日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Identification of potent and reversible piperidine carboxamides that are species-selective orally active proteasome inhibitors to treat malaria.

鉴定出强效且可逆的哌啶甲酰胺类化合物,它们是具有物种选择性的口服活性蛋白酶体抑制剂,可用于治疗疟疾

Lawong Aloysus, Gahalawat Suraksha, Ray Sneha, Ho Nhi, Han Yan, Ward Kurt E, Deng Xiaoyi, Chen Zhe, Kumar Ashwani, Xing Chao, Hosangadi Varun, Fairhurst Kate J, Tashiro Kyuto, Liszczak Glen, Shackleford David M, Katneni Kasiram, Chen Gong, Saunders Jessica, Crighton Elly, Casas Arturo, Robinson Joshua J, Imlay Leah S, Zhang Xiaoyu, Lemoff Andrew, Zhao Zhiyu, Angulo-Barturen Iñigo, Jiménez-Díaz María Belén, Wittlin Sergio, Campbell Simon F, Fidock David A, Laleu Benoît, Charman Susan A, Ready Joseph M, Phillips Margaret A

DNDI-6174 is a preclinical candidate for visceral leishmaniasis that targets the cytochrome bc(1)

DNDI-6174 是一种用于治疗内脏利什曼病的临床前候选药物,其靶点为细胞色素 bc(1)

Braillard, Stéphanie; Keenan, Martine; Breese, Karen J; Heppell, Jacob; Abbott, Michael; Islam, Rafiqul; Shackleford, David M; Katneni, Kasiram; Crighton, Elly; Chen, Gong; Patil, Rahul; Lee, Given; White, Karen L; Carvalho, Sandra; Wall, Richard J; Chemi, Giulia; Zuccotto, Fabio; González, Silvia; Marco, Maria; Deakyne, Julianna; Standing, David; Brunori, Gino; Lyon, Jonathan J; Castañeda-Casado, Pablo; Camino, Isabel; Martinez Martinez, Maria S; Zulfiqar, Bilal; Avery, Vicky M; Feijens, Pim-Bart; Van Pelt, Natascha; Matheeussen, An; Hendrickx, Sarah; Maes, Louis; Caljon, Guy; Yardley, Vanessa; Wyllie, Susan; Charman, Susan A; Chatelain, Eric

Lead Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series for the Treatment of Malaria.

吡咯基二氢乳清酸脱氢酶抑制剂系列先导化合物的优化及其在疟疾治疗中的应用

Kokkonda Sreekanth, Deng Xiaoyi, White Karen L, El Mazouni Farah, White John, Shackleford David M, Katneni Kasiram, Chiu Francis C K, Barker Helena, McLaren Jenna, Crighton Elly, Chen Gong, Angulo-Barturen Inigo, Jimenez-Diaz Maria Belen, Ferrer Santiago, Huertas-Valentin Leticia, Martinez-Martinez Maria Santos, Lafuente-Monasterio Maria Jose, Chittimalla Rajesh, Shahi Shatrughan P, Wittlin Sergio, Waterson David, Burrows Jeremy N, Matthews Dave, Tomchick Diana, Rathod Pradipsinh K, Palmer Michael J, Charman Susan A, Phillips Margaret A