日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Subtype-selective positron emission tomography imaging of poly ADP-ribose polymerase-1 binding in non-human primates, healthy volunteers, and patients with glioblastoma using [11C]AZ14193391

利用[11C]AZ14193391对非人灵长类动物、健康志愿者和胶质母细胞瘤患者进行亚型选择性正电子发射断层扫描成像,以检测聚ADP核糖聚合酶-1的结合情况。

Cselényi, Zsolt; Jucaite, Aurelija; Stragliotto, Giuseppe; Bartek, Jiri; Johnström, Peter; Pike, Andy; Cortés González, Miguel A; Högnäsbacka, Antonia; Dahl, Kenneth; Ghosh, Avipsa; Johannes, Jeffrey W; Staniszewska, Anna D; Leo, Elisabetta; Hamerlik, Petra; Davies, Barry; Cosulich, Sabina; Swales, John; Lawrence, Rachel; Squatrito, Massimo; Mueller, Nancy Kathryn; Khani, Yasir; Sousa, Vasco C; Stenkrona, Per; Halldin, Christer; Farde, Lars; Schou, Magnus

AZ14289671 is a highly selective and blood-brain barrier penetrant irreversible TKI that targets EGFRExon20 insertions.

AZ14289671 是一种高选择性且能穿透血脑屏障的不可逆 TKI,靶向 EGFRExon20 插入

Swaih Aisha M, Talbot Sara, Savoca Adriana, Thorpe Hannah, Flemington Vikki, Phillips Benjamin, Colclough Nicola, McCoull William, Radeva Veronika, Hargreaves David, Packer Martin J, Felisberto-Rodrigues Catarina, Thomson Clare, Orme Jonathan P, Deane Carly, Smith Aaron, Johnström Peter, Schou Magnus, McWilliams Lisa, Davey Paul, Enget Marianne, O'Neill Daniel, Cosulich Sabina, Floc'h Nicolas

Derivation of AZD5335, a Novel FRα-Targeted TOP1i-Loaded ADC, for the Treatment of FRα-Expressing Cancers

AZD5335 的衍生化,一种新型的 FRα 靶向 TOP1i 负载抗体偶联药物 (ADC),用于治疗表达 FRα 的癌症

Zoeller, Jason J; Tammali, Ravinder; Dodd, Roger B; Patel, Neki V; Andoni, Alma; Bisha, Ina; Cronin, Shane; De Almeida, Ana; Lee, Nancy; Meekin, John H 3rd; Tilmont, Isabella; Gasper, Diana; Lan, Lingyun; Cox, Megan; Thomas, Tima; Ward, Christopher; Chesebrough, Jon; Anderton, Judith; Neal, Frances; Zenonos, Zenon; Shandilya, Harini; Chooi, K Phin; Pugh, Kathryn; Saleh, Ali; Wang, Jixin; Mitchell, Pat; Naseer, Humaira; Beaumont, Kevin; Hood, John; Myers, Claire; Christ, Simon; Dino, Iris; Guza, Xhenifer; Falck, Tillmann; Lehmann, Michael; Sargeant, Rebecca; Godfrey, Lisa; Recolin, Benedicte; Brier, Tim; Turner, Simon; Rosfjord, Edward; Fraenkel, Paula G; Cosulich, Sabina; Gymnopoulos, Marco; Hurt, Elaine; Sapra, Puja

Genome-Wide Estrogen Receptor Activity in Breast Cancer

乳腺癌中全基因组雌激素受体活性

Farcas, Anca M; Nagarajan, Sankari; Cosulich, Sabina; Carroll, Jason S

How is the acyl chain composition of phosphoinositides created and does it matter?

磷酸肌醇的酰基链组成是如何形成的?它重要吗?

Barneda, David; Cosulich, Sabina; Stephens, Len; Hawkins, Phillip