胰腺癌的风险。

Malatesta, Silvia; Vigiano Benedetti, Virginia; Salviati, Emanuela; Illi, Barbara; Manni, Isabella; Middonti, Emanuele; Rampioni Vinciguerra, Gian Luca; Licursi, Valerio; Troilo, Francesca; Colotti, Gianni; Cipolla, Lina; Sabbioneda, Simone; Perfetto, Livia; Piaggio, Giulia; Bussolino, Federico; Di Nicolantonio, Federica; Campiglia, Pietro; Sommella, Eduardo Maria; Mori, Mattia; Cencioni, Chiara; Spallotta, Francesco

The ATC12 small molecule inhibits the Aurora-A/TPX2 interaction and impairs the proliferation of breast cancer cells

ATC12小分子抑制Aurora-A/TPX2相互作用,从而抑制乳腺癌细胞增殖。

Boi, Dalila; Fianco, Giulia; Polverino, Federica; Fiorentino, Francesco; Mastrangelo, Anna; Rossi, Simone; Rubini, Elisabetta; Rosignoli, Serena; Troilo, Francesca; Antonelli, Maria Rosaria; Tarquini, Dalila; Cervoni, Laura; Rinaldo, Serena; Tramonti, Angela; Scarpone, Eleonora Kristina; Naro, Chiara; Sette, Claudio; Stagni, Venturina; Colotti, Gianni; Rotili, Dante; Paiardini, Alessandro; Guarguaglini, Giulia; Asteriti, Italia Anna

Immunomodulatory functions of glutaminyl cyclases QPCTL and QPCT

谷氨酰环化酶QPCTL和QPCT的免疫调节功能

Smid, Hannah Elaine; Colotti, Jana; Nölp, Sophia; Arlt, Nike Sophia; Weber, Sophie; Gumann, Amelie; von Hörsten, Stephan; Karow, Axel; Schuh, Wolfgang

PACS deficiency disrupts Golgi architecture and causes cytokinesis failures and seizure-like phenotype in Drosophila melanogaster

PACS 缺陷会破坏高尔基体结构,导致果蝇胞质分裂失败和癫痫样表型

Anna Frappaolo, Gianluca Zaccagnini, Maria Giovanna Riparbelli, Gianni Colotti, Giuliano Callaini, Maria Grazia Giansanti

Structural analysis of cancer-relevant TCR-CD3 and peptide-MHC complexes by cryoEM

利用冷冻电镜技术对癌症相关TCR-CD3和肽-MHC复合物进行结构分析

Kei Saotome ,Drew Dudgeon ,Kiersten Colotti ,Michael J Moore ,Jennifer Jones ,Yi Zhou ,Ashique Rafique ,George D Yancopoulos ,Andrew J Murphy ,John C Lin ,William C Olson ,Matthew C Franklin

Structural analysis of cancer-relevant TCR-CD3 and peptide-MHC complexes by cryoEM

利用冷冻电镜技术对癌症相关TCR-CD3和肽-MHC复合物进行结构分析

Kei Saotome,Drew Dudgeon,Kiersten Colotti,Michael J Moore,Jennifer Jones,Yi Zhou,Ashique Rafique,George D Yancopoulos,Andrew J Murphy,John C Lin,William C Olson,Matthew C Franklin

Bcl-2 family inhibitors sensitize human cancer models to therapy

Bcl-2 家族抑制剂使人类癌症模型对治疗敏感

Elisabetta Valentini #, Marta Di Martile #, Matteo Brignone, Marica Di Caprio, Isabella Manni, Michela Chiappa, Ilaria Sergio, Martina Chiacchiarini, Chiara Bazzichetto, Fabiana Conciatori, Simona D'Aguanno, Carmen D'Angelo, Rino Ragno, Michelangelo Russillo, Gianni Colotti, Francesco Marchesi, Mari

Bcl-2 family inhibitors sensitize human cancer models to therapy

Bcl-2家族抑制剂可增强人类癌症模型对治疗的敏感性

Elisabetta Valentini #,Marta Di Martile #,Matteo Brignone,Marica Di Caprio,Isabella Manni,Michela Chiappa,Ilaria Sergio,Martina Chiacchiarini,Chiara Bazzichetto,Fabiana Conciatori,Simona D'Aguanno,Carmen D'Angelo,Rino Ragno,Michelangelo Russillo,Gianni Colotti,Francesco Marchesi,Maria Laura Bellone,Fabrizio Dal Piaz,Maria Pia Felli,Giovanna Damia,Donatella Del Bufalo

Novel 1,4-Dihydropyridines as Specific Binders and Activators of SIRT3 Impair Cell Viability and Clonogenicity and Downregulate Hypoxia-Induced Targets in Cancer Cells

新型 1,4-二氢吡啶作为 SIRT3 的特异性结合剂和激活剂,会损害细胞活力和克隆形成能力,并下调癌细胞中缺氧诱导的靶标

Clemens Zwergel, Michele Aventaggiato, Sabrina Garbo, Elisabetta Di Bello, Bruno Fassari, Beatrice Noce, Carola Castiello, Chiara Lambona, Federica Barreca, Dante Rotili, Rossella Fioravanti, Thomas Schmalz, Michael Weyand, Amelie Niedermeier, Marco Tripodi, Gianni Colotti, Clemens Steegborn, Cecili

Targeting the anti-apoptotic Bcl-2 family proteins: machine learning virtual screening and biological evaluation of new small molecules

针对抗凋亡Bcl-2家族蛋白:机器学习虚拟筛选及新型小分子的生物学评价

Elisabetta Valentini, Simona D'Aguanno, Marta Di Martile, Camilla Montesano, Virginia Ferraresi, Alexandros Patsilinakos, Manuela Sabatino, Lorenzo Antonini, Martina Chiacchiarini, Sergio Valente, Antonello Mai, Gianni Colotti, Rino Ragno, Daniela Trisciuoglio, Donatella Del Bufalo