日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Phenolic Profile and Bioactive Prospects of Wild Annona Species From Angola

安哥拉野生番荔枝属植物的酚类成分及生物活性前景

Rangel, Josefa; Liberal, Ângela; Finimundy, Tiane C; Pires, Tânia S P; Cravo, Pedro; Conceição Silva, Maria; Cassiano, Gustavo Capatti; Barros, Lillian; Romeiras, Maria M; Fernandes, Ângela

Evaluation of the Activity of 4‑Quinolones against Multi-Life Stages of Plasmodium spp

评价4-喹诺酮类药物对疟原虫多个生命阶段的活性

Annunciato, Yasmin; da Silva, Everton M; Araújo, Jéssica E; Martinez, Leandro do N; Santana, Sofia; Workneh, Eyob A; S Alvarez, Luís C; Magalhães, Marcela L; Andrade, Alice Oliveira; da Costa, Wallyson de J; Campolina, Guilherme; Nascimento Santana, Matheus; Barbosa, Camila S; Peres, Erica P M L; Moura, Caio S; Dos Santos, Najara A C; Bastos, Alessandra da S; Barros, Roberto Rudge de M; Gazarini, Marcos L; Medeiros, Jansen Fernandes; Teles, Carolina B G; Costa, Fabio T M; Alves, Ana C; Pereira, Dhelio B; Pinto, João; Cravo, Pedro V L; Guido, Rafael Victorio Carvalho; Prudêncio, Miguel; Araujo, Maisa da S; Corrêa, Arlene G; Cassiano, Gustavo C; Aguiar, Anna C C

A novel 4-aminoquinoline chemotype with multistage antimalarial activity and lack of cross-resistance with PfCRT and PfMDR1 mutants

一种新型的4-氨基喹啉化学类型,具有多阶段抗疟活性,且与PfCRT和PfMDR1突变体无交叉耐药性。

Ferreira, Letícia Tiburcio; Cassiano, Gustavo Capatti; Alvarez, Luis Carlos Salazar; Okombo, John; Calit, Juliana; Fontinha, Diana; Gil-Iturbe, Eva; Coyle, Rachael; Andrade, Carolina Horta; Sunnerhagen, Per; Bargieri, Daniel Youssef; Prudêncio, Miguel; Quick, Matthias; Cravo, Pedro V; Lee, Marcus C S; Fidock, David A; Costa, Fabio Trindade Maranhão

Whole genome sequencing identifies novel mutations in malaria parasites resistant to artesunate (ATN) and to ATN + mefloquine combination

全基因组测序鉴定出对青蒿琥酯 (ATN) 和 ATN + 甲氟喹联合疗法产生耐药性的疟原虫的新突变。

Cassiano, Gustavo Capatti; Martinelli, Axel; Mottin, Melina; Neves, Bruno Junior; Andrade, Carolina Horta; Ferreira, Pedro Eduardo; Cravo, Pedro

Mutation in the 26S proteasome regulatory subunit rpn2 gene in Plasmodium falciparum confers resistance to artemisinin

恶性疟原虫26S蛋白酶体调节亚基rpn2基因的突变赋予其对青蒿素的耐药性

Gonçalves, Adriana F; Lima-Pinheiro, Ana; Teixeira, Miguel; Cassiano, Gustavo Capatti; Cravo, Pedro; Ferreira, Pedro E

Innovative Multistage ML-QSAR Models for Malaria: From Data to Discovery

疟疾创新型多阶段机器学习-定量构效关系模型:从数据到发现

Borba, Joyce V B; Salazar-Alvarez, Luis Carlos; Ferreira, Letícia Tiburcio; Silva-Mendonça, Sabrina; Silva, Meryck Felipe Brito da; Sanches, Igor H; Clementino, Leandro da Costa; Magalhães, Marcela Lucas; Rimoldi, Aline; Calit, Juliana; Santana, Sofia; Prudêncio, Miguel; Cravo, Pedro V; Bargieri, Daniel Y; Cassiano, Gustavo C; Costa, Fabio T M; Andrade, Carolina Horta

Antimalarial and Cytotoxic Activity of Native Plants Used in Cabo Verde Traditional Medicine

佛得角传统医学中使用的本土植物的抗疟疾和细胞毒活性

Essoh, Anyse P; Cassiano, Gustavo Capatti; Mandim, Filipa; Barros, Lillian; Gomes, Isildo; Medeiros, Márcia Melo; Moura, Mónica; Cravo, Pedro Vitor Lemos; Romeiras, Maria M

Computational Chemogenomics Drug Repositioning Strategy Enables the Discovery of Epirubicin as a New Repurposed Hit for Plasmodium falciparum and P. vivax

计算化学基因组学药物重定位策略促成了表柔比星作为一种新的可用于治疗恶性疟原虫和间日疟原虫的先导化合物的发现

Ferreira, Letícia Tiburcio; Rodrigues, Juliana; Cassiano, Gustavo Capatti; Tavella, Tatyana Almeida; Tomaz, Kaira Cristina Peralis; Baia-da-Silva, Djane Clarys; Souza, Macejane Ferreira; Lima, Marilia Nunes do Nascimento; Mottin, Melina; Almeida, Ludimila Dias; Calit, Juliana; Puça, Maria Carolina Silva de Barros; Melo, Gisely Cardoso; Bargieri, Daniel Youssef; Lopes, Stefanie Costa Pinto; Lacerda, Marcus Vinicius Guimarães; Bilsland, Elizabeth; Sunnerhagen, Per; Neves, Bruno Junior; Andrade, Carolina Horta; Cravo, Pedro Vitor Lemos; Costa, Fabio Trindade Maranhão

Correction for Ferreira et al., "Computational Chemogenomics Drug Repositioning Strategy Enables the Discovery of Epirubicin as a New Repurposed Hit for Plasmodium falciparum and P. vivax"

对 Ferreira 等人的论文“计算化学基因组学药物重定位策略促成了表柔比星作为恶性疟原虫和间日疟原虫新用途先导化合物的发现”的更正

Ferreira, Letícia Tiburcio; Rodrigues, Juliana; Cassiano, Gustavo Capatti; Tavella, Tatyana Almeida; Tomaz, Kaira Cristina Peralis; Baia-da-Silva, Djane Clarys; Souza, Macejane Ferreira; Lima, Marilia Nunes do Nascimento; Mottin, Melina; Almeida, Ludimila Dias; Calit, Juliana; Puça, Maria Carolina Silva de Barros; Melo, Gisely Cardoso; Bargieri, Daniel Youssef; Lopes, Stefanie Costa Pinto; Lacerda, Marcus Vinicius Guimarães; Bilsland, Elizabeth; Sunnerhagen, Per; Neves, Bruno Junior; Andrade, Carolina Horta; Cravo, Pedro Vitor Lemos; Costa, Fabio Trindade Maranhão

QSAR-Driven Design and Discovery of Novel Compounds With Antiplasmodial and Transmission Blocking Activities

基于QSAR的抗疟疾和阻断传播活性新型化合物的设计与发现

Lima, Marilia N N; Melo-Filho, Cleber C; Cassiano, Gustavo C; Neves, Bruno J; Alves, Vinicius M; Braga, Rodolpho C; Cravo, Pedro V L; Muratov, Eugene N; Calit, Juliana; Bargieri, Daniel Y; Costa, Fabio T M; Andrade, Carolina H