日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Inactive structures of the vasopressin V2 receptor reveal distinct binding modes for Tolvaptan and Mambaquaretin toxin.

血管加压素 V2 受体的非活性结构揭示了托伐普坦和曼巴奎汀毒素的不同结合模式

Fouillen Aurélien, Bous Julien, Couvineau Pierre, Orcel Hélène, Mary Charline, Lafleur Lucie, Pierre Timothé, Mendre Christiane, Gilles Nicolas, Schulte Gunnar, Granier Sébastien, Mouillac Bernard

Metabolically stable apelin analogs: development and functional role in water balance and cardiovascular function

代谢稳定的apelin类似物:其在水平衡和心血管功能中的发育和作用

Couvineau, Pierre; Llorens-Cortes, Catherine

Biased activation of the vasopressin V2 receptor probed by molecular dynamics simulations, NMR and pharmacological studies.

通过分子动力学模拟、核磁共振和药理学研究探究加压素 V2 受体的偏向性激活

Fouillen Aurélien, Couvineau Pierre, Gaibelet Gérald, Riché Stéphanie, Orcel Hélène, Mendre Christiane, Kanso Ali, Lanotte Romain, Nguyen Julie, Dimon Juliette, Urbach Serge, Sounier Rémy, Granier Sébastien, Bonnet Dominique, Cong Xiaojing, Mouillac Bernard, Déméné Hélène

Structure, dynamics and transferability of the metal-dependent polyhistidine tetramerization motif TetrHis for single-chain Fv antibodies

金属依赖性多组氨酸四聚体化基序 TetrHis 的结构、动力学和单链 Fv 抗体的转移性

Healey, Robert D; Couillaud, Louise; Hoh, François; Mouhand, Assia; Fouillen, Aurelien; Couvineau, Pierre; Granier, Sébastien; Leyrat, Cédric

Role of the Vasopressin/Apelin Balance and Potential Use of Metabolically Stable Apelin Analogs in Water Metabolism Disorders

血管加压素/阿佩林平衡的作用及代谢稳定的阿佩林类似物在水代谢紊乱中的潜在应用

Flahault, Adrien; Couvineau, Pierre; Alvear-Perez, Rodrigo; Iturrioz, Xavier; Llorens-Cortes, Catherine

Crucial role of the orexin-B C-terminus in the induction of OX1 receptor-mediated apoptosis: analysis by alanine scanning, molecular modelling and site-directed mutagenesis

食欲素B C端在OX1受体介导的细胞凋亡诱导中的关键作用:丙氨酸扫描、分子建模和定点诱变分析

Nicole, Pascal; Couvineau, Pierre; Jamin, Nadege; Voisin, Thierry; Couvineau, Alain