日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

PTRAMP, CSS and Ripr form a conserved complex required for merozoite invasion of Plasmodium species into erythrocytes

PTRAMP、CSS 和 Ripr 形成一个保守的复合物,该复合物是疟原虫裂殖子入侵红细胞所必需的。

Seager, Benjamin A; Lim, Pailene S; Xiao, Xiao; Lai, Keng Heng; Feufack-Donfack, Lionel Brice; Dass, Sheena; Jung, Nicolai C; Abraham, Anju; Grigg, Matthew J; Anstey, Nicholas M; William, Timothy; Sattabongkot, Jetsumon; Leis, Andrew; Longley, Rhea J; Duraisingh, Manoj T; Popovici, Jean; Wilson, Danny W; Cowman, Alan F; Scally, Stephen W

GID/CTLH E3 ligase complex control cell fate programs for sexual development of Plasmodium falciparum

GID/CTLH E3连接酶复合物控制恶性疟原虫有性发育的细胞命运程序

Marapana, Danushka S; Lopaticki, Sash; Balan, Balu; Reaksudsan, Kitsanapong; Cobbold, Simon A; Geoghegan, Niall D; Khurana, Sachin; Scally, Stephen W; Hickey, Peter; Jayakrishnan, Niva; Vaibhav, Vineet; Spall, Sukhdeep; Yousef, Jumana M; Dagley, Laura F; Goodman, Christopher D; Cozijnsen, Anton; McFadden, Geoffrey I; Rogers, Kelly L; Jex, Aaron; Komander, David; McCarthy, James S; Tonkin, Christopher J; Dixon, Matthew W A; Cowman, Alan F

MK-7602: a potent multi-stage dual-targeting antimalarial

MK-7602:一种强效的多阶段双靶点抗疟药

Favuzza, Paola; Palandri, Josephine; de Lera Ruiz, Manuel; Bailey, Wendy; Boyce, Christopher W; Danziger, Andrew; Fawaz, Maria V; Kelly, Michael; Murgolo, Nicholas; Robbins, Jonathan A; Vavrek, Marissa; Zhao, Lianyun; Lei, Zhiyu; Guo, Zhuyan; Reaksudsan, Kitsanapong; Steel, Ryan W J; Hodder, Anthony N; Ngo, Anna; Dziekan, Jerzy M; Thompson, Jennifer K; Triglia, Tony; Birkinshaw, Richard W; Penington, Jocelyn Sietsma; Scally, Stephen W; Dans, Madeline G; Coyle, Rachael; Sevilleno, Nicole; Orban, Agnes; Feufack-Donfack, Lionel Brice; Popovici, Jean; Lee, Marcus C S; Papenfuss, Anthony; Lowes, Kym N; Sleebs, Brad E; McCarthy, James S; McCauley, John A; Boddey, Justin A; Olsen, David B; Cowman, Alan F

First-in-human safety and pharmacokinetics of MK-7602, the antimalarial inhibitor of plasmepsins IX/X, in single- and multiple-ascending-dose studies

MK-7602(一种抗疟疾药物,可抑制疟原虫蛋白酶IX/X)的首次人体安全性和药代动力学研究(单次和多次递增剂量研究)

Stanley, Susan E; Carstens, Russ P; Liberti, Maria V; Eertmans, Ward; Vranckx, Myrthel; Longo, Diane; Ghosal, Nairita; Vavrek, Marissa; Olsen, David B; Cowman, Alan F; Reynders, Tom; Cilissen, Caroline; Laethem, Tine; Rottey, Sylvie; Robbins, Jonathan A; Stoch, S Aubrey; Nussbaum, Jesse

Exploration and Characterization of the Antimalarial Activity of Pyrimidine-2,4-Diamines for which Resistance is Mediated by the ABCI3 Transporter

探索和表征嘧啶-2,4-二胺的抗疟活性及其由ABCI3转运蛋白介导的耐药性

Mansouri, Mahta; Dans, Madeline G; Low, Zijun; Loi, Katie; Jarman, Kate E; Penington, Jocelyn S; Qiu, Deyun; Lehane, Adele M; Crespo, Benigno; Gamo, Franciso-Javier; Baud, Delphine; Brand, Stephen; Jackson, Paul F; Cowman, Alan F; Sleebs, Brad E

CD44 cross-linking promotes Plasmodium falciparum invasion

CD44交联促进恶性疟原虫入侵

Kongsomboonvech, Angel K; Scally, Stephen W; Le Guen, Yann; Valissery, Praveesh; Salinas, Nichole D; Cowman, Alan F; Tolia, Niraj H; Egan, Elizabeth S

Integrated structural biology of the native malarial translation machinery and its inhibition by an antimalarial drug

天然疟原虫翻译机制的整合结构生物学及其被抗疟药物抑制的研究

Anton, Leonie; Cheng, Wenjing; Haile, Meseret T; Dziekan, Jerzy M; Cobb, David W; Zhu, Xiyan; Han, Leyan; Li, Emerson; Nair, Anjali; Lee, Carolyn L; Wang, Hanyu; Ke, Hangjun; Zhang, Guoan; Doud, Emma H; Cowman, Alan F; Ho, Chi-Min

Optimization and Characterization of N-Acetamide Indoles as Antimalarials That Target PfATP4

优化和表征靶向 PfATP4 的 N-乙酰胺吲哚类抗疟药

Awalt, Jon Kyle; Ooi, Zi Kang; Ashton, Trent D; Mansouri, Mahta; Calic, Petar P S; Zhou, Qingmiao; Vasanthan, Santhya; Lee, Serena; Loi, Katie; Jarman, Kate E; Penington, Jocelyn S; Qiu, Deyun; Zhang, Xinxin; Lehane, Adele M; Mao, Emma Y; Gancheva, Maria R; Wilson, Danny W; Giannangelo, Carlo; MacRaild, Christopher A; Creek, Darren J; Yeo, Tomas; Sheth, Tanaya; Fidock, David A; Churchyard, Alisje; Baum, Jake; Famodimu, Mufuliat T; Delves, Michael J; Kristan, Mojca; Stewart, Lindsay; Sutherland, Colin J; Coyle, Rachael; Jagoe, Hannah; Lee, Marcus C S; Chowdury, Mrittika; de Koning-Ward, Tania F; Baud, Delphine; Brand, Stephen; Jackson, Paul F; Cowman, Alan F; Dans, Madeline G; Sleebs, Brad E

Functional characterisation of components in two Plasmodium falciparum Cullin-RING-Ligase complexes.

对两种恶性疟原虫 Cullin-RING-连接酶复合物的组分进行功能表征

Marapana Danushka, Cobbold Simon A, Pasternak Michal, Shami Gerald J, Ralph Stuart A, Lopaticki Sash, Yousef Jumana, Vaibhav Vineet, Dagley Laura F, Komander David, Cowman Alan F

Structure-activity analysis of imino-pyrimidinone-fused pyrrolidines aids the development of dual plasmepsin V and plasmepsin X inhibitors

亚氨基嘧啶酮稠合吡咯烷的结构活性分析有助于开发双重血浆素V和血浆素X抑制剂。

Hodder, Anthony N; Sleebs, Brad E; Adams, Greg; Rezazadeh, Sina; Ngo, Anna; Jarman, Kate; Scally, Stephen; Czabotar, Peter; Wang, Hongwu; McCauley, John A; Olsen, David B; Cowman, Alan F