日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Indole-3-propionic acid links gut dysfunction to diabetic retinopathy: a biomarker and novel therapeutic approach

吲哚-3-丙酸将肠道功能障碍与糖尿病视网膜病变联系起来:一种生物标志物和一种新的治疗方法

Prasad, Ram; Adu-Rutledge, Yvonne; Ziani, Borhane; Floyd, Jason L; Ready, Edgar L; Paul, Sarbodeep; Sheini, Fadeela; Sharma, Rati; Rosencrans, Robert F; Li Calzi, Sergio; Sielski, Micheli Severo; Medawar, Nicholas G; Dutta, Roshan; Johnson, Emory Brennis; Qi, Xiaoping; Bansal, Mohit; Lamendella, Regina; Wright, Justin R; Verma, Suresh Kumar; Boulton, Michael E; Stevens, Bruce R; Vander Kooi, Craig W; Sun, Ramon C; Oudit, Gavin Y; Li, Qiuhong; Grant, Maria B

Drug Repurposing: Conversion of the Peripherally Restricted HIV Protease Inhibitor Amprenavir to Potent, Selective, and CNS-Penetrant Agonists for the Cannabinoid Receptor 2

药物再利用:将外周限制性 HIV 蛋白酶抑制剂安普那韦转化为强效、选择性强且能穿透血脑屏障的大麻素受体 2 激动剂

Haymer, Daniel H; Duncan, Renn A; Rodriguez, Alice L; Han, Allie; Lindsay, Richard J; Wijesiri, N Kithmini; Thompson Gray, Analisa; Krishnan, Srinivasan; Qi, Aidong; Brown, Benjamin P; Boutaud, Olivier; Engers, Darren W; Jones, Carrie K; Niswender, Colleen M; Lindsley, Craig W; Bender, Aaron M

Monkeypox Virus Antibodies in Healthy Persons after Vaccination with MVA-BN, United Kingdom

英国健康人群接种MVA-BN疫苗后猴痘病毒抗体的研究

Sheridan, Victoria H; Duffy, Craig W; Dunning, Jake; Turtle, Lance; Hiscox, Julian A; Subramaniam, Krishanthi S

Mapping glycogen accumulation and treatment effect in Pompe disease with saturation transfer MRI

利用饱和转移磁共振成像技术绘制庞贝病中糖原积累及治疗效果图

Zeng, Qing; Li, Yuguo; Timm, Derek; Johnson, Tyler; Mehta, Nickita; Martin, Lukas; Fox, Brian; van Zijl, Peter C M; Walter, Glenn A; Rosenberg, Jens T; Kooi, Craig W Vander; Corti, Manuela; Gentry, Matthew S; Sun, Ramon C; Byrne, Barry J; Yadav, Nirbhay N

The relative contribution of modifiable and non-modifiable factors for determining cognition in mid-life individuals at risk for late-life Alzheimer's disease

可改变因素和不可改变因素对中年人认知能力的影响(这些人群有患晚年阿尔茨海默病的风险)

Cao, Bolin; Qi, Qing; Hutchinson, Siobhan; Ferguson, Damien; Malhotra, Paresh; Koychev, Ivan; O'Brien, John T; Bridgeman, Katie; Ritchie, Craig W; Lawlor, Brian; Naci, Lorina

Discovery of VU6025733 (AG06827): A Highly Selective, Orally Bioavailable, and Structurally Distinct M(4) Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM) with Robust In Vivo Efficacy

VU6025733 (AG06827) 的发现:一种高选择性、口服生物利用度高、结构独特的 M(4) 毒蕈碱乙酰胆碱受体正向变构调节剂 (PAM),具有强大的体内疗效

Gregro, Alison R; Park, Charlotte; Long, Madeline F; Baker, Logan A; Bollinger, Katrina A; Ringuette, Anna E; Peng, Li; Luscombe, Vincent B; Billard, Natasha B; Rodriguez, Alice L; Niswender, Colleen M; Peng, Weimin; Dickerson, Jonathan W; Rook, Jerri M; O'Neill, Jordan; Chang, Sichen; Boonen, Harrie C M; Jensen, Thomas; Thomsen, Morten S; Bridges, Thomas M; Boutaud, Olivier; Conn, P Jeffrey; Engers, Darren W; Lindsley, Craig W; Temple, Kayla J

Discovery of 7-(Pyridin-3-yl)thieno[3,2-b]pyridine-5-carboxamides as Negative Allosteric Modulators of Metabotropic Glutamate Receptor Subtype 5

发现 7-(吡啶-3-基)噻吩并[3,2-b]吡啶-5-甲酰胺类化合物作为代谢型谷氨酸受体5亚型的负变构调节剂

Henderson, Scott H; Ringuette, Anna E; Whomble, David L; Capstick, Rory A; Richardson, Alexa E; Maurer, Mallory A; Billard, Natasha B; Lei, Xia; Wilkinson, Joshua C; Kethanapalli, Sri H; Cho, Hyekyung P; Rodriguez, Alice L; Niswender, Colleen M; Peng, Weimin; Rook, Jerri M; Chang, Sichen; Blobaum, Anna L; Boutaud, Olivier; Felts, Andrew S; Conn, P Jeffrey; Lindsley, Craig W; Temple, Kayla J

The biochemical dynamics of the glycogen phosphatase laforin directly impact brain metabolism

糖原磷酸酶拉福林的生化动力学直接影响脑代谢

Brewer, M Kathryn; Donohue, Katherine J; Singh, Pankaj K; Raththagala, Madushi; Simmons, Zoe R; Wayne, Jeremiah L; Li, Sheng; Viana, Rosa; Segvich, Dyann M; Contreras, Christopher J; Cantrell, Alex R; Sanz, Pascual; Sun, Ramon C; Vander Kooi, Craig W; Roach, Peter J; DePaoli-Roach, Anna; Gentry, Matthew S

Discovery of VU6083859, a TAOK1 Selective Inhibitor, and VU6080195, a pan-TAOK Activator

发现 VU6083859(一种 TAOK1 选择性抑制剂)和 VU6080195(一种泛 TAOK 激活剂)

Schultz, Daniel C; Parr, Lauren C; Sweet, Hunter; Lamb, Sean; Engers, Julie L; Napier, Nathaniel C; McKinnie, Hallie G; Whomble, David; Kramlinger, Valerie; Boutaud, Olivier; Lindsley, Craig W

Associations between gut microbiota and personality traits: insights from a captive common marmoset (Callithrix jacchus) colony

肠道菌群与人格特质之间的关联:来自圈养普通狨猴(Callithrix jacchus)群体的启示

Ye, Huimin; Šlipogor, Vedrana; Hanson, Buck T; Séneca, Joana; Hausmann, Bela; Herbold, Craig W; Pjevac, Petra; Bugnyar, Thomas; Loy, Alexander