Peptidomimetic α-Acyloxymethylketone Warheads with Six-Membered Lactam P1 Glutamine Mimic: SARS-CoV-2 3CL Protease Inhibition, Coronavirus Antiviral Activity, and in Vitro Biological Stability
具有六元内酰胺 P1 谷氨酰胺模拟物的肽模拟 α-酰氧甲基酮弹头：SARS-CoV-2 3CL 蛋白酶抑制、冠状病毒抗病毒活性和体外生物稳定性
期刊:Journal of Medicinal Chemistry
影响因子:6.8
doi:10.1021/acs.jmedchem.1c00616
Bing Bai, Alexandr Belovodskiy, Mostofa Hena, Appan Srinivas Kandadai, Michael A Joyce, Holly A Saffran, Justin A Shields, Muhammad Bashir Khan, Elena Arutyunova, Jimmy Lu, Sardeev K Bajwa, Darren Hockman, Conrad Fischer, Tess Lamer, Wayne Vuong, Marco J van Belkum, Zhengxian Gu, Fusen Lin, Yanhua D
