日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Design, Synthesis, and Evaluation of Novel Inhibitors of Aminoglycoside-Resistance 16S Ribosomal RNA Methyltransferases

新型氨基糖苷类抗性16S核糖体RNA甲基转移酶抑制剂的设计、合成与评价

Deprez, Benjamin E; Dey, Debayan; Zelinskaya, Natalia; Csatary, Erika E; Yang, Qimin Winnie; Nie, Minhua; Conn, Graeme L; Wuest, William M

nTZDpa (non-thiazolidinedione PPARγ partial agonist) derivatives retain antimicrobial activity without improving renal toxicity

nTZDpa(非噻唑烷二酮类PPARγ部分激动剂)衍生物保留了抗菌活性,且不增加肾毒性。

Dekarske, Madeline M; Felix, Lewis Oscar; Ortiz, Carlos Monteagudo; Csatary, Erika E; Mylonakis, Elefterios; Wuest, William M

The histone-like protein AlgP regulon is distinct in mucoid and nonmucoid Pseudomonas aeruginosa and does not include alginate biosynthesis genes

组蛋白样蛋白AlgP调控子在黏液型和非黏液型铜绿假单胞菌中存在差异,且不包含藻酸盐生物合成基因。

Cross, Ashley R; Csatary, Erika E; Raghuram, Vishnu; Diggle, Frances L; Whiteley, Marvin; Wuest, William M; Goldberg, Joanna B

The Natural Product Elegaphenone Potentiates Antibiotic Effects against Pseudomonas aeruginosa

天然产物依拉菲酮增强了抗生素对铜绿假单胞菌的作用

Zhao, Weining; Cross, Ashley R; Crowe-McAuliffe, Caillan; Weigert-Munoz, Angela; Csatary, Erika E; Solinski, Amy E; Krysiak, Joanna; Goldberg, Joanna B; Wilson, Daniel N; Medina, Eva; Wuest, William M; Sieber, Stephan A

A selective membrane-targeting repurposed antibiotic with activity against persistent methicillin-resistant Staphylococcus aureus

一种选择性靶向膜的再利用抗生素,对持续耐甲氧西林金黄色葡萄球菌具有活性

Kim, Wooseong; Zou, Guijin; Hari, Taylor P A; Wilt, Ingrid K; Zhu, Wenpeng; Galle, Nicolas; Faizi, Hammad A; Hendricks, Gabriel L; Tori, Katerina; Pan, Wen; Huang, Xiaowen; Steele, Andrew D; Csatary, Erika E; Dekarske, Madeline M; Rosen, Jake L; Ribeiro, Noelly de Queiroz; Lee, Kiho; Port, Jenna; Fuchs, Beth Burgwyn; Vlahovska, Petia M; Wuest, William M; Gao, Huajian; Ausubel, Frederick M; Mylonakis, Eleftherios

Discovery and Optimization of nTZDpa as an Antibiotic Effective Against Bacterial Persisters

发现和优化 nTZDpa 作为一种对细菌持续感染有效的抗生素

Kim, Wooseong; Steele, Andrew D; Zhu, Wenpeng; Csatary, Erika E; Fricke, Nico; Dekarske, Madeline M; Jayamani, Elamparithi; Pan, Wen; Kwon, Bumsup; Sinitsa, Isabelle F; Rosen, Jake L; Conery, Annie L; Fuchs, Beth Burgwyn; Vlahovska, Petia M; Ausubel, Frederick M; Gao, Huajian; Wuest, William M; Mylonakis, Eleftherios