日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

4-(5-Chloro-3-(3,4,5-trimethoxybenzoyl)-1H-indol-1-yl)benzenesulfonamide: A Novel Polypharmacology Agent to Target Carbonic Anhydrase IX and XII With Improved Selectivity, Wnt/β-Catenin Signaling Pathway, and P-Glycoprotein

4-(5-氯-3-(3,4,5-三甲氧基苯甲酰基)-1H-吲哚-1-基)苯磺酰胺:一种新型多靶点药物,可选择性地靶向碳酸酐酶IX和XII、Wnt/β-catenin信号通路以及P-糖蛋白。

Puxeddu, Michela; Bordone, Rosa; Colla, Claudia; Rotili, Gabriele; Coluccia, Antonio; Sciò, Pietro; Cuřínová, Petra; Nocentini, Alessio; Supuran, Claudiu T; Filiberti, Serena; Turati, Marta; Ronca, Roberto; Kopecka, Joanna; Riganti, Chiara; Jimenez, Lucia; Link, Wolfgang; Bigogno, Chiara; Dondio, Giulio; Barba, Martina; Canettieri, Gianluca; Silvestri, Romano; La Regina, Giuseppe

Exploring structure-activity relationships of pyrrolyl diketo acid derivatives as non-nucleoside inhibitors of terminal deoxynucleotidyl transferase enzyme

探索吡咯基二酮酸衍生物作为末端脱氧核苷酸转移酶非核苷类抑制剂的构效关系

Madia, Valentina Noemi; Garibaldi, Nadia; Ialongo, Davide; Patacchini, Elisa; Tudino, Valeria; Ruggieri, Giuseppe; Zarbo, Laura; Cara, Emanuele; Coluccia, Antonio; Artico, Marco; Scipione, Luigi; Messore, Antonella; Saccoliti, Francesco; Mentegari, Elisa; Maga, Giovanni; Di Santo, Roberto; Crespan, Emmanuele; Costi, Roberta

Structure-function relationship of the Pseudomonas aeruginosa AsmA-like proteins YhdP and YdbH involved in outer membrane biogenesis

铜绿假单胞菌AsmA样蛋白YhdP和YdbH参与外膜生物合成的结构-功能关系

Sposato, Davide; Pederzoli, Camilla; Bufano, Marianna; Sciò, Pietro; Rossi, Ludovica; Leoni, Livia; Rampioni, Giordano; Visca, Paolo; Coluccia, Antonio; Imperi, Francesco

Identification of a New FtsZ Inhibitor by Virtual Screening, Mechanistic Insights, and Structure-Activity Relationship Analyses

通过虚拟筛选、机制研究和构效关系分析鉴定一种新的FtsZ抑制剂

Sciò, Pietro; Scoffone, Viola Camilla; Parisi, Anastasia; Bufano, Marianna; Caneva, Martina; Trespidi, Gabriele; Irudal, Samuele; Barbieri, Giulia; Cariani, Lisa; Orena, Beatrice Silvia; Daccò, Valeria; Imperi, Francesco; Buroni, Silvia; Coluccia, Antonio

Microwave-assisted synthesis of tubulin assembly inhibitors as anticancer agents by aryl ring reversal and conjunctive approach.

利用芳环反转和连接方法微波辅助合成微管蛋白组装抑制剂作为抗癌剂

Masci Domiziana, Puxeddu Michela, Colla Claudia, Coluccia Antonio, Santelli Martina, Sciò Pietro, Mariotto Elena, Viola Giampietro, Hamel Ernest, Lerose Rosa, Mazzoccoli Carmela, Silvestri Romano, La Regina Giuseppe

Strain-based method for fatigue failure prediction of additively manufactured lattice structures

基于应变的增材制造晶格结构疲劳失效预测方法

Coluccia, Antonio; De Pasquale, Giorgio

Exploring CCRL2 chemerin binding using accelerated molecular dynamics

利用加速分子动力学探索CCRL2趋化蛋白结合

Bufano, Marianna; Laffranchi, Mattia; Sozzani, Silvano; Raimondo, Domenico; Silvestri, Romano; Coluccia, Antonio

Targeting PDZ domains as potential treatment for viral infections, neurodegeneration and cancer

以PDZ结构域为靶点,探索治疗病毒感染、神经退行性疾病和癌症的潜在疗法

Nardella, Caterina; Visconti, Lorenzo; Malagrinò, Francesca; Pagano, Livia; Bufano, Marianna; Nalli, Marianna; Coluccia, Antonio; La Regina, Giuseppe; Silvestri, Romano; Gianni, Stefano; Toto, Angelo

Discovery of Zika Virus NS2B/NS3 Inhibitors That Prevent Mice from Life-Threatening Infection and Brain Damage

发现寨卡病毒NS2B/NS3抑制剂可预防小鼠发生危及生命的感染和脑损伤

Coluccia, Antonio; Puxeddu, Michela; Nalli, Marianna; Wei, Chih-Ku; Wu, Yu-Hsuan; Mastrangelo, Eloise; Elamin, Tasneem; Tarantino, Delia; Bugert, Joachim Jakob; Schreiner, Benno; Nolte, Juliane; Schwarze, Frank; La Regina, Giuseppe; Lee, Jin-Ching; Silvestri, Romano

Modeling Epac1 interactions with the allosteric inhibitor AM-001 by co-solvent molecular dynamics

利用共溶剂分子动力学模拟Epac1与变构抑制剂AM-001的相互作用

Bufano, Marianna; Laudette, Marion; Blondeau, Jean-Paul; Lezoualc'h, Frank; Nalli, Marianna; Silvestri, Romano; Brancale, Andrea; Coluccia, Antonio