日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fat or flat? The impact of dipole moment vectors on non-covalent interactions between aromatic tags and macromolecules

胖还是扁?偶极矩矢量对芳香标签与大分子间非共价相互作用的影响

Holub, Josef; Jílková, Adéla; Lemke, Carina; Cianni, Lorenzo; Spiwoková, Petra; Horn, Martin; Breuer, Christian; Leontovyč, Adrian; Brynda, Jiří; Mertlíková-Kaiserová, Helena; Chanová, Marta; Dos Reis Rocho, Fernanda; Montanari, Carlos A; El-Sakkary, Nelly; Caffrey, Conor R; Gütschow, Michael; Hnyk, Drahomír; Mareš, Michael; Fanfrlík, Jindřich

Secure and scalable gene expression quantification with pQuant

pQuant 提供安全且可扩展的基因表达定量分析

Hong, Seungwan; Walker, Conor R; Choi, Yoolim A; Gürsoy, Gamze

CPSF1 inhibition promotes widespread use of intergenic polyadenylation sites and impairs glycolysis in prostate cancer cells

CPSF1抑制促进基因间多聚腺苷酸化位点的广泛利用,并损害前列腺癌细胞的糖酵解。

Kiel T Tietz,Braedan M McCluskey,Conor R Miller,Yingming Li,Sarah A Munro,Scott M Dehm

Discovery of benzyl carbamate inhibitors of coronavirus M(pro) enzymes from a legacy collection of cysteine protease inhibitors

从一系列已知的半胱氨酸蛋白酶抑制剂中发现冠状病毒M(pro)酶的苄基氨基甲酸酯抑制剂

Sá Magalhães Serafim, Mateus; Kronenberger, Thales; Francisco, Karol R; de Sousa Reis, Erik Vinicius; Gonçalves de Oliveira, Ellen; Marcelino E Oliveira, Fernanda Kelly; Serraglio Fortes, Isadora; Maciel Fernandes, Thaís Helena; Barbosa da Silva, Elany; Fajtova, Pavla; Skinner, Danielle E; Syed, Rafay O; Lage de Siqueira-Neto, Jair; Poso, Antti; Fernandes Mota, Bruno Eduardo; Alves Coelho-Dos-Reis, Jordana Grazziela; Santos Abrahão, Jônatas; Gonçalves Maltarollo, Vinícius; O'Donoghue, Anthony J; Caffrey, Conor R

Detecting Interspecific Positive Selection Using Convolutional Neural Networks

利用卷积神经网络检测种间正选择

West, Charlotte; Walker, Conor R; Arasti, Shayesteh; Vasilev, Viacheslav; Xu, Xingze; De Maio, Nicola; Goldman, Nick

Enhancing schistosomiasis drug discovery approaches with optimized proteasome substrates.

利用优化的蛋白酶体底物增强血吸虫病药物发现方法

Silva Elany B, Jiang Zhenze, Liu Chenxi, Fajtová Pavla, Teixeira Thaiz R, de Castro Fiorini Maia Giovana, Liu Lawrence J, El-Sakkary Nelly, Skinner Danielle E, Syed Ali, Wang Steven C, Caffrey Conor R, O'Donoghue Anthony J

Chalcogen Derivatives for the Treatment of African Trypanosomiasis: Biological Evaluation of Thio- and Seleno-Semicarbazones and Their Azole Derivatives.

硫族元素衍生物治疗非洲锥虫病:硫代和硒代氨基脲及其唑类衍生物的生物学评价

Rubio-Hernández Mercedes, Teixeira Thaiz R, Nguyen Tina P, Shingyoji Mai, da Silva Elany Barbosa, O'Donoghue Anthony J, Caffrey Conor R, Pérez-Silanes Silvia, Martínez-Sáez Nuria

Nitroquinolones and nitroquinolines: syntheses and antitrypanosomal activity

硝基喹诺酮类和硝基喹啉类:合成及抗锥虫活性

Dube, Phelelisiwe S; Francisco, Karol R; Legoabe, Lesetja J; Sun, Yujie Uli; Kaur, Yashpreet; Nguyen, Tina P; Caffrey, Conor R; Beteck, Richard M

Identification of Substituted 4-Aminocinnolines as Broad-Spectrum Antiparasitic Agents

鉴定取代的4-氨基喹啉类化合物作为广谱抗寄生虫药物

Spaulding, Andrew; Sharma, Amrita; Giardini, Miriam A; Hoffman, Benjamin; Bernatchez, Jean A; McCall, Laura-Isobel; Calvet, Claudia M; Ackermann, Jasmin; Souza, Julia M; Thomas, Diane; Millard, Caroline C; Devine, William G; Singh, Baljinder; Silva, Everton M; Leed, Susan E; Roncal, Norma E; Penn, Erica C; Erath, Jessey; Kumar, Gaurav; Sepulveda, Yadira; Garcia, Arnold; Rodriguez, Ana; El-Sakkary, Nelly; Sciotti, Richard J; Campbell, Robert F; Momper, Jeremiah D; McKerrow, James H; Caffrey, Conor R; Siqueira-Neto, Jair L; Pollastri, Michael P; Mensa-Wilmot, Kojo; Ferrins, Lori

Aza-peptide aldehydes and ketones: synthesis and evaluation as human 20S proteasome inhibitors

氮杂肽醛和酮:合成及作为人20S蛋白酶体抑制剂的评价

Corrigan, Thomas S; Border, Sarah E; Lotti Diaz, Leilani M; Kasper, Kayla Q; Noonchester, Abigail M; Amer, Rasmiah; Kucway, Kayla S; Fleisher, Michael; Fernandez, Joseph P; Lovins, Alex R; Serrano, Ana K; Caffrey, Conor R; O'Donoghue, Anthony J; Benson, Don M Jr; Hadad, Christopher M; Ekici, Özlem Doğan