Discovery of a Series of Pyrazinone RORγ Antagonists and Identification of the Clinical Candidate BI 730357
发现一系列吡嗪酮类RORγ拮抗剂并鉴定临床候选药物BI 730357
期刊:ACS Medicinal Chemistry Letters
影响因子:4
doi:10.1021/acsmedchemlett.0c00575
Harcken, Christian; Csengery, Johanna; Turner, Michael; Wu, Lifen; Liang, Shuang; Sibley, Robert; Brunette, Steven; Labadia, Mark; Hoyt, Kathleen; Wayne, Anita; Wieckowski, Thomas; Davis, Gregg; Panzenbeck, Mark; Souza, Donald; Kugler, Stanley; Terenzio, Donna; Collin, Delphine; Smith, Dustin; Fryer, Ryan M; Tseng, Yin-Chao; Hehn, Jörg P; Fletcher, Kim; Hughes, Robert O