日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Fluorinated Isoindolinone-Based Glucosylceramide Synthase Inhibitors with Low Human Dose Projections

基于氟化异吲哚啉酮的葡萄糖基神经酰胺合成酶抑制剂的低剂量人体预测

Loughran, H Marie; Schirripa, Kathy M; Roecker, Anthony J; Breslin, Michael J; Tong, Ling; Fillgrove, Kerry L; Kuo, Yuhsin; Bleasby, Kelly; Collier, Hannah; Altman, Michael D; Ford, Melissa C; Newman, Justin A; Drolet, Robert E; Cosden, Mali; Jinn, Sarah; Flick, Rosemarie B; Liu, Xiaomei; Minnick, Christina; Watt, Marla L; Lemaire, Wei; Burlein, Christine; Adam, Gregory C; Austin, Lauren A; Marcus, Jacob N; Smith, Sean M; Fraley, Mark E

Pyrazole Ureas as Low Dose, CNS Penetrant Glucosylceramide Synthase Inhibitors for the Treatment of Parkinson's Disease

吡唑脲类药物作为低剂量、可穿透血脑屏障的中枢神经系统葡糖基神经酰胺合成酶抑制剂,用于治疗帕金森病

Roecker, Anthony J; Schirripa, Kathy M; Loughran, H Marie; Tong, Ling; Liang, Tao; Fillgrove, Kerry L; Kuo, Yuhsin; Bleasby, Kelly; Collier, Hannah; Altman, Michael D; Ford, Melissa C; Drolet, Robert E; Cosden, Mali; Jinn, Sarah; Hatcher, Nathan G; Yao, Lihang; Kandebo, Monika; Vardigan, Joshua D; Flick, Rosemarie B; Liu, Xiaomei; Minnick, Christina; Price, Laura A; Watt, Marla L; Lemaire, Wei; Burlein, Christine; Adam, Gregory C; Austin, Lauren A; Marcus, Jacob N; Smith, Sean M; Fraley, Mark E

Discovery of MK-8768, a Potent and Selective mGluR2 Negative Allosteric Modulator

发现MK-8768,一种强效且选择性的mGluR2负变构调节剂

Rudd, Michael T; Manley, Peter J; Hanney, Barbara; Meng, Zhaoyang; Shu, Youheng; de Leon, Pablo; Frie, Jessica L; Han, Yongxin; Wai, Jenny Miu-Chun; Yang, Zhi-Qiang; Perkins, James J; Hurzy, Danielle M; Manikowski, Jesse J; Zhu, Hong; Bungard, Christopher J; Converso, Antonella; Meissner, Robert S; Cosden, Mali L; Hayashi, Ikuo; Ma, Lei; O'Brien, Julie; Uebele, Victor N; Schachter, Joel B; Bhandari, Neetesh; Ward, Gwendolyn J; Fillgrove, Kerry L; Lu, Bing; Liang, Yuexia; Dubost, David C; Puri, Vanita; Eddins, Donnie M; Vardigan, Joshua D; Drolet, Robert E; Kern, Jonathan T; Uslaner, Jason M

Development of obstetric anesthesia core competencies for USA residency programs through a Delphi process

通过德尔菲法制定美国住院医师培训项目的产科麻醉核心能力

Lilaonitkul, Maytinee; Cosden, Christopher W; Markley, John C; Pian-Smith, May; Lim, Grace; Yeh, Peter; Aleshi, Pedram; Boscardin, Christy; Sullivan, Kristina; George, Ronald B

A novel glucosylceramide synthase inhibitor attenuates alpha synuclein pathology and lysosomal dysfunction in preclinical models of synucleinopathy

一种新型葡萄糖神经酰胺合酶抑制剂可减轻突触核蛋白病临床前模型中的 α 突触核蛋白病理和溶酶体功能障碍

Mali Cosden, Sarah Jinn, Lihang Yao, Cheryl A Gretzula, Monika Kandebo, Dawn Toolan, Nathan G Hatcher, Lei Ma, Wei Lemaire, Gregory C Adam, Christine Burlein, Christina Minnick, Rose Flick, Marla L Watt, James Mulhearn, Mark Fraley, Robert E Drolet, Jacob N Marcus, Sean M Smith

Decreased glucocerebrosidase activity and substrate accumulation of glycosphingolipids in a novel GBA1 D409V knock-in mouse model

新型 GBA1 D409V 敲入小鼠模型中葡萄糖脑苷脂酶活性降低和糖鞘脂底物积累

Nicole K Polinski, Terina N Martinez, Alexander Gorodinsky, Ralph Gareus, Michael Sasner, Mark Herberth, Robert Switzer, Syed O Ahmad, Mali Cosden, Monika Kandebo, Robert E Drolet, Peter D Buckett, Weisong Shan, Yi Chen, Lee J Pellegrino, Gregory D Ellsworth, Leo B Dungan, Warren D Hirst, Sean W Cla

Early intervention of tau pathology prevents behavioral changes in the rTg4510 mouse model of tauopathy

早期干预 tau 病理可预防 rTg4510 小鼠 tau 蛋白病模型中的行为变化

Xiaohai Wang, Karen Smith, Michelle Pearson, Anna Hughes, Mali L Cosden, Jacob Marcus, J Fred Hess, Mary J Savage, Thomas Rosahl, Sean M Smith, Joel B Schachter, Jason M Uslaner

Structural and functional analysis of intra-articular interzone tissue in axolotl salamanders

蝾螈关节内间隙组织的结构和功能分析

R S Cosden-Decker, M M Bickett, C Lattermann, J N MacLeod

Intrinsic repair of full-thickness articular cartilage defects in the axolotl salamander

蝾螈全层关节软骨缺损的内在修复

R S Cosden, C Lattermann, S Romine, J Gao, S R Voss, J N MacLeod