Discovery of isoquinoline sulfonamides as allosteric gyrase inhibitors with activity against fluoroquinolone-resistant bacteria
发现异喹啉磺胺类药物作为变构旋转酶抑制剂,具有抗氟喹诺酮耐药细菌的活性
期刊:Nature Chemistry
影响因子:19.2
doi:10.1038/s41557-024-01516-x
Alexander T Bakker #, Ioli Kotsogianni #, Mariana Avalos, Jeroen M Punt, Bing Liu, Diana Piermarini, Berend Gagestein, Cornelis J Slingerland, Le Zhang, Joost J Willemse, Leela B Ghimire, Richard J H B N van den Berg, Antonius P A Janssen, Tom H M Ottenhoff, Constant A A van Boeckel, Gilles P van We