日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Polyfunctionalized N-Arylsulfonyl Indoles: Identification of (E)-N-Hydroxy-3-{3-[(5-(3-(piperidin-1-yl)propoxy]-1H-indol-1-yl)sulfonyl]phenyl}acrylamide (MTP150) for the Epigenetic-Based Therapy of Parkinson's Disease

多功能化N-芳基磺酰基吲哚:(E)-N-羟基-3-{3-[(5-(3-(哌啶-1-基)丙氧基]-1H-吲哚-1-基)磺酰基]苯基}丙烯酰胺 (MTP150) 的鉴定及其在帕金森病表观遗传治疗中的应用

Toledano-Pinedo, Mireia; Porro-Pérez, Alicia; Schäker-Hübner, Linda; Diez-Iriepa, Daniel; Iriepa, Isabel; Siwek, Agata; Wolak, Małgorzata; Satała, Grzegorz; Bojarski, Andrzej J; Doroz-Płonka, Agata; Handzlik, Jadwiga; Godyń, Justyna; Dallemagne, Patrick; Rochais, Christophe; Davis, Audrey; Since, Marc; Pérez, Belén; Bellver-Sanchis, Aina; Irisarri, Alba; Pallàs, Mercè; Solana-Manrique, Cristina; López-Muñoz, Francisco; Ismaili, Lhassane; Griñán-Ferré, Christian; Paricio, Nuria; K Hansen, Finn; Więckowska, Anna; Marco-Contelles, José

NLRP3 Inflammasome Role and NLRP3 Inhibitors in Sensorineural Hearing Loss

NLRP3炎症小体及其抑制剂在感觉神经性听力损失中的作用

Toledano-Pinedo, Mireia; Marco-Contelles, José; Dobrydnev, Alexey V

Behavioural Impact of Parental Presence Versus Absence in Paediatric Dentistry: A Systematic Review

家长在场与不在场对儿童牙科行为的影响:一项系统性综述

Vello-Ribes, M Angeles; Aura-Tormos, J Ignacio; Valero-Contelles, Carolina; Casaña-Ruiz, M Dolores; Catala-Pizarro, Montserrat

Generation and validation of a novel multitarget small molecule in glioblastoma.

胶质母细胞瘤新型多靶点小分子的生成与验证

Artetxe-Zurutuza Aizpea, Iturrioz-Rodriguez Nerea, Elizazu Joseba, Toledano-Pinedo Mireia, Porro-Pérez Alicia, De Goñi Irati, Elua-Pinin Alejandro, Schäker-Hübner Linda, Azkargorta Mikel, Elortza Felix, Iriepa Isabel, Lòpez-Muñoz Francisco, Moncho-Amor Veronica, Hansen Finn K, Sampron Nicolás, Marco-Contelles Jose Luis, Matheu Ander

Generation and Characterization of Novel Contilisant+Tubastatin a Multitarget Small Molecules Against Glioblastoma.

新型 Contilisant+Tubastatin 的生成和表征:一种针对胶质母细胞瘤的多靶点小分子。

de Goñi Irati, Artetxe-Zurutuza Aizpea, Elizazu Joseba, Garcia-Garcia de Garayo Raul, Vergara-Arce Jhonatan, Azkargorta Mikel, Toledano-Pinedo Mireia, Porro-Pérez Alicia, Elortza Felix, Marco-Contelles Jose Luis, Sampron Nicolas, Iturrioz-Rodriguez Nerea, Matheu Ander

Coinage Metal-Catalyzed Divergent Heterocyclizations of Underexplored N-Propargyl Hydrazides

贵金属催化的未充分研究的N-炔丙基酰肼的发散性杂环化反应

Diez-Iriepa, Daniel; Toledano-Pinedo, Mireia; Herrera-Hernández, Lorena; Samadi, Abdelouahid; Raouf, Yasir S; Rodríguez-Fernández, M Mercedes; Flores-Galán, Paula; Yanai, Hikaru; Alonso, José M; Marco-Contelles, José; Almendros, Pedro

Neuroprotective and Antioxidant Properties of Different Novel Steroid-Derived Nitrones and Oximes on Cerebral Ischemia In Vitro

不同新型甾体衍生的硝酮和肟类化合物对体外脑缺血的神经保护和抗氧化特性

Izquierdo-Bermejo, Sara; Chioua, Mourad; Hadjipavlou-Litina, Dimitra; López-Muñoz, Francisco; Marco-Contelles, José; Oset-Gasque, María Jesús

Characterization of a Novel Family of Contilisant + Belinostat Multitarget Small Molecules in Glioblastoma

胶质母细胞瘤中新型 Contilisant + Belinostat 多靶点小分子家族的特性分析

Artetxe-Zurutuza, Aizpea; Iturrioz-Rodriguez, Nerea; Elizazu, Joseba; Garcia-Garcia de Garayo, Raul; de Goñi, Irati; Vergara, Jhonatan; Toledano-Pinedo, Mireia; Porro-Pérez, Alicia; Azkargorta, Mikel; Elortza, Felix; Marco-Contelles, Jose Luis; Sampron, Nicolás; Matheu, Ander

Multicomponent Synthesis of Multi-Target Quinazolines Modulating Cholinesterase, Oxidative Stress, and Amyloid Aggregation Activities for the Therapy of Alzheimer's Disease

利用多组分合成法制备多靶点喹唑啉类化合物,调节胆碱酯酶、氧化应激和淀粉样蛋白聚集活性,用于治疗阿尔茨海默病

Chakhari, Saida; Marco-Contelles, José; Iriepa, Isabel; Carreiras, Maria do Carmo; Chabchoub, Fakher; Ismaili, Lhassane; Refouvelet, Bernard

Quinolylnitrone 23 Protects from Auditory Cell Oxidative Injury and Noise-Induced Hearing Loss

喹诺基硝酮 23 可保护听觉细胞免受氧化损伤和噪声性听力损失

Murillo-Cuesta, Silvia; Contreras, Julio; Chioua, Mourad; García-Montoya, Carmen; Rodríguez-de la Rosa, Lourdes; Méndez-Grande, Inés; Piotrowska, Dorota G; Głowacka, Iwona E; Varela-Nieto, Isabel; Marco-Contelles, José