Prodrugs of a 1-Hydroxy-2-oxopiperidin-3-yl Phosphonate Enolase Inhibitor for the Treatment of ENO1-Deleted Cancers
用于治疗ENO1缺失癌症的1-羟基-2-氧代哌啶-3-基膦酸酯烯醇化酶抑制剂前药
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.2c01039
Yan, Victoria C; Pham, Cong-Dat; Ballato, Elliot S; Yang, Kristine L; Arthur, Kenisha; Khadka, Sunada; Barekatain, Yasaman; Shrestha, Prakriti; Tran, Theresa; Poral, Anton H; Washington, Mykia; Raghavan, Sudhir; Czako, Barbara; Pisaneschi, Federica; Lin, Yu-Hsi; Satani, Nikunj; Hammoudi, Naima; Ackroyd, Jeffrey J; Georgiou, Dimitra K; Millward, Steven W; Muller, Florian L