日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Prey for the Proteasome: Targeted Protein Degradation-A Medicinal Chemist's Perspective

蛋白酶体的猎物:靶向蛋白质降解——药物化学家的视角

Luh, Laura M; Scheib, Ulrike; Juenemann, Katrin; Wortmann, Lars; Brands, Michael; Cromm, Philipp M

Lipidated Stapled Peptides Targeting the Acyl Binding Protein UNC119

靶向酰基结合蛋白UNC119的脂化交联肽

Cromm, Philipp M; Adihou, Hélène; Kapoor, Shobhna; Vazquez-Chantada, Mercedes; Davey, Paul; Longmire, David; Hennes, Elisabeth; Hofer, Walter; Küchler, Philipp; Chiarparin, Elisabetta; Waldmann, Herbert; Grossmann, Tom N

Development of Novel Melanocortin Receptor Agonists Based on the Cyclic Peptide Framework of Sunflower Trypsin Inhibitor-1.

基于向日葵胰蛋白酶抑制剂-1的环肽骨架开发新型黑皮质素受体激动剂

Durek Thomas, Cromm Philipp M, White Andrew M, Schroeder Christina I, Kaas Quentin, Weidmann Joachim, Ahmad Fuaad Abdullah, Cheneval Olivier, Harvey Peta J, Daly Norelle L, Zhou Yang, Dellsén Anita, Österlund Torben, Larsson Niklas, Knerr Laurent, Bauer Udo, Kessler Horst, Cai Minying, Hruby Victor J, Plowright Alleyn T, Craik David J

The Proteasome in Modern Drug Discovery: Second Life of a Highly Valuable Drug Target

蛋白酶体在现代药物发现中的作用:高价值药物靶点的第二次生命

Cromm, Philipp M; Crews, Craig M

Targeted Protein Degradation: from Chemical Biology to Drug Discovery

靶向蛋白质降解:从化学生物学到药物发现

Cromm, Philipp M; Crews, Craig M

Constraining an Irregular Peptide Secondary Structure through Ring-Closing Alkyne Metathesis

通过闭环炔烃复分解反应限制不规则肽的二级结构

Cromm, Philipp M; Wallraven, Kerstin; Glas, Adrian; Bier, David; Fürstner, Alois; Ottmann, Christian; Grossmann, Tom N