Different contributions of chemokine N-terminal features attest to a different ligand binding mode and a bias towards activation of ACKR3/CXCR7 compared with CXCR4 and CXCR3.
趋化因子 N 端特征的不同贡献证明了不同的配体结合模式,并且与 CXCR4 和 CXCR3 相比,ACKR3/CXCR7 更倾向于激活
期刊:British Journal of Pharmacology
影响因子:7.7
doi:10.1111/bph.14132
Szpakowska Martyna, Nevins Amanda M, Meyrath Max, Rhainds David, D'huys Thomas, Guité-Vinet François, Dupuis Nadine, Gauthier Pierre-Arnaud, Counson Manuel, Kleist Andrew, St-Onge Geneviève, Hanson Julien, Schols Dominique, Volkman Brian F, Heveker Nikolaus, Chevigné Andy