日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Computational Design of Cyclic Peptide Inhibitors of a Bacterial Membrane Lipoprotein Peptidase

细菌膜脂蛋白肽酶环肽抑制剂的计算设计

Craven, Timothy W; Nolan, Mark D; Bailey, Jonathan; Olatunji, Samir; Bann, Samantha J; Bowen, Katherine; Ostrovitsa, Nikita; Da Costa, Thaina M; Ballantine, Ross D; Weichert, Dietmar; Levine, Paul M; Stewart, Lance J; Bhardwaj, Gaurav; Geoghegan, Joan A; Cochrane, Stephen A; Scanlan, Eoin M; Caffrey, Martin; Baker, David

Generation of Potent and Stable GLP-1 Analogues Via "Serine Ligation"

通过“丝氨酸连接”生成高效稳定的GLP-1类似物

Levine, Paul M; Craven, Timothy W; Li, Xinting; Balana, Aaron T; Bird, Gregory H; Godes, Marina; Salveson, Patrick J; Erickson, Patrick W; Lamb, Mila; Ahlrichs, Maggie; Murphy, Michael; Ogohara, Cassandra; Said, Meerit Y; Walensky, Loren D; Pratt, Matthew R; Baker, David

Anchor extension: a structure-guided approach to design cyclic peptides targeting enzyme active sites

锚定延伸:一种以结构为导向的环肽设计方法,靶向酶活性位点

Hosseinzadeh, Parisa; Watson, Paris R; Craven, Timothy W; Li, Xinting; Rettie, Stephen; Pardo-Avila, Fátima; Bera, Asim K; Mulligan, Vikram Khipple; Lu, Peilong; Ford, Alexander S; Weitzner, Brian D; Stewart, Lance J; Moyer, Adam P; Di Piazza, Maddalena; Whalen, Joshua G; Greisen, Per Jr; Christianson, David W; Baker, David

Isolating Conformers to Assess Dynamics of Peptidic Catalysts Using Computationally Designed Macrocyclic Peptides

利用计算机设计的环状肽分离构象异构体以评估肽催化剂的动力学

Stone, Elizabeth A; Hosseinzadeh, Parisa; Craven, Timothy W; Robertson, Michael J; Han, Yaodong; Hsieh, Sheng-Ying; Metrano, Anthony J; Baker, David; Miller, Scott J

Design of Peptoid-peptide Macrocycles to Inhibit the β-catenin TCF Interaction in Prostate Cancer.

设计肽类肽大环化合物以抑制前列腺癌中的β-catenin TCF相互作用

Schneider Jeffrey A, Craven Timothy W, Kasper Amanda C, Yun Chi, Haugbro Michael, Briggs Erica M, Svetlov Vladimir, Nudler Evgeny, Knaut Holger, Bonneau Richard, Garabedian Michael J, Kirshenbaum Kent, Logan Susan K

Comprehensive computational design of ordered peptide macrocycles

有序肽大环的综合计算设计

Hosseinzadeh, Parisa; Bhardwaj, Gaurav; Mulligan, Vikram Khipple; Shortridge, Matthew D; Craven, Timothy W; Pardo-Avila, Fátima; Rettie, Stephen A; Kim, David E; Silva, Daniel-Adriano; Ibrahim, Yehia M; Webb, Ian K; Cort, John R; Adkins, Joshua N; Varani, Gabriele; Baker, David

Adding diverse noncanonical backbones to rosetta: enabling peptidomimetic design

为 Rosetta 添加多种非典型骨架:实现肽模拟设计

Drew, Kevin; Renfrew, P Douglas; Craven, Timothy W; Butterfoss, Glenn L; Chou, Fang-Chieh; Lyskov, Sergey; Bullock, Brooke N; Watkins, Andrew; Labonte, Jason W; Pacella, Michael; Kilambi, Krishna Praneeth; Leaver-Fay, Andrew; Kuhlman, Brian; Gray, Jeffrey J; Bradley, Philip; Kirshenbaum, Kent; Arora, Paramjit S; Das, Rhiju; Bonneau, Richard