日期:
2020 年 — 2026 年
2020
2021
2022
2023
2024
2025
2026
影响因子:

Discovery of a Series of Pyrazinone RORγ Antagonists and Identification of the Clinical Candidate BI 730357

发现一系列吡嗪酮类RORγ拮抗剂并鉴定临床候选药物BI 730357

Harcken, Christian; Csengery, Johanna; Turner, Michael; Wu, Lifen; Liang, Shuang; Sibley, Robert; Brunette, Steven; Labadia, Mark; Hoyt, Kathleen; Wayne, Anita; Wieckowski, Thomas; Davis, Gregg; Panzenbeck, Mark; Souza, Donald; Kugler, Stanley; Terenzio, Donna; Collin, Delphine; Smith, Dustin; Fryer, Ryan M; Tseng, Yin-Chao; Hehn, Jörg P; Fletcher, Kim; Hughes, Robert O

Tumor-selective, antigen-independent delivery of a pH sensitive peptide-topoisomerase inhibitor conjugate suppresses tumor growth without systemic toxicity

肿瘤选择性、抗原非依赖性递送 pH 敏感肽拓扑异构酶抑制剂缀合物可抑制肿瘤生长且无全身毒性

Sophia Gayle, Robert Aiello, Nalin Leelatian, Jason M Beckta, Jane Bechtold, Patricia Bourassa, Johanna Csengery, Robert J Maguire, Dan Marshall, Ranjini K Sundaram, Jinny Van Doorn, Kelli Jones, Hunter Moore, Lori Lopresti-Morrow, Timothy Paradis, Laurie Tylaska, Qing Zhang, Hannah Visca, Yana K Re

Correction to 'Tumor-selective, antigen-independent delivery of a pH sensitive peptide-topoisomerase inhibitor conjugate suppresses tumor growth without systemic toxicity'

更正“肿瘤选择性、抗原非依赖性递送pH敏感肽-拓扑异构酶抑制剂偶联物可抑制肿瘤生长且无全身毒性”

Gayle, Sophia; Aiello, Robert; Leelatian, Nalin; Beckta, Jason M; Bechtold, Jane; Bourassa, Patricia; Csengery, Johanna; Maguire, Robert J; Marshall, Dan; Sundaram, Ranjini K; Van Doorn, Jinny; Jones, Kelli; Moore, Hunter; Lopresti-Morrow, Lori; Paradis, Timothy; Tylaska, Laurie; Zhang, Qing; Visca, Hannah; Reshetnyak, Yana K; Andreev, Oleg A; Engelman, Donald M; Glazer, Peter M; Bindra, Ranjit S; Paralkar, Vishwas M