日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Sodium-glucose co-transporter 2 inhibition improves age-dependent kidney microvascular rarefaction

钠-葡萄糖协同转运蛋白2抑制剂可改善与年龄相关的肾脏微血管稀疏

Paulmann, Anastasia; Cox, Matthew D; Boewer, Tom; Somers, Hannah M; Fuqua, Heath; Seaman, Ryan P; Graber, Joel H; Mahajan, Anchal; Johnson, Cory P; Beverly-Staggs, Laura L; Sandhi, Sonia; Schenk, Heiko; Haller, Hermann

Sexually Dimorphic Response to Dietary Restriction-induced Longevity and Muscle Rejuvenation in Nothobranchius furzeri

饮食限制诱导的寿命延长和肌肉再生对诺氏鲵的性二态性反应

Sandhi, Sonia; Somers, Hannah; Cox, Matthew; Nobrega, Celeste; Seaman, Ryan; Bakers, Elizabeth; Letchner, Olivia; Reeve, Robyn; Menard, Romain; Godwin, James; Paulmann, Anastasia; Rogers, Aric; Valenzano, Dario Riccardo; Graber, Joel; Haller, Hermann; Madelaine, Romain

Discovery and Characterization of a First-in-Class LIV1-TLR7/8 Immunomodulatory Conjugate with Robust Myeloid Activation and Antitumor Activity.

发现并表征了具有强大髓系激活和抗肿瘤活性的首创 LIV1-TLR7/8 免疫调节偶联物

Yamazoe Sayumi, Poudel Yam, Sega Emanuela, Mukhopadhyay Anandaroop, Ramakrishnan Radha, Ukairo Okechukwu, Liu Scot, Akter Rahima, Sadanala Keerthi, Que Kathryn, Cheng Qinqin, Kotapati Srikanth, Deshpande Madhura, Cox Matthew, Chourey Shishir, Gupta Anuradha, Kempson James, Pabbisetty Kumar, Kaspady Mahammed, Bhattasali Debabrata, Yip Shiuhang, Wu Dauh-Rurng, Pookot Deepa, Li Yvonne, Kozhich Alexander, Drexler Dieter, Carl Stephen, Deyanova Ekaterina, Smith Michael, Chan Henry, West Sean, Diong S J, Chang Aram, Florin Lore, Mathur Arvind, Strop Pavel, Zapf Christoph W, Law Deborah, Wilson Nicholas, Broz Miranda, Chekler Eugene P

Structure-Based Design of Novel TLR7/8 Agonist Payloads Enabling an Immunomodulatory Conjugate Approach

基于结构的新型TLR7/8激动剂有效载荷设计,可实现免疫调节偶联物策略

Poudel, Yam B; Lo, Julian C; Norris, Derek J; Cox, Matthew; He, Liqi; Johnson, Walter L; A M Subbaiah, Murugaiah; Mondal, Santigopal; Thangavel, Soodamani; Subramani, Lakshumanan; Reddy, Maheswara; Jain, Suraksha; Weiss, Dahlia R; Sivaprakasam, Prasanna; Critton, David; Mulligan, Dawn; Xie, Chunshan; Dhar, Payal; Li, Yvonne; Sega, Emanuela; Yamazoe, Sayumi; Gavai, Ashvinikumar V; Mathur, Arvind; Zapf, Christoph W; Chekler, Eugene P

SGLT2 Inhibition Ameliorates Age-Dependent Renovascular Rarefaction

SGLT2抑制剂可改善年龄相关性肾血管稀疏

Paulmann, Anastasia; Cox, Matthew D; Boewer, Tom; Somers, Hannah M; Fuqua, Heath; Seaman, Ryan P; Graber, Joel H; Mahajan, Anchal; Johnson, Cory P; Beverly-Staggs, Laura L; Sandhi, Sonia; Schenk, Heiko; Haller, Hermann

Discovery of Novel TLR7 Agonists as Systemic Agent for Combination With aPD1 for Use in Immuno-oncology

发现新型TLR7激动剂作为全身性药物与抗PD-1抗体联合用于免疫肿瘤学

Poudel, Yam B; He, Liqi; Cox, Matthew; Zhang, Qian; Johnson, Walter L; Cong, Qiang; Cheng, Heng; Chowdari, Naidu S; Tarby, Christine; Donnell, Andrew F; Broekema, Matthais; O'Malley, Daniel P; Zhang, Yong; A M Subbaiah, Murugaiah; Kumar, Boda Vijay; Subramani, Lakshumanan; Wang, Bei; Li, Yi-Xin; Sivaprakasam, Prasanna; Critton, David; Mulligan, Dawn; Sandhu, Bhupindar; Xie, Chunshan; Ramakrishnan, Radha; Nagar, Jignesh; Dudhgaonkar, Shailesh; Oderinde, Martins S; Murtaza, Anwar; Schieven, Gary L; Mathur, Arvind; Gavai, Ashvinikumar V; Vite, Gregory; Gangwar, Sanjeev

Identification and Optimization of Small Molecule Pyrazolopyrimidine TLR7 Agonists for Applications in Immuno-oncology

鉴定和优化小分子吡唑并嘧啶类TLR7激动剂在免疫肿瘤学中的应用

He, Liqi; Zhang, Meng Yao; Cox, Matthew; Zhang, Qian; Donnell, Andrew F; Zhang, Yong; Tarby, Christine; Gill, Patrice; Subbaiah, Murugaiah A M; Ramar, Thangeswaran; Reddy, Maheswara; Puttapaka, Vijaya; Li, Yi-Xin; Sivaprakasam, Prasanna; Critton, David; Mulligan, Dawn; Xie, Chunshan; Ramakrishnan, Radha; Nagar, Jignesh; Dudhgaonkar, Shailesh; Murtaza, Anwar; Oderinde, Martins S; Schieven, Gary L; Mathur, Arvind; Gavai, Ashvinikumar V; Vite, Gregory; Gangwar, Sanjeev; Poudel, Yam B

Neuronal CBP-1 is Required for Enhanced Body Muscle Proteostasis in Response to Reduced Translation Downstream of mTOR

神经元CBP-1对于mTOR下游翻译减少时增强身体肌肉蛋白质稳态是必需的。

Snow, Santina; Ahmad Mir, Dilawar; Ma, Zhengxin; Horrocks, Jordan; Cox, Matthew; Ruzga, Marissa; Sayed, Hussein; Rogers, Aric N

Durability of the moderate-to-heavy-intensity transition is related to the effects of prolonged exercise on severe-intensity performance

中强度到重强度转换的持久性与长时间锻炼对高强度运动表现的影响有关

Kate Hamilton, Andrew E Kilding, Daniel J Plews, Mathew J Mildenhall, Mark Waldron, Thanchanok Charoensap, Tobias H Cox, Matthew J Brick, Warren B Leigh, Ed Maunder

Successful kinetic impact into an asteroid for planetary defence

利用动能撞击成功攻击小行星,用于行星防御

Daly, R Terik; Ernst, Carolyn M; Barnouin, Olivier S; Chabot, Nancy L; Rivkin, Andrew S; Cheng, Andrew F; Adams, Elena Y; Agrusa, Harrison F; Abel, Elisabeth D; Alford, Amy L; Asphaug, Erik I; Atchison, Justin A; Badger, Andrew R; Baki, Paul; Ballouz, Ronald-L; Bekker, Dmitriy L; Bellerose, Julie; Bhaskaran, Shyam; Buratti, Bonnie J; Cambioni, Saverio; Chen, Michelle H; Chesley, Steven R; Chiu, George; Collins, Gareth S; Cox, Matthew W; DeCoster, Mallory E; Ericksen, Peter S; Espiritu, Raymond C; Faber, Alan S; Farnham, Tony L; Ferrari, Fabio; Fletcher, Zachary J; Gaskell, Robert W; Graninger, Dawn M; Haque, Musad A; Harrington-Duff, Patricia A; Hefter, Sarah; Herreros, Isabel; Hirabayashi, Masatoshi; Huang, Philip M; Hsieh, Syau-Yun W; Jacobson, Seth A; Jenkins, Stephen N; Jensenius, Mark A; John, Jeremy W; Jutzi, Martin; Kohout, Tomas; Krueger, Timothy O; Laipert, Frank E; Lopez, Norberto R; Luther, Robert; Lucchetti, Alice; Mages, Declan M; Marchi, Simone; Martin, Anna C; McQuaide, Maria E; Michel, Patrick; Moskovitz, Nicholas A; Murphy, Ian W; Murdoch, Naomi; Naidu, Shantanu P; Nair, Hari; Nolan, Michael C; Ormö, Jens; Pajola, Maurizio; Palmer, Eric E; Peachey, James M; Pravec, Petr; Raducan, Sabina D; Ramesh, K T; Ramirez, Joshua R; Reynolds, Edward L; Richman, Joshua E; Robin, Colas Q; Rodriguez, Luis M; Roufberg, Lew M; Rush, Brian P; Sawyer, Carolyn A; Scheeres, Daniel J; Scheirich, Petr; Schwartz, Stephen R; Shannon, Matthew P; Shapiro, Brett N; Shearer, Caitlin E; Smith, Evan J; Steele, R Joshua; Steckloff, Jordan K; Stickle, Angela M; Sunshine, Jessica M; Superfin, Emil A; Tarzi, Zahi B; Thomas, Cristina A; Thomas, Justin R; Trigo-Rodríguez, Josep M; Tropf, B Teresa; Vaughan, Andrew T; Velez, Dianna; Waller, C Dany; Wilson, Daniel S; Wortman, Kristin A; Zhang, Yun