日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Conformational Remodeling Underlies Activity Loss in Disease-Linked Asparagine Synthetase Variant

构象重塑是疾病相关天冬酰胺合成酶变体活性丧失的根本原因

Pearce, Lucciano A; Coricello, Adriana; Nardone, Alanya J; Bottegoni, Giovanni; Takagi, Yuichiro; Zhu, Wen

Adiabatic-Bias Molecular Dynamics Simulations Reveal the Impact of Mutations on Muscarinic Antagonist Unbinding Kinetics

绝热偏压分子动力学模拟揭示突变对毒蕈碱拮抗剂解离动力学的影响

Coricello, Adriana; Chiaravalle, Anna Lisa; Musgaard, Maria; Tehan, Benjamin Gerald; Elisi, Gian Marco; Bottegoni, Giovanni

3D variability analysis reveals a hidden conformational change controlling ammonia transport in human asparagine synthetase

三维变异性分析揭示了控制人天冬酰胺合成酶氨转运的隐藏构象变化

Coricello, Adriana; Nardone, Alanya J; Lupia, Antonio; Gratteri, Carmen; Vos, Matthijn; Chaptal, Vincent; Alcaro, Stefano; Zhu, Wen; Takagi, Yuichiro; Richards, Nigel G J

3D Variability Analysis Reveals a Hidden Conformational Change Controlling Ammonia Transport in Human Asparagine Synthetase

三维变异性分析揭示了控制人天冬酰胺合成酶氨转运的隐藏构象变化

Coricello, Adriana; Nardone, Alanya J; Lupia, Antonio; Gratteri, Carmen; Vos, Matthijn; Chaptal, Vincent; Alcaro, Stefano; Zhu, Wen; Takagi, Yuichiro; Richards, Nigel G J

Discovery of AD258 as a Sigma Receptor Ligand with Potent Antiallodynic Activity

发现 AD258 是一种具有强效抗痛活性的 Sigma 受体配体

Maria Dichiara, Francesca Alessandra Ambrosio, Sang Min Lee, M Carmen Ruiz-Cantero, Jessica Lombino, Adriana Coricello, Giosuè Costa, Dhara Shah, Giuliana Costanzo, Lorella Pasquinucci, Kyung No Son, Giuseppe Cosentino, Rafael González-Cano, Agostino Marrazzo, Vinay Kumar Aakalu, Enrique J Cobos, St

Exploiting DNA Ligase III addiction of multiple myeloma by flavonoid Rhamnetin

利用黄酮类化合物鼠李素对多发性骨髓瘤DNA连接酶III的依赖性

Caracciolo, Daniele; Juli, Giada; Riillo, Caterina; Coricello, Adriana; Vasile, Francesca; Pollastri, Sara; Rocca, Roberta; Scionti, Francesca; Polerà, Nicoletta; Grillone, Katia; Arbitrio, Mariamena; Staropoli, Nicoletta; Caparello, Basilio; Britti, Domenico; Loprete, Giovanni; Costa, Giosuè; Di Martino, Maria Teresa; Alcaro, Stefano; Tagliaferri, Pierosandro; Tassone, Pierfrancesco

ABCC Transporters Mediate the Vacuolar Accumulation of Crocins in Saffron Stigmas

ABCC 转运蛋白介导藏红花柱头中藏红花素的液泡积累

Olivia Costantina Demurtas, Rita de Brito Francisco, Gianfranco Diretto, Paola Ferrante, Sarah Frusciante, Marco Pietrella, Giuseppe Aprea, Lorenzo Borghi, Mistianne Feeney, Lorenzo Frigerio, Adriana Coricello, Giosuè Costa, Stefano Alcaro, Enrico Martinoia, Giovanni Giuliano

High-resolution crystal structure of human asparagine synthetase enables analysis of inhibitor binding and selectivity

人类天冬酰胺合成酶的高分辨率晶体结构可以分析抑制剂的结合和选择性

Wen Zhu, Ashish Radadiya, Claudine Bisson, Sabine Wenzel, Brian E Nordin, Francisco Martínez-Márquez, Tsuyoshi Imasaki, Svetlana E Sedelnikova, Adriana Coricello, Patrick Baumann, Alexandria H Berry, Tyzoon K Nomanbhoy, John W Kozarich, Yi Jin, David W Rice, Yuichiro Takagi, Nigel G J Richards

Erratum: Author Correction: High-resolution crystal structure of human asparagine synthetase enables analysis of inhibitor binding and selectivity

勘误:作者更正:人类天冬酰胺合成酶的高分辨率晶体结构能够分析抑制剂的结合和选择性。

Zhu, Wen; Radadiya, Ashish; Bisson, Claudine; Wenzel, Sabine; Nordin, Brian E; Martínez-Márquez, Francisco; Imasaki, Tsuyoshi; Sedelnikova, Svetlana E; Coricello, Adriana; Baumann, Patrick; Berry, Alexandria H; Nomanbhoy, Tyzoon K; Kozarich, John W; Jin, Yi; Rice, David W; Takagi, Yuichiro; Richards, Nigel G J