日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification and characterization of a first-generation inhibitor of claudin-1 in colon cancer progression and metastasis

第一代 claudin-1 抑制剂在结肠癌进展和转移中的鉴定和特性

Iram Fatima, Jaya Prakash Uppada, Yashpal S Chhonker, Saiprasad Gowrikumar, Susmita Barman, Sourav Roy, Kirsten T Tolentino, Nicholas Palermo, Amar Natarajan, Daniel R Beauchamp, Alex Vecchio, Daryl J Murry, Amar B Singh, Corey R Hopkins, Punita Dhawan

Bidirectional Influence of Limbic GIRK Channel Activation on Innate Avoidance Behavior

边缘 GIRK 通道激活对先天回避行为的双向影响

Baovi N Vo, Ezequiel Marron Fernandez de Velasco, Timothy R Rose, Hannah Oberle, Haichang Luo, Corey R Hopkins, Kevin Wickman

TRPC5 Channel Inhibition Protects Podocytes in Puromycin-Aminonucleoside Induced Nephrosis Models

TRPC5 通道抑制可保护嘌呤霉素-氨基核苷诱发的肾病模型中的足细胞

Yiming Zhou, Choah Kim, Juan Lorenzo B Pablo, Fan Zhang, Ji Yong Jung, Li Xiao, Silvana Bazua-Valenti, Maheswarareddy Emani, Corey R Hopkins, Astrid Weins, Anna Greka

Discovery and Characterization of VU0529331, a Synthetic Small-Molecule Activator of Homomeric G Protein-Gated, Inwardly Rectifying, Potassium (GIRK) Channels

发现并表征 VU0529331,一种同源 G 蛋白门控内向整流钾 (GIRK) 通道的合成小分子激活剂

Krystian A Kozek, Yu Du, Swagat Sharma, Francis J Prael 3rd, Brittany D Spitznagel, Sujay V Kharade, Jerod S Denton, Corey R Hopkins, C David Weaver

Discovery, Characterization, and Effects on Renal Fluid and Electrolyte Excretion of the Kir4.1 Potassium Channel Pore Blocker, VU0134992

Kir4.1 钾通道孔阻滞剂 VU0134992 的发现、特性及对肾液和电解质排泄的影响

Sujay V Kharade, Haruto Kurata, Aaron M Bender, Anna L Blobaum, Eric E Figueroa, Amanda Duran, Meghan Kramer, Emily Days, Paige Vinson, Daniel Flores, Lisa M Satlin, Jens Meiler, C David Weaver, Craig W Lindsley, Corey R Hopkins, Jerod S Denton

ML418: The First Selective, Sub-Micromolar Pore Blocker of Kir7.1 Potassium Channels

ML418:首个选择性亚微摩尔 Kir7.1 钾通道孔阻滞剂

Daniel R Swale, Haruto Kurata, Sujay V Kharade, Jonathan Sheehan, Rene Raphemot, Karl R Voigtritter, Eric E Figueroa, Jens Meiler, Anna L Blobaum, Craig W Lindsley, Corey R Hopkins, Jerod S Denton

Activation of Metabotropic Glutamate Receptor 7 Is Required for Induction of Long-Term Potentiation at SC-CA1 Synapses in the Hippocampus

代谢型谷氨酸受体 7 的激活是海马 SC-CA1 突触诱导长期增强的必要条件

Rebecca Klar, Adam G Walker, Dipanwita Ghose, Brad A Grueter, Darren W Engers, Corey R Hopkins, Craig W Lindsley, Zixiu Xiang, P Jeffrey Conn, Colleen M Niswender

Discovery and characterization of 2-(cyclopropanesulfonamido)-N-(2-ethoxyphenyl)benzamide, ML382: a potent and selective positive allosteric modulator of MrgX1

2-(环丙烷磺酰胺基)-N-(2-乙氧基苯基)苯甲酰胺 ML382 的发现和表征:一种强效且选择性的 MrgX1 正变构调节剂

Wandong Wen, Yan Wang, Zhe Li, Pang-Yen Tseng, Owen B McManus, Meng Wu, Min Li, Craig W Lindsley, Xinzhong Dong, Corey R Hopkins

Specific activin receptor-like kinase 3 inhibitors enhance liver regeneration

特异性激活素受体样激酶 3 抑制剂可增强肝脏再生

Daisuke Tsugawa, Yuki Oya, Ryota Masuzaki, Kevin Ray, Darren W Engers, Martin Dib, Nhue Do, Kaori Kuramitsu, Karen Ho, Audrey Frist, Paul B Yu, Kenneth D Bloch, Craig W Lindsley, Corey R Hopkins, Charles C Hong, Seth J Karp

Inhibition of the TRPC5 ion channel protects the kidney filter

抑制TRPC5离子通道保护肾脏过滤器

Thomas Schaldecker, Sookyung Kim, Constantine Tarabanis, Dequan Tian, Samy Hakroush, Philip Castonguay, Wooin Ahn, Hanna Wallentin, Hans Heid, Corey R Hopkins, Craig W Lindsley, Antonio Riccio, Lisa Buvall, Astrid Weins, Anna Greka