日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

StabLyzeGraph: High-throughput screening of combinatorial mutations using graph neural networks

StabLyzeGraph:利用图神经网络进行组合突变的高通量筛选

Waqas, Muhammad; Natale, Benito; Roggia, Michele; Saha, Prasenjit Prasad; Mileni, Mauro; Cosconati, Sandro

Synthesis of New Asymmetrical Chalcones and Evaluation of Their Use in Combination with Curcumin Against Rhodesain of T. brucei rhodesiense

合成新型不对称查尔酮及其与姜黄素联合治疗罗得西亚锥虫病的效果评价

Di Chio, Carla; Starvaggi, Josè; Natale, Benito; Previti, Santo; De Luca, Fabiola; Cosconati, Sandro; Schirmeister, Tanja; Zappalà, Maria; Ettari, Roberta

AI-Enforced Ultra-Large Virtual Screening Discovers Potent CD28 Binders

AI辅助的超大规模虚拟筛选发现强效CD28结合剂

Upadhyaya, Saurabh; Roggia, Michele; Yuan, Shaoren; Cosconati, Sandro; Gabr, Moustafa T

Sustainable Ultrasound-Assisted Solid-Phase peptide synthesis (SUS-SPPS): Less Waste, more efficiency

可持续超声辅助固相肽合成(SUS-SPPS):减少浪费,提高效率

Mottola, Salvatore; Bene, Alessandra Del; Mazzarella, Vincenzo; Cutolo, Roberto; Boccino, Ida; Merlino, Francesco; Cosconati, Sandro; Maro, Salvatore Di; Messere, Anna

Trimethylamine N-Oxide (TMAO) Acts as Inhibitor of Endothelial Nitric Oxide Synthase (eNOS) and Hampers NO Production and Acetylcholine-Mediated Vasorelaxation in Rat Aortas.

三甲胺 N-氧化物 (TMAO) 可作为内皮型一氧化氮合酶 (eNOS) 的抑制剂,阻碍大鼠主动脉中 NO 的产生和乙酰胆碱介导的血管舒张

Martelli Alma, Abate Federico, Roggia Michele, Benedetti Giada, Caradonna Eugenio, Calderone Vincenzo, Tenore Gian Carlo, Cosconati Sandro, Novellino Ettore, Stornaiuolo Mariano

Cigarette smoke destabilizes G-quadruplex structures and antagonizes G4-ligand effects in macrophages

香烟烟雾会破坏巨噬细胞中G-四链体结构的稳定性,并拮抗G4配体的作用。

Mirra, Davida; Salvati, Erica; Esposito, Renata; Spaziano, Giuseppe; Panico, Francesca; Perelli, Agnese; Cutolo, Roberto; Di Maro, Salvatore; Cosconati, Sandro; D'Agostino, Bruno

From genetic code to global health: the impact of nucleic acid vaccines on disease prevention and treatment

从基因密码到全球健康:核酸疫苗对疾病预防和治疗的影响

Del Bene, Alessandra; D'Aniello, Antonia; Mottola, Salvatore; Mazzarella, Vincenzo; Cutolo, Roberto; Campagna, Erica; Benedetti, Rosaria; Altucci, Lucia; Cosconati, Sandro; Di Maro, Salvatore; Messere, Anna

Development of Novel Peptidyl Nitriles Targeting Rhodesain and Falcipain-2 for the Treatment of Sleeping Sickness and Malaria.

开发针对 Rhodesain 和 Falcipain-2 的新型肽基腈,用于治疗昏睡病和疟疾

Di Chio Carla, Starvaggi Josè, Totaro Noemi, Previti Santo, Natale Benito, Cosconati Sandro, Bogacz Marta, Schirmeister Tanja, Legac Jenny, Rosenthal Philip J, Zappalà Maria, Ettari Roberta

Quinolinonyl Derivatives as Dual Inhibitors of the HIV-1 Integrase Catalytic Site and Integrase-RNA interactions

喹啉酮衍生物作为HIV-1整合酶催化位点和整合酶-RNA相互作用的双重抑制剂

Patacchini, Elisa; Madia, Valentina Noemi; Albano, Aurora; Ruggieri, Giuseppe; Messore, Antonella; Ialongo, Davide; Saccoliti, Francesco; Scipione, Luigi; Cosconati, Sandro; Koneru, Pratibha C; Haney, Reed; Kvaratskhelia, Mamuka; Di Santo, Roberto; Costi, Roberta

Discovery of N-substituted-2-oxoindolin benzoylhydrazines as c-MET/SMO modulators in EGFRi-resistant non-small cell lung cancer.

在 EGFRi 耐药的非小细胞肺癌中发现 N-取代-2-氧代吲哚啉苯甲酰肼作为 c-MET/SMO 调节剂

Tomassi Stefano, Natale Benito, Roggia Michele, Amato Luisa, De Rosa Caterina, Della Corte Carminia Maria, Baglini Emma, Amendola Giorgio, Messere Anna, Di Maro Salvatore, Barresi Elisabetta, Da Settimo Federico, Trincavelli Maria Letizia, Ciardiello Fortunato, Taliani Sabrina, Morgillo Floriana, Cosconati Sandro